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Daneshyari Pharmaceutical Science Journas Latest Articles

Pharmaceutical Science Research Articles

Intestinal uptake and biodistribution of novel polymeric micelles after oral administration
Fulltext Access 9 Pages 2006
Metabolism of Dopamine by the Nasal Mucosa
Fulltext Access 9 Pages 2006
Prise en charge thérapeutique de la migraine
Fulltext Access 9 Pages 2006
Nasal absorption of metoclopramide from different Carbopol® 981 based formulations: In vitro, ex vivo and in vivo evaluation
Fulltext Access 9 Pages 2006
Comparison of permeation enhancing strategies for an oral factor Xa inhibitor using the Caco-2 cell monolayer model
Fulltext Access 9 Pages 2006
Anionic clays for sunscreen agent safe use: Photoprotection, photostability and prevention of their skin penetration
Fulltext Access 9 Pages 2006
In vitro uptake of gelatin nanoparticles by murine dendritic cells and their intracellular localisation
Fulltext Access 9 Pages 2006
Compaction behaviour and new predictive approach to the compressibility of binary mixtures of pharmaceutical excipients
Fulltext Access 9 Pages 2006
Use of κ-carrageenan as alternative pelletisation aid to microcrystalline cellulose in extrusion/spheronisation. I. Influence of type and fraction of filler
Fulltext Access 9 Pages 2006
Practical method for choosing diluent that ensures the best temperature uniformity in the case of pharmaceutical microwave vacuum drying of a heat sensitive product
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Silk fibroin as an organic polymer for controlled drug delivery
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Photochemically stimulated drug delivery increases the cytotoxicity and specificity of EGF–saporin
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Effect of particle size reduction on dissolution and oral absorption of a poorly water-soluble drug, cilostazol, in beagle dogs
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Release-Controlling Absorption Enhancement of Enterally Administered Ophiopogon Japonicus Polysaccharide by Sodium Caprate in Rats
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Formulation optimization for the nanoparticles-in-microsphere hybrid oral delivery system using factorial design
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Formation of drug–arylsulfonate complexes inside liposomes: A novel approach to improve drug retention
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Enhancement of bronchial octreotide absorption by chitosan and N-trimethyl chitosan shows linear in vitro/in vivo correlation
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Colon-specific 9-aminocamptothecin-HPMA copolymer conjugates containing a 1,6-elimination spacer
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A multi-scale stochastic drug release model for polymer-coated targeted drug delivery systems
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The “inverted cup” - A novel in vitro release technique for drugs in lipid formulations
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Delivery of gadolinium-labeled nanoparticles to the sentinel lymph node: Comparison of the sentinel node visualization and estimations of intra-nodal gadolinium concentration by the magnetic resonance imaging
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New self-assembled nanogels based on host–guest interactions: Characterization and drug loading
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Efficacy of orally active chemical conjugate of low molecular weight heparin and deoxycholic acid in rats, mice and monkeys
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Crosslinked chitosan implants as potential degradable devices for brachytherapy: In vitro and in vivo analysis
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PLGA: Poloxamer and PLGA: Poloxamine blend nanostructures as carriers for nasal gene delivery
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Transcellular route of diffusion through stratum corneum: Results from finite element models
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Development and evaluation of an artificial membrane for determination of drug availability
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Platelet adsorption and hemolytic properties of liquid crystal/composite polymers
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Effect of milling conditions on the solid-state conversion of ranitidine hydrochloride form 1
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The effect of carrier surface treatment on drug particle detachment from crystalline carriers in adhesive mixtures for inhalation
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Crystal structure and physical properties of two polymorphs of ropivacaine HCl
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Electromigration of ions across the skin: Determination and prediction of transport numbers
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Effects of citronellal, a monoterpenoid in Zanthoxyli Fructus, on the intestinal absorption of digoxin in vitro and in vivo
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Polymorphism on Leflunomide: Stability and Crystal Structures
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Effect of cationized gelatins on the paracellular transport of drugs through caco-2 cell monolayers
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Hyperthermia-Induced Antitumor Activity of Thermosensitive Polymer Modified Temperature-Sensitive Liposomes
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Near-infrared analysis of protein secondary structure in aqueous solutions and freeze-dried solids
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Tetrazole compounds: The effect of structure and pH on Caco-2 cell permeability
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Novel ultra-deformable vesicles entrapped with bleomycin and enhanced to penetrate rat skin
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Investigation of Solid-State NMR Line Widths of Ibuprofen in Drug Formulations
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Bioadhesive monolayer film for the in vitro transdermal delivery of sumatriptan
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The Effects of Surface Lactone Hydrolysis and Temperature on the Specific and Nonspecific Interactions Between Phenobarbital and Activated Carbon Surfaces
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Prediction of Tablet Hardness Based on Near Infrared Spectra of Raw Mixed Powders by Chemometrics
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Deep Percutaneous Penetration into Muscles and Joints
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Bile Acid Salt Binding with Colesevelam HCl is Not Affected by Suspension in Common Beverages
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Primary Microparticles and Agglomerates of Morphine for Nasal Insufflation
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Thiol exchange: An in vitro assay that predicts the efficacy of novel homocysteine lowering therapies
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Labetalol absorption kinetics: Rat small intestine and colon studies
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Static light scattering and small-angle neutron scattering study on aggregated recombinant gelatin in aqueous solution
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An efficient approach for the rapid assessment of oral rat exposures for new chemical entities in drug discovery
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Influence of plasmid DNA topology on the transfection properties of DOTAP/DOPE lipoplexes
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Biodegradable polymersomes loaded with both paclitaxel and doxorubicin permeate and shrink tumors, inducing apoptosis in proportion to accumulated drug
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Disassembly of polyethylenimine-DNA particles in vitro: Implications for polyethylenimine-mediated DNA delivery
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Prolonged blood concentration of prednisolone after intravenous injection of liposomal palmitoyl prednisolone
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Biodistribution characteristics of amino acid dendrimers and their PEGylated derivatives after intravenous administration
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Histidine-conjugated poly(amino acid) derivatives for the novel endosomolytic delivery carrier of doxorubicin
Fulltext Access 9 Pages 2006
DNA/cationic polymer complex attachment on a human vascular endothelial cell monolayer exposed to a steady laminar flow
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Improved intestinal delivery of salmon calcitonin by Lys18-amine specific PEGylation: Stability, permeability, pharmacokinetic behavior and in vivo hypocalcemic efficacy
Fulltext Access 9 Pages 2006
A polymeric micelle MRI contrast agent with changeable relaxivity
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Preparation and evaluation of lectin-conjugated PLGA nanoparticles for oral delivery of thymopentin
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Wet sol–gel derived silica for controlled release of proteins
Fulltext Access 9 Pages 2006
Self-assembled thermo- and pH responsive micelles of poly(10-undecenoic acid-b-N-isopropylacrylamide) for drug delivery
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Floating hot-melt extruded tablets for gastroretentive controlled drug release system
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Tumor accumulation, degradation and pharmacokinetics of elastin-like polypeptides in nude mice
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Silk sericin–insulin bioconjugates: Synthesis, characterization and biological activity
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Drugs acting as plasticizers in polymeric systems: A quantitative treatment
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Positively charged polyethylenimines enhance nasal absorption of the negatively charged drug, low molecular weight heparin
Fulltext Access 9 Pages 2006
Cervical cancer treatment with a locally insertable controlled release delivery system
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Release of ibuprofen from beads for embolization: In vitro and in vivo studies
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Synthesis, structure, toxicological and pharmacological investigations of 4-hydroxycoumarin derivatives
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Syntheses and odor of “bulky group”-modified sandalwood odorants: isophorono-β-santalol analogues
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Air to fat and blood to fat distribution of volatile organic compounds and drugs: Linear free energy analyses
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Structural modifications of benzanilide derivatives, effective potassium channel openers. X.
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Antihelminthic activity of some newly synthesized 5(6)-(un)substituted-1H-benzimidazol-2-ylthioacetylpiperazine derivatives
Fulltext Access 9 Pages 2006
Synthesis, crystal structure and anticancer activity of novel derivatives of ethyl 1-(4-oxo-8-aryl-4,6,7,8-tetrahydroimidazo[2,1-c][1,2,4]triazin-3-yl)formate
Fulltext Access 9 Pages 2006
N-acetyl histidine-conjugated glycol chitosan self-assembled nanoparticles for intracytoplasmic delivery of drugs: Endocytosis, exocytosis and drug release
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Enhancement of transdermal delivery of 6-β-naltrexol via a codrug linked to hydroxybupropion
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Microsphere-integrated collagen scaffolds for tissue engineering: Effect of microsphere formulation and scaffold properties on protein release kinetics
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Calcium phosphate cements as bone drug delivery systems: A review
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Biodegradable nanoparticles loaded with insulin–phospholipid complex for oral delivery: Preparation, in vitro characterization and in vivo evaluation
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Effect of mannose density on mannose receptor-mediated cellular uptake of mannosylated O/W emulsions by macrophages
Fulltext Access 9 Pages 2006
Tracking the in vivo fate of recombinant polypeptides by isotopic labeling
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Polymeric conjugates of mono- and bi-cyclic αVβ3 binding peptides for tumor targeting
Fulltext Access 9 Pages 2006
Painless electroporation with a new needle-free microelectrode array to enhance transdermal drug delivery
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Well-ordered mesoporous bioactive glasses (MBG): A promising bioactive drug delivery system
Fulltext Access 9 Pages 2006
Targeted drug delivery crossing cytoplasmic membranes of intended cells via ligand-grafted sterically stabilized liposomes
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Inducing effect of liposomalization on the transdermal delivery of hydrocortisone: Creation of a drug supersaturated state
Fulltext Access 9 Pages 2006
Insights into synergistic interactions in binary mixtures of chemical permeation enhancers for transdermal drug delivery
Fulltext Access 9 Pages 2006
Air to brain, blood to brain and plasma to brain distribution of volatile organic compounds: linear free energy analyses
Fulltext Access 9 Pages 2006
Block ionomer complexes as prospective nanocontainers for drug delivery
Fulltext Access 9 Pages 2006
Development and in vitro validation of a targeted delivery vehicle for DNA vaccines
Fulltext Access 9 Pages 2006
Melittin analogs with high lytic activity at endosomal pH enhance transfection with purified targeted PEI polyplexes
Fulltext Access 9 Pages 2006
Electrochemical Time-of-Flight in crosslinked collagen matrix solution: Implications of structural changes for drug delivery systems
Fulltext Access 9 Pages 2006
Efficient delivery of a Bcl-2-specific antisense oligodeoxyribonucleotide (G3139) via transferrin receptor-targeted liposomes
Fulltext Access 9 Pages 2006
Intramuscular delivery of DNA releasing microspheres: Microsphere properties and transgene expression
Fulltext Access 9 Pages 2006
Deamidation, acylation and proteolysis of a model peptide in PLGA films
Fulltext Access 9 Pages 2006
New loading process and release properties of insulin from polysaccharide microcapsules fabricated through layer-by-layer assembly
Fulltext Access 9 Pages 2006
In vivo targeting of dendritic cells in lymph nodes with poly(propylene sulfide) nanoparticles
Fulltext Access 9 Pages 2006
Imprinted soft contact lenses as norfloxacin delivery systems
Fulltext Access 9 Pages 2006
Role of SLC xenobiotic transporters and their regulatory mechanisms PDZ proteins in drug delivery and disposition
Fulltext Access 9 Pages 2006
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