Preparation of α-silyl- or α,α-bis(silyl)-substituted alkylcopper reagents and their synthetic use Fulltext Access 9 Pages 2005
An improved Ullmann-Ukita-Buchwald-Li conditions for CuI-catalyzed coupling reaction of 2-pyridones with aryl halides Fulltext Access 9 Pages 2005
Bellisosides A-F, six novel acylated triterpenoid saponins from Bellis perennis (compositae) Fulltext Access 9 Pages 2005
Synthesis of 2-aryl-4-chloropyrroles via ring expansion of 2-aryl-1-chlorocyclopropanecarbaldehydes Fulltext Access 9 Pages 2005
Synthesis of functionalized m-bistrifluoromethylbenzenes via cyclocondensation of 1,1,1,5,5,5-hexafluoroacetylacetone with enamines Fulltext Access 9 Pages 2005
The reaction between 3-aminocrotonates and oxindole-3-ylidene derivatives: synthesis of highly substituted pyrroles Fulltext Access 9 Pages 2005
Synthesis of isomerically pure carboxylate- and sulfonate-substituted xanthene fluorophores Fulltext Access 9 Pages 2005
Oligothienylenevinylenes incorporating 3,4-ethylenedioxythiophene (EDOT) units Fulltext Access 9 Pages 2005
A new one-pot synthesis of α-Gal epitope derivatives involved in the hyperacute rejection response in xenotransplantation Fulltext Access 9 Pages 2005
The site-selective functionalization of halogen-bearing phenols: an exercise in diversity-oriented organometallic synthesis Fulltext Access 9 Pages 2005
Pyridino-directed lithiation of anisylpyridines: new access to functional pyridylphenols Fulltext Access 9 Pages 2005
Can relief of ring-strain in a cyclopropylmethyllithium drive the Brook rearrangement? Fulltext Access 9 Pages 2005
Synthesis of cordiaquinone J and K via B-alkyl Suzuki-Miyaura coupling as a key step and determination of the absolute configuration of natural products Fulltext Access 9 Pages 2005
Efficient electrocatalytic addition reactions of allyl phenyl sulfone to electron deficient alkenes Fulltext Access 9 Pages 2005
Convenient synthesis of 2-alkylamino-6-carboxy-5,7-diarylcyclopenteno[1,2-b]pyridines via direct acylamination with imidoyl chlorides Fulltext Access 9 Pages 2005
Aryl alkynylation versus alkyne homocoupling: unprecedented selectivity switch in Cu, phosphine and solvent-free heterogeneous Pd-catalysed couplings Fulltext Access 9 Pages 2005
Sonogashira reaction of aryl halides with propiolaldehyde diethyl acetal catalyzed by a tetraphosphine/palladium complex Fulltext Access 9 Pages 2005
8-Methylquinoline palladacycles: stable and efficient catalysts for carbon-carbon bond formation Fulltext Access 9 Pages 2005
Structure-activity relationship of trihexyphenidyl analogs with respect to the dopamine transporter in the on going search for a cocaine inhibitor Fulltext Access 9 Pages 2005
Non-thiol farnesyltransferase inhibitors: N-(4-aminoacylamino-3-benzoylphenyl)-3-[5-(4-nitrophenyl)-2 furyl]acrylic acid amides and their antimalarial activity Fulltext Access 9 Pages 2005
Homology models of the cannabinoid CB1 and CB2 receptors. A docking analysis study Fulltext Access 9 Pages 2005
Non-imidazole histamine H3 ligands. Part III. New 4-n-propylpiperazines as non-imidazole histamine H3-antagonists Fulltext Access 9 Pages 2005
Estimation of the effect of the acidosis and alkalosis on the anesthetic potency of local anesthetics by biopartitioning micellar chromatography and micellar electrokinetic chromatography Fulltext Access 9 Pages 2005
Novel inhibitors of acetyl- and butyrylcholinesterase derived from the alkaloids dehydroevodiamine and rutaecarpine Fulltext Access 9 Pages 2005
Synthesis and evaluation of new tripeptide phosphonate inhibitors of MMP-8 and MMP-2 Fulltext Access 9 Pages 2005
Synthesis and in vitro cytotoxic evaluation of 1,3-bisubstituted and 1,3,9-trisubstituted β-carboline derivatives Fulltext Access 9 Pages 2005
Benzenesulfonamide analogs of fluoroquinolones. Antibacterial activity and QSAR studies Fulltext Access 9 Pages 2005
Construction of a virtual combinatorial library using SMILES strings to discover potential structure-diverse PPAR modulators Fulltext Access 9 Pages 2005
Synthesis of 2-substituted β-cyclodextrin derivatives with a hydrolytic activity against the organophosphorylester paraoxon Fulltext Access 9 Pages 2005
Synthesis and evaluation of the antitrypanosomal and antiplasmodial activities of new 4-aminobicyclo[2.2.2]octane derivatives Fulltext Access 9 Pages 2005
Design, synthesis and bioactivities of TAR RNA targeting β-carboline derivatives based on Tat-TAR interaction Fulltext Access 9 Pages 2005
Palladacycles bearing pendant benzamidinate ligands as catalysts for the Suzuki and Heck coupling reactions Fulltext Access 9 Pages 2005
Design, synthesis and biological activity of acyl substituted 3-amino-5-methyl-1,4,5,7-tetrahydropyrazolo[3,4-b]pyridin-6-ones as potential hypnotic drugs Fulltext Access 9 Pages 2005
AMBER force field implementation of the boronate function to simulate the inhibition of β-lactamases by alkyl and aryl boronic acids Fulltext Access 9 Pages 2005
Synthesis of 2,5- and 3,5-diphenylpyridine derivatives for DNA recognition and cytotoxicity Fulltext Access 9 Pages 2005
Novel milrinone analogs of pyridine-3-carbonitrile derivatives as promising cardiotonic agents Fulltext Access 9 Pages 2005
A new potential cyclooxygenase-2 inhibitor, pyridinic analogue of nimesulide Fulltext Access 9 Pages 2005
Synthesis and biological evaluation of functionalized coumarins as acetylcholinesterase inhibitors Fulltext Access 9 Pages 2005
Structural changes of benzylether derivatives of vesamicol and their influence on the binding selectivity to the vesicular acetylcholine transporter Fulltext Access 9 Pages 2005
Synthesis of α,α-disubstituted amino acids based on tandem reaction of dehydroamino acid derivatives Fulltext Access 9 Pages 2005
2-Bromoethyl glycosides for synthesis of glycoconjugates on solid support Fulltext Access 9 Pages 2005
Synthesis of a β-turn mimetic suitable for incorporation in the peptide hormone LHRH Fulltext Access 9 Pages 2005
Galanthamine analogs: 6H-benzofuro[3a,3,2,-e,f][1]benzazepine and 6H-benzofuro[3a,3,2-e,f][3]benzazepine Fulltext Access 9 Pages 2005
Efficient synthesis of new 11-thiasteroids and their oxides and dioxides Fulltext Access 9 Pages 2005
Synthesis, X-ray crystallographic, and dynamic 1H NMR studies of crown-tetrathia[3.3.3.3]metacyclophanes-conformational control by cooperative intramolecular C-Hâ¯Ï interaction both in solid state and in solution Fulltext Access 9 Pages 2005
5-Hydroxy-3-phenyl-5-vinyl-2-isoxazoline and 3-phenyl-5-vinylisoxazole: synthesis and reactivity Fulltext Access 9 Pages 2005
Preparation of novel 3H-trifluoromethyldiazirine-based photoactivatable potassium channel antagonists Fulltext Access 9 Pages 2005
Arylzinc species by microwave assisted Grignard formation-transmetallation sequence: application in the Negishi coupling Fulltext Access 9 Pages 2005
Nitrogen is a requirement for the photochemical induced 3-azabicyclo[3.3.1]nonane skeletal rearrangement! Fulltext Access 9 Pages 2005
Silver acetate-catalysed asymmetric 1,3-dipolar cycloadditions of imines and chiral acrylamides Fulltext Access 9 Pages 2005
Formal total synthesis of (+)-wortmannin using catalytic asymmetric intramolecular aldol condensation reaction Fulltext Access 9 Pages 2005
An approach to the synthesis of α-(1-6)-C-disaccharides by tandem Tebbe methylenation and Claisen rearrangement Fulltext Access 9 Pages 2005
Utilization of 2-ethoxymethylene-3-oxobutanenitrile in the synthesis of heterocycles possessing biological activity Fulltext Access 9 Pages 2005
Substituent effects in the ring-chain tautomerism of 4-aryl-1,3,4,6,7,11b-hexahydro-2H-pyrimido[6,1-a]isoquinolines Fulltext Access 9 Pages 2005
Two-dimensional oligoarylenes: synthesis and structure-properties relationships Fulltext Access 9 Pages 2005
Organozinc alkoxide-promoted aldol-Tishchenko reaction of aliphatic aldehydes: an expedient entry to prepare the α-methylene ketones Fulltext Access 9 Pages 2005
Acid-catalysed synthesis and deprotection of dimethyl acetals in a miniaturised electroosmotic flow reactor Fulltext Access 9 Pages 2005
Efficient and versatile single pot approach to dipyrromethanes and bis(heterocyclyl)methanes Fulltext Access 9 Pages 2005
Fluorescence modification of Gb3 oligosaccharide and rapid synthesis of oligosaccharide moieties using fluorous protective group Fulltext Access 9 Pages 2005
X=Y-ZH systems as potential 1,3-dipoles. Part 61: Metal exchanged zeolites, silver(I) oxide, Ni(II) and Cu(I) complexes as catalysts for 1,3-dipolar cycloaddition reactions of imines generating proline derivatives Fulltext Access 9 Pages 2005
Synthesis and properties of 5-[bis(1-heteroazulen-3-yl)methylidene]pyrimidine-2,4,6(1,3,5H)-triones Fulltext Access 9 Pages 2005
A stereoselective route to multi-substituted tetrahydropyrans by vinyl radical cyclization Fulltext Access 9 Pages 2005
Conformationally restricted analogues of both (S)-β-homoserine and (S)-aspartic acid from chiral 3-acylamino pyrrolidin-2-ones Fulltext Access 9 Pages 2005
Organometallic alkylation of 2-chloro-4,6-dimethoxy-1,3,5-triazine: a study Fulltext Access 9 Pages 2005
Synthesis of alkyl 4-(diethoxymethyl)-3-pyridin-3-ylisoxazole-5-carboxylates: useful scaffold for highly functionalised 3-(pyridin-3-yl)isoxazoles Fulltext Access 9 Pages 2005
Ligand creation via linking-a rapid and convenient method for construction of novel supported PyOX-ligands Fulltext Access 9 Pages 2005
Development of a new traceless aniline linker for solid-phase synthesis of azomethines. Application to parallel synthesis of a rod-shaped liquid crystalline library Fulltext Access 9 Pages 2005
Micellar effect on the electron transfer reaction of chromium(V) ion with organic sulfides Fulltext Access 9 Pages 2005
Efficient syntheses of thiadiazoline and thiadiazole derivatives by the cyclization of 3-aryl-4-formylsydnone thiosemicarbazones with acetic anhydride and ferric chloride Fulltext Access 9 Pages 2005
A new (R)-hydroxynitrile lyase from Prunus mume: asymmetric synthesis of cyanohydrins Fulltext Access 9 Pages 2005
New reaction of enamines with aryldiazoacetates catalyzed by transition metal complexes Fulltext Access 9 Pages 2005
Trifluoromethyl group as a pharmacophore: Effect of replacing a CF3 group on binding and agonist activity of a glucocorticoid receptor ligand Fulltext Access 9 Pages 2005
Synthesis and solvent dependence of the photophysical properties of [60]fullerene-sugar conjugates Fulltext Access 9 Pages 2005
One-pot three-component reaction of fluoroalkanesulfonyl azide, vinyl ether and aldehyde: the formation of polysubstituted fluorinated oxazolidines Fulltext Access 9 Pages 2005
Synthesis and properties of 3-arylcyclohepta[4,5]imidazo[1,2-a]-1,3,5-triazine-2,4(3H)-diones and related compounds: photo-induced autorecycling oxidation of some amines Fulltext Access 9 Pages 2005
Regioselective formation of N-alkyl-3,5-pyrazole derived ligands. A synthetic and computational study Fulltext Access 9 Pages 2005
The optimization for cyclization reaction of 2-(2-carbomethoxyethynyl)aniline derivatives and formal synthesis of pyrroloquinoline quinone and its analogue utilizing a sequential coupling-cyclization reaction Fulltext Access 9 Pages 2005
Structural analyses of 4-benzoylpyridine thiosemicarbazone using NMR techniques and theoretical calculations Fulltext Access 9 Pages 2005
Photoinduced electron transfer across linearly fused oligo-norbornyl structures Fulltext Access 9 Pages 2005