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Daneshyari Pharmaceutical Science Journas Latest Articles

Pharmaceutical Science Research Articles

Selectivity of Similar Compounds Identification Using IR Spectroscopy: Steroids
Fulltext Access 10 Pages 2007
Stability and degradation kinetics of etoposide‐loaded parenteral lipid emulsion
Fulltext Access 10 Pages 2007
Influence of crystal structure on the tableting properties of n‐alkyl 4‐hydroxybenzoate esters (parabens)
Fulltext Access 10 Pages 2007
A comparative study of the antigen‐specific immune response induced by co‐delivery of CpG ODN and antigen using fusion molecules or biodegradable microparticles*
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Interactions of azole antifungal agents with the human breast cancer resistance protein (BCRP)
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Onion Phases of PEG-8 Distearate
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Solid‐state properties and relationship between anhydrate and monohydrate of baclofen
Fulltext Access 10 Pages 2007
Single-Droplet Evaporation Kinetics and Particle Formation in an Acoustic Levitator. Part 1: Evaporation of Water Microdroplets Assessed Using Boundary-Layer and Acoustic Levitation Theories
Fulltext Access 10 Pages 2007
A Solid-State Chemist's View of the Crystal Polymorphism of Organic Compounds
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Modifying Drug Release and Tablet Properties of Starch Acetate Tablets by Dry Powder Agglomeration
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In vivo drug metabolism model for human cytochrome P450 enzyme using chimeric mice with humanized liver
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Effect of Moisture and Pressure on Tablet Compaction Studied With FTIR Spectroscopic Imaging
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Air-Liquid Interface (ALI) Culture of Human Bronchial Epithelial Cell Monolayers as an in vitro Model for Airway Drug Transport Studies
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Characterization of Prednisolone in Controlled Porosity Osmotic Pump Pellets using Solid-State NMR Spectroscopy
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Predicting Human Drug Pharmacokinetics from In Vitro Permeability Using an Absorption-Disposition Model
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Relative in Vitro Efficacy of the Phosphate Binders Lanthanum Carbonate and Sevelamer Hydrochloride
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Grapefruit Juice-Drug Interactions: Grapefruit Juice and Its Components Inhibit P‐Glycoprotein (ABCB1) Mediated Transport of Talinolol in Caco‐2 Cells
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In Vitro Penetration of a Novel Oxaborole Antifungal (AN2690) Into the Human Nail Plate
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Design of ocular inserts of brimonidine tartrate by response surface methodology
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Formulation and physicochemical characterisation of buccoadhesive films containing ketorolac
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Novel physically structured lipid matrices of beeswax and a homolipid from Capra hircus (goat fat): a physicochemical characterization for application in drug delivery
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The preparation of pellets containing a surfactant or a mixture of mono- and di-gylcerides by extrusion/spheronization
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Synthesis of indolizine derivatives with selective antibacterial activity against Mycobacterium tuberculosis
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Biodistribution of doxorubicin-alkylated poly(l-lysine citramide imide) conjugates in an experimental model of peritoneal carcinomatosis after intraperitoneal administration
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Comparison between immobilized artificial membrane (IAM) HPLC data and lipophilicity in n-octanol for quinolone antibacterial agents
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Biowaiver Monographs for Immediate Release Solid Oral Dosage Forms: Isoniazid*
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Current perspectives in dissolution testing of conventional and novel dosage forms
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Distribution, transition, adhesion and release of insulin loaded nanoparticles in the gut of rats
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Preparation of monolithic matrices for oral drug delivery using a supercritical fluid assisted hot melt extrusion process
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Evaluation of an eucalyptus oil containing topical drug delivery system for selected steroid hormones
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Tumor necrosis factor alpha blocking peptide loaded PEG-PLGA nanoparticles: Preparation and in vitro evaluation
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Nanoparticles—a historical perspective
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Antiproliferative activity and induction of apoptosis in human colon cancer cells treated in vitro with constituents of a product derived from Pistacia lentiscus L. var. chia
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In vitro evaluation of human cytochrome P450 and P-glycoprotein-mediated metabolism of some phytochemicals in extracts and formulations of African potato
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A randomized, placebo-controlled, double-blind clinical trial of curcuminoids in oral lichen planus
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Specific reversal of multidrug resistance to colchicine in CEM/VLB100 cells by Gynostemma pentaphyllum extract
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The herbal medicines Saireito and Boiogito improve the hypertension of pre-eclamptic rats induced by Nω-Nitro-l-arginine methyl ester
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Investigation of Drying Stresses on Proteins during Lyophilization: Differentiation between Primary and Secondary-Drying Stresses on Lactate Dehydrogenase Using a Humidity Controlled Mini Freeze-Dryer
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Thermodynamic analysis of binding between drugs and glycosaminoglycans by isothermal titration calorimetry and fluorescence spectroscopy
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Species Differences of Inhibitory Effects on P‐glycoprotein‐mediateD Drug Transport
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Different HPMC Viscosity Grades as Coating Agents for an Oral Time and/or Site‐Controlled Delivery System: An Investigation into the Mechanisms Governing Drug Release
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Biowaiver Monographs for Immediate Release Solid Oral Dosage Forms: Prednisone
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Ex Vivo Study of Transdermal Permeation of Four Diclofenac Salts from Different Vehicles
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Gelatin‐stabilised microemulsion‐based organogels facilitates percutaneous penetration of Cyclosporin A In Vitro and dermal pharmacokinetics In Vivo
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The 3-D model: Experimental Testing of the Parameters d, e, and ω and Validation of the Analysis
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Transformation of Pharmaceutical Compounds upon Milling and Comilling: The Role of Tg
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Process Analytical Technology: Chemometric Analysis of Raman and Near Infra-Red Spectroscopic Data for Predicting Physical Properties of Extended Release Matrix Tablets
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Hydrates and Solid-State Reactivity: A Survey of β-Lactam Antibiotics
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Solvent Influences on Metastable Polymorph Lifetimes: Real-Time Interconversions Using Energy Dispersive X-Ray Diffractometry*
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Thermal Expansion of Organic Crystals and Precision of Calculated Crystal Density: A Survey of Cambridge Crystal Database
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Two galactomannans and scleroglucan as matrices for drug delivery: Preparation and release studies
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Microstructural and drug release properties of oven-dried and of slowly or fast frozen freeze-dried MCC-Carbopol® pellets
Fulltext Access 10 Pages 2007
Probing the skin permeation of eicosapentaenoic acid and ketoprofen: 2. Comparative depth profiling and metabolism of eicosapentaenoic acid
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The effect of different lipid based formulations on the oral absorption of lipophilic drugs: The ability of in vitro lipolysis and consecutive ex vivo intestinal permeability data to predict in vivo bioavailability in rats
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Development, characterization and in vivo evaluation of benzocaine-loaded liposomes
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Reduced hepatic toxicity, enhanced cellular uptake and altered pharmacokinetics of stavudine loaded galactosylated liposomes
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Solid lipid nanodispersions containing mixed lipid core and a polar heterolipid: Characterization
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Release modulating hydrophilic matrix systems of losartan potassium: Optimization of formulation using statistical experimental design
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Influence of moisture content on the mechanical properties of methyl methacrylate–starch copolymers
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Cellulose acetate butyrate–pH/thermosensitive polymer microcapsules containing aminated poly(vinyl alcohol) microspheres for oral administration of DNA
Fulltext Access 10 Pages 2007
An integrated early formulation strategy – From hit evaluation to preclinical candidate profiling
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Permeability assessment for solid oral drug formulations based on Caco-2 monolayer in combination with a flow through dissolution cell
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Synchronized and sustained release of multiple components in silymarin from erodible glyceryl monostearate matrix system
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In vitro release of a water-soluble agent from low viscosity biodegradable, injectable oligomers
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Investigation into the subambient behavior of aqueous mannitol solutions using temperature-controlled Raman microscopy
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Preparation of a novel freeze thawed poly(vinyl alcohol) composite hydrogel for drug delivery applications
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Cross-linking of chitosan and chitosan/poly(ethylene oxide) beads: A theoretical treatment
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Long-circulating poly(ethylene glycol)-coated emulsions to target solid tumors
Fulltext Access 10 Pages 2007
Production of solid lipid nanoparticle suspensions using supercritical fluid extraction of emulsions (SFEE) for pulmonary delivery using the AERx system
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Delivery of drugs and macromolecules to mitochondria
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Oral lipid-based formulations
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Non-viral siRNA delivery to the lung
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Cellular and multicellular form and function
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Transdermal skin delivery: Predictions for humans from in vivo, ex vivo and animal models
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Transgenic animal models of neurodegenerative diseases and their application to treatment development
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Enhanced cytotoxicity of monoclonal anticancer antibody 2C5-modified doxorubicin-loaded PEGylated liposomes against various tumor cell lines
Fulltext Access 10 Pages 2007
An alkylpolyglucoside surfactant as a prospective pharmaceutical excipient for topical formulations: The influence of oil polarity on the colloidal structure and hydrocortisone in vitro/in vivo permeation
Fulltext Access 10 Pages 2007
Structural characterization of insulin NPH formulations
Fulltext Access 10 Pages 2007
Effects of block length on the enzymatic degradation and erosion of oxazoline linked poly-ɛ-caprolactone
Fulltext Access 10 Pages 2007
Formulation development and manufacturing of a gastrin/CCK-2 receptor targeting peptide as an intermediate drug product for a clinical imaging study
Fulltext Access 10 Pages 2007
Morphological observations on a lipid-based drug delivery system during in vitro digestion
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Characterization of human cytochrome P450 enzymes involved in the metabolism of cyamemazine
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Helium pycnometry as a tool for assessment of sealing efficiency in microencapsulation
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Long-circulating, pH-sensitive liposomes sterically stabilized by copolymers bearing short blocks of lipid-mimetic units
Fulltext Access 10 Pages 2007
Development of simulated intestinal fluids containing nutrients as transport media in the Caco-2 cell culture model: Assessment of cell viability, monolayer integrity and transport of a poorly aqueous soluble drug and a substrate of efflux mechanisms
Fulltext Access 10 Pages 2007
Theoretical assessment of a new experimental protocol for determining kinetic values describing mechanism (time)-based enzyme inhibition
Fulltext Access 10 Pages 2007
The study of the influence of surfactant charge on alkaline hydrolysis reactions of acetylsalicylic acid (ASA) and triflusal (TFL) using spectrophotometric methods
Fulltext Access 10 Pages 2007
Influence of erythrocytes on the hepatic distribution kinetics of urea and thiourea
Fulltext Access 10 Pages 2007
Design, synthesis and melatoninergic activity of new unsubstituted and β,β′-difunctionalised 2,3-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-6-alkanamides
Fulltext Access 10 Pages 2007
Hypertension artérielle pulmonaire : stratégies de prise en charge
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Médicaments sous autorisation temporaire d'utilisation (ATU)
Fulltext Access 10 Pages 2007
Innovations thérapeutiques hors ATU
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Resistance to echinocandin-class antifungal drugs
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Roots of imatinib resistance: A question of self-renewal?
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Effect of surfactant on dissolution of spherical particles in micellar systems
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Contents for Volumes 65-67
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Immediate release of poorly soluble drugs from starch-based pellets prepared via extrusion/spheronisation
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Nanoparticles based on N-trimethylchitosan: Evaluation of absorption properties using in vitro (Caco-2 cells) and ex vivo (excised rat jejunum) models
Fulltext Access 10 Pages 2007
Solid lipid microparticles as a sustained release system for pulmonary drug delivery
Fulltext Access 10 Pages 2007
A comparison of the effectiveness of cationic polymers poly-l-lysine (PLL) and polyethylenimine (PEI) for non-viral delivery of plasmid DNA to bone marrow stromal cells (BMSC)
Fulltext Access 10 Pages 2007
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