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Daneshyari Drug Discovery Journas Latest Articles

Drug Discovery Research Articles

Local inner-ear drug delivery and pharmacokinetics
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Genes for rheumatoid arthritis offer new insights into disease mechanisms
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Akt-directed metabolic alterations in cancer
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Krebs cycle enzymes as tumor suppressors
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Akt, hexokinase, mTOR: Targeting cellular energy metabolism for cancer therapy
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Allogeneic graft-versus-tumor effects: Mechanistic insights and therapeutic promise
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Botanical immunodrugs: scope and opportunities
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Functional genomics using high-throughput RNA interference
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Histone deacetylase inhibitors: new drugs for the treatment of inflammatory diseases?
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'The 39 steps' in gene expression profiling: critical issues and proposed best practices for microarray experiments
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Laser microdissection in CNS research
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Assessment of the feasibility of oral controlled release in an exploratory development setting
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Therapeutics of hearing loss: expectations vs reality
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S-Glutathiolation in redox-sensitive signaling
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Compounds for the prevention and treatment of noise-induced hearing loss
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Tinnitus: neurobiological substrates
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Metabolomics: from pattern recognition to biological interpretation
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Measurements of binding thermodynamics in drug discovery
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Drug design using the example of the complement system inhibitors' development
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High-throughput target discovery using cell-based genetics
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Targeting DHFR in parasitic protozoa
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Thalidomide as a novel therapeutic agent: new uses for an old product
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Global properties of biological networks
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From genome to antivirals: SARS as a test tube
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Strategies for producing faster acting antidepressants
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Information extraction technologies for the life science industry
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Cholesteryl ester transfer protein inhibition and the treatment of metabolic syndrome
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Cell transplantation for the treatment of heart failure
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L-selectin in inflammation, infection and immunity
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Capillary electrophoresis technologies for screening in drug discovery
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G-protein-coupled receptor screening technologies
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Ion channel screening technologies today
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Physiology-based pharmacokinetic modeling: ready to be used
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Molecular motors as drug delivery vehicles
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Subcutaneous drug delivery and the role of the lymphatics
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Vesicles as a tool for transdermal and dermal delivery
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Performance-driven, pulmonary delivery of systemically acting drugs
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Phospho-specific flow cytometry in drug discovery
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Phenotype-first screening for the identification of novel drug targets
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Managing genomic and proteomic knowledge
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Experimental autoimmune encephalomyelitis: A heterogeneous group of animal models to study human multiple sclerosis
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Chronic models of airway inflammation, mucus hypersecretion and remodelling
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Ectodermal dysplasia: Skinny models on the catwalk
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Models of congenital deafness: Mouse and zebrafish
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Role of Alzheimer's disease models in designing and testing experimental therapeutics
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Models of insulin signalling and longevity
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Models of anorexia
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Metabolic perturbations in the diabetic heart: Mechanisms and molecular targets
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AMPK - A pivotal rheostat in the control of cardiac metabolism
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Inflammatory mechanisms in vascular disease
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Characterising neural representation in terms of the dynamics of cell membrane potential activity: a control theoretic approach using differential geometry
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Mechanisms of disease: Atypical familial mycobacteriosis
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Mechanisms of neuronal degeneration after ischemic stroke - Emerging targets for novel therapeutic strategies
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Mechanisms in myasthenia gravis
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Predicting protein druggability
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Significance of release technology in tissue engineering
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Pitch detection of dynamic iterated rippled noise by humans and a modified auditory model
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Spike encoding mechanisms in the sound localization pathway
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A model of visual backward masking
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Identification of development and autonomic nerve activity from heart rate variability in preterm infants
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On the dynamics of a pair of coupled neurons subject to alternating input rates
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Emergence of oscillations and spatio-temporal coherence states in a continuum-model of excitatory and inhibitory neurons
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What is signal and what is noise in the brain?
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Lessons from autoimmune lymphoproliferative syndrome
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Synaptic modifications depend on synapse location and activity: a biophysical model of STDP
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Aging: gene silencing or gene activation?
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The role of lipoprotein (a) in pregnancies complicated by pre-eclampsia
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Nutraceutical resources for diabetes prevention - an update
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Iminium metabolite mechanism for nicotine toxicity and addiction: Oxidative stress and electron transfer
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Potentiation of immunological tolerance induction in adult mice by co-administration of pooled normal IgG and oral tolerogens: a potential therapeutic approach for autoimmune diseases
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Alzheimer disease is substantially preventable in the United States - review of risk factors, therapy, and the prospects for an expert software system
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Endogenous psychoactive tryptamines reconsidered: an anxiolytic role for dimethyltryptamine
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T waves are independently generated in both right and left ventricles: The clinically recorded T is a summation of two separate repolarizations, and is thus always biventricular
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A theory of blindsight - The anatomy of the unconscious: A proposal for the koniocellular projections and intralaminar thalamus
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Transient global amnesia may be caused by cerebral vein thrombosis
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Investigating Wnt signaling: a chemogenomic safari
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Using imaging biomarkers to accelerate drug development and clinical trials
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Bioinformatic methods for integrating whole-genome expression results into cellular networks
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Incretin mimetics and DPP-IV inhibitors for the treatment of type 2 diabetes
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FT-ICR mass spectrometry in the drug discovery process
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cGMP-dependent protein kinases in drug discovery
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The transcriptome's drugable frequenters
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Kinomics: characterizing the therapeutically validated kinase space
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Analyzing and mining image databases
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Combinatorial biomarkers: From early toxicology assays to patient population profiling
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Using microarray gene signatures to elucidate mechanisms of antibiotic action and resistance
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BiTEs: bispecific antibody constructs with unique anti-tumor activity
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Beyond annotation transfer by homology: novel protein-function prediction methods to assist drug discovery
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Asymmetric dimethylarginine: A molecule responsible for the coexistence of insulin resistance and atherosclerosis via dual nitric oxide synthase inhibition
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Can smooth muscle represent a useful target for the treatment of rapid ejaculation?
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PEGylation, successful approach to drug delivery
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High throughput P450 inhibition screens in early drug discovery
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Organotypic cultures as tools for functional screening in the CNS
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Role of mutational bias and natural selection on genome-wide nucleotide bias in prokaryotic organisms
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Simulation of rat behavior by a reinforcement learning algorithm in consideration of appearance probabilities of reinforcement signals
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The effect of species models on estimates of within-lineage variation in integration
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Automated derivation and refinement of sequence length patterns for protein sequences using evolutionary computation
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Why does the mammalian red blood cell have aquaporins?
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Cancer vaccines: The next generation
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Molecular mechanisms of human prion diseases
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