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Daneshyari Drug Discovery Journas Latest Articles

Drug Discovery Research Articles

Synthesis and biological evaluation of benzimidazole derivatives as potent AMP-activated protein kinase activators
Fulltext Access 29 Pages 2006
Synthetic applications of fluorous solid-phase extraction (F-SPE)
Fulltext Access 29 Pages 2006
A Multiphase Microscopic Diffusion Model for Stratum Corneum permeability. I. Formulation, Solution, and Illustrative Results for Representative Compounds
Fulltext Access 29 Pages 2006
Strategies and approaches for constructing 1-oxadecalins
Fulltext Access 29 Pages 2006
Stereochemistry abstracts
Fulltext Access 29 Pages 2006
Solvent and in situ catalyst preparation impacts upon Noyori reductions of aryl-chloromethyl ketones: application to syntheses of chiral 2-amino-1-aryl-ethanols
Fulltext Access 29 Pages 2006
Stereochemistry abstracts
Fulltext Access 29 Pages 2006
Syntheses and applications of C2-symmetric chiral diols
Fulltext Access 29 Pages 2006
Recent developments in the clinical activity of topoisomerase-1 inhibitors
Fulltext Access 29 Pages 2006
Plasma cell dyscrasias and leukemias
Fulltext Access 29 Pages 2006
Qualitative simulation of the carbon starvation response in Escherichia coli
Fulltext Access 29 Pages 2006
Stereochemistry abstracts
Fulltext Access 30 Pages 2006
Stereochemistry abstracts
Fulltext Access 30 Pages 2006
Stereochemistry abstracts
Fulltext Access 30 Pages 2006
Stereochemistry abstracts
Fulltext Access 30 Pages 2006
Correlation of blood–brain penetration using structural descriptors
Fulltext Access 30 Pages 2006
Design, synthesis, structure–activity relationship, and in vivo activity of azabicyclic aryl amides as α7 nicotinic acetylcholine receptor agonists
Fulltext Access 30 Pages 2006
A journey across the sequential development of macrolides and ketolides related to erythromycin
Fulltext Access 30 Pages 2006
ASMS Directory of Members: 224S-254S, E Bruns-E De Oliveira
Fulltext Access 31 Pages 2006
ASMS Directory of Members: 255S-285S, E De Pauw-BY Giang
Fulltext Access 31 Pages 2006
ASMS Directory of Members: 286S-316S, AK Gianotto-RA Huagn
Fulltext Access 31 Pages 2006
ASMS Directory of Members: 317S-347S, B Huang-S Kumar
Fulltext Access 31 Pages 2006
ASMS Directory of Members: 348S-378S, S Kumar-R Martin
Fulltext Access 31 Pages 2006
ASMS Directory of Members: 379S-409S, S A Martin-T Owens
Fulltext Access 31 Pages 2006
ASMS Directory of Members: 410S-440S, D Owusu-F Salama
Fulltext Access 31 Pages 2006
ASMS Directory of Members: 193S-223S, D Aaserud-A Brunnstrom
Fulltext Access 31 Pages 2006
ASMS Directory of Members: 441S-471S, GA Salazar-S Suzuki
Fulltext Access 31 Pages 2006
ASMS Directory of Members: 472S-502S, S Suzuki-Z Wen
Fulltext Access 31 Pages 2006
Modern Pummerer-type reactions
Fulltext Access 32 Pages 2006
ASMS Directory of Members: 503S-534S, Z Wen-Z Zych
Fulltext Access 32 Pages 2006
Stereochemistry abstracts
Fulltext Access 33 Pages 2006
Pyrrole protection
Fulltext Access 33 Pages 2006
Stereochemistry abstracts
Fulltext Access 33 Pages 2006
Stereochemistry abstracts
Fulltext Access 34 Pages 2006
Stereochemistry abstracts
Fulltext Access 35 Pages 2006
Stereochemistry abstracts
Fulltext Access 35 Pages 2006
Synthesis of amino- and diaminoconduritols and their applications
Fulltext Access 36 Pages 2006
Stereochemistry abstracts
Fulltext Access 37 Pages 2006
Chiral non-racemic sulfinimines: versatile reagents for asymmetric synthesis
Fulltext Access 37 Pages 2006
Neuropharmacology of cognition and memory: A unifying theory of neuromodulator imbalance in psychiatry and amnesia
Fulltext Access 38 Pages 2006
Lung cancer
Fulltext Access 38 Pages 2006
Central nervous system tumors
Fulltext Access 39 Pages 2006
Stereochemistry abstracts
Fulltext Access 39 Pages 2006
The chemistry of recently isolated naturally occurring quinazolinone alkaloids
Fulltext Access 40 Pages 2006
Integration of hepatic drug transporters and phase II metabolizing enzymes: Mechanisms of hepatic excretion of sulfate, glucuronide, and glutathione metabolites
Fulltext Access 40 Pages 2006
Les systèmes de délivrance des médicaments : un réel progress pour la thérapeutique*
Fulltext Access 41 Pages 2006
Stereochemistry abstracts
Fulltext Access 42 Pages 2006
Stereochemistry abstracts
Fulltext Access 43 Pages 2006
Heterocyclic compounds with a silicon atom and another non-adjacent different heteroatom
Fulltext Access 43 Pages 2006
Use of chiral sulfoxides in asymmetric synthesis
Fulltext Access 43 Pages 2006
Stereochemistry abstracts
Fulltext Access 44 Pages 2006
Tetrahedron report number 762Synthesis and biological activity of pyrrole, pyrroline and pyrrolidine derivatives with two aryl groups on adjacent positions
Fulltext Access 44 Pages 2006
A synthon approach to spiro compounds
Fulltext Access 50 Pages 2006
Synthesis and role of glycosylthio heterocycles in carbohydrate chemistry
Fulltext Access 56 Pages 2006
Estimation of Melting Points of Organic Compounds-II
Fulltext Access 57 Pages 2006
Author index
Fulltext Access 59 Pages 2006
Lipase-promoted dynamic kinetic resolution of racemic β-hydroxyalkyl sulfones
Fulltext Access 4 Pages 2005
Instructions to contributors
Fulltext Access 4 Pages 2005
Catalytic and stereoselective iodination of prochiral C–H bonds
Fulltext Access 4 Pages 2005
Organocatalysis of asymmetric epoxidation mediated by iminium salts: comments on the mechanism
Fulltext Access 4 Pages 2005
Diastereoselective rhodium-catalyzed nitrene transfer starting from chiral sulfonimidamide-derived iminoiodanes
Fulltext Access 4 Pages 2005
Diastereoselective alkylation of chiral 2-imidazolidinone glycolates: asymmetric synthesis of α-hydroxy carboxylic acids
Fulltext Access 4 Pages 2005
Extending the solvent-free MALDI sample preparation method
Fulltext Access 4 Pages 2005
An in situ silver cationization method for hydrocarbon mass spectrometry
Fulltext Access 4 Pages 2005
Instructions to contributors
Fulltext Access 4 Pages 2005
Phosphoramidite ligands for the enantioselective iridium-catalyzed asymmetric hydroboration of meso-bicyclic hydrazines
Fulltext Access 4 Pages 2005
Synthesis of optically active (+)-2-benzyl-, (+)-2-octyl-, and (+)-2-tetradec-5′-enylcyclobutanones via metallated chiral imines or hydrazones
Fulltext Access 4 Pages 2005
A versatile synthesis of phosphine–aminophosphine ligands for asymmetric catalysis
Fulltext Access 4 Pages 2005
Ionic-Liquid Matrices for Improved Analysis of Phospholipids by MALDI-TOF Mass Spectrometry
Fulltext Access 4 Pages 2005
Unusual base dependent enantioselectivity in a transfer hydrogenation using axially chiral Ir(III)-catalysts
Fulltext Access 4 Pages 2005
Instructions to contributors
Fulltext Access 4 Pages 2005
Instructions to contributors
Fulltext Access 4 Pages 2005
Chiral separation of amino acids by chiral octamide derivatives of calixarenes derived from resorcinol by impregnation on a polymeric support
Fulltext Access 4 Pages 2005
A highly enantioselective, moderately anti-selective aldol reaction using a novel hydrazone moiety as stereo director
Fulltext Access 4 Pages 2005
Stereocontrolled synthesis of conformationally restricted enantiopure triols and dihydroxy acids based on the norbornane framework
Fulltext Access 4 Pages 2005
Asymmetric synthesis of (S)-homocitric acid lactone
Fulltext Access 4 Pages 2005
Instructions to contributors
Fulltext Access 4 Pages 2005
Instructions to contributors
Fulltext Access 4 Pages 2005
Instructions to contributors
Fulltext Access 4 Pages 2005
Graphical contents list
Fulltext Access 4 Pages 2005
Microwave-assisted ethylene–alkyne cross-metathesis: synthesis of chiral 2-(N-1-acetyl-1-arylmethyl)-1,3-butadienes
Fulltext Access 4 Pages 2005
Stereochemistry of the Diels–Alder reaction at high pressure: diastereo- and enantioselective [4+2]cycloaddition of buta-1,3-diene to glyoxylic acid derivatives catalysed by (salen) chromium(III) complexes
Fulltext Access 4 Pages 2005
Instructions to contributors
Fulltext Access 4 Pages 2005
Asymmetric synthesis of 1-substituted tetrahydro-3-benzoazepines
Fulltext Access 4 Pages 2005
The first total synthesis of (R)-7-butyl-6,8-dihydroxy-3-pentylisochroman-1-one
Fulltext Access 4 Pages 2005
Synthesis and characterization of axially chiral enantiopure novel dendrimers
Fulltext Access 4 Pages 2005
Enzymatic resolution of (±)-2-endo-hydroxymethyl and acetoxymethyl substituted hexachloronorbornene derivatives
Fulltext Access 4 Pages 2005
Chiral tertiary alcohols from a trans-1-arenesulfonyl-amino-2-isoborneolsulfonylaminocyclohexane-catalyzed addition of organozincs to ketones
Fulltext Access 4 Pages 2005
Instructions to contributors
Fulltext Access 4 Pages 2005
Asymmetric synthesis of α-methoxyarylacetic acid derivatives
Fulltext Access 4 Pages 2005
Improved catalytic asymmetric carbon–carbon bond formation using combinations of chiral and achiral monodentate ligands
Fulltext Access 4 Pages 2005
Instructions to contributors
Fulltext Access 4 Pages 2005
Furanoside thioether-phosphinite ligands for Rh-catalyzed asymmetric hydrosilylation of ketones
Fulltext Access 4 Pages 2005
Enzymatic desymmetrization of 2-amino-2-methyl-1,3-propanediol: asymmetric synthesis of (S)-N-Boc-N,O-isopropylidene-α-methylserinal and (4R)-methyl-4-[2-(thiophen-2-yl)ethyl]oxazolidin-2-one
Fulltext Access 4 Pages 2005
Asymmetric conjugate addition of metal alkyl reagents catalyzed by copper complexes with BINPO: a hemilabile P,O-heterobidentate axially chiral ligand
Fulltext Access 4 Pages 2005
‘Green’ synthesis of important pharmaceutical building blocks: enzymatic access to enantiomerically pure α-chloroalcohols
Fulltext Access 4 Pages 2005
A new chemoenzymatic synthesis of d-cloprostenol
Fulltext Access 4 Pages 2005
Catalytic enantioselective Michael addition in the synthesis of α-aminophosphonates
Fulltext Access 4 Pages 2005
Instructions to contributors
Fulltext Access 4 Pages 2005
Chemoenzymatic formal total synthesis of (−)-bestatin
Fulltext Access 4 Pages 2005
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