Synthesis and evaluation of phenylalanine-derived trifluoromethyl ketones for peptide-based oxidation catalysis Fulltext Access 4 Pages 2016
Synthesis of a norcantharidin-tethered guanosine: Protein phosphatase-1 inhibitors that change alternative splicing Fulltext Access 4 Pages 2016
Oxidative rearrangement strategy for synthesis of 2,4,5-trisubstituted oxazoles utilizing hypervalent iodine reagent Fulltext Access 5 Pages 2016
A red-emitting fluorescent probe for biothiols detection with a large Stokes shift Fulltext Access 5 Pages 2016
Reduction of diphenylacetylene using Al powder in the presence of noble metal catalysts in water Fulltext Access 5 Pages 2016
Base-catalyzed hydrogen–deuterium exchange and dehalogenation reactions of 1,2,3-triazole derivatives Fulltext Access 5 Pages 2016
Ionic liquids as a reusable media for copper catalysis. Green access to alkenes using catalytic olefination reaction Fulltext Access 5 Pages 2016
Synthesis, photophysical and electrochemical properties of symmetric silicon-linked coumarin-oxadiazole derivatives Fulltext Access 5 Pages 2016
Direct synthesis of thiophosphates by reaction of diphenylphosphine oxide with sulfonyl chlorides Fulltext Access 5 Pages 2016
Herbivore-induced volatile organic compounds emitted by maize: Electrophysiological responses in Spodoptera frugiperda females Fulltext Access 5 Pages 2016
Cytotoxic and antimalarial constituents from the roots of Toddalia asiatica Fulltext Access 5 Pages 2016
Synthesis and enantiomeric recognition studies of optically active 5,5-dioxophenothiazine bis(urea) and bis(thiourea) derivatives Fulltext Access 5 Pages 2016
Development of curcumin–cyclodextrin/cellulose nanocrystals complexes: New anticancer drug delivery systems Fulltext Access 5 Pages 2016
Synthesis, anti-inflammatory, ulcerogenic and cyclooxygenase activities of indenopyrimidine derivatives Fulltext Access 5 Pages 2016
Synthesis, antimicrobial activity of Schiff base compounds of cinnamaldehyde and amino acids Fulltext Access 5 Pages 2016
The semi-synthesis of novel andrographolide analogues and anti-influenza virus activity evaluation of their derivatives Fulltext Access 5 Pages 2016
Carbamate substituted 2-amino-4,6-diphenylpyrimidines as adenosine receptor antagonists Fulltext Access 5 Pages 2016
Design and synthesis of sarolaner, a novel, once-a-month, oral isoxazoline for the control of fleas and ticks on dogs Fulltext Access 5 Pages 2016
Discovery of boronic acid-based fluorescent probes targeting amyloid-beta plaques in Alzheimer’s disease Fulltext Access 5 Pages 2016
Carbon nanodots as molecular scaffolds for development of antimicrobial agents Fulltext Access 5 Pages 2016
Synthesis of novel ethyl 1-ethyl-6-fluoro-7-(fatty amido)-1,4-dihydro-4-oxoquinoline-3-carboxylate derivatives and their biological evaluation Fulltext Access 5 Pages 2016
Design and evaluation of novel oxadiazole derivatives as potential prostate cancer agents Fulltext Access 5 Pages 2016
Development of novel proteasome inhibitors based on phthalazinone scaffold Fulltext Access 5 Pages 2016
Synthesis, structure and antimicrobial evaluation of a new gossypol triazole conjugates functionalized with aliphatic chains and benzyloxy groups Fulltext Access 5 Pages 2016
Design, synthesis and biological evaluation of photoaffinity probes of antiangiogenic homoisoflavonoids Fulltext Access 5 Pages 2016
Synthesis and biological evaluation of matrine derivatives as anti-hepatocellular cancer agents Fulltext Access 5 Pages 2016
Self-assembling tryptophan-based designer peptides as intracellular delivery vehicles Fulltext Access 5 Pages 2016
Synthesis and biological activity of diisothiocyanate-derived mercapturic acids Fulltext Access 5 Pages 2016
Synthesis and fluorescent study of 5-phenyl furocoumarin derivatives as vasodilatory agents Fulltext Access 5 Pages 2016
Bifunctional primary amine 2-aminobenzimidazole organocatalyst anchored to trans-cyclohexane-1,2-diamine in enantioselective conjugate additions of aldehydes Fulltext Access 5 Pages 2016
Synthesis of a new inhibitor of breast cancer resistance protein with significantly improved pharmacokinetic profiles Fulltext Access 5 Pages 2016
Design, synthesis and in vivo screening of some novel quinazoline analogs as anti-hyperlipidemic and hypoglycemic agents Fulltext Access 5 Pages 2016
Increase of rutin antioxidant activity by generating Maillard reaction products with lysine Fulltext Access 5 Pages 2016
Synthesis and biological evaluation of aryloxyacetamide derivatives as neuroprotective agents Fulltext Access 5 Pages 2016
New ligands of the ghrelin receptor based on the 1,2,4-triazole scaffold by introduction of a second chiral center Fulltext Access 5 Pages 2016
(7-Diethylaminocoumarin-4-yl)methyl ester of suberoylanilide hydroxamic acid as a caged inhibitor for photocontrol of histone deacetylase activity Fulltext Access 5 Pages 2016
Novel method of simultaneous multiple immunogold localization on resin sections in high resolution scanning electron microscopy Fulltext Access 5 Pages 2016
Surprising lack of liposome-induced complement activation by artificial 1,3-diamidophospholipids in vitro Fulltext Access 5 Pages 2016
A cell-based approach to characterize antimicrobial compounds through kinetic dose response Fulltext Access 5 Pages 2016
Design and synthesis of novel hybrid sydnonimine and prodrug useful for glaucomatous optic neuropathy Fulltext Access 5 Pages 2016
One-pot synthesis and antifungal activity against plant pathogens of quinazolinone derivatives containing an amide moiety Fulltext Access 5 Pages 2016
Synthesis and docking studies of pyrazine–thiazolidinone hybrid scaffold targeting dormant tuberculosis Fulltext Access 5 Pages 2016
Rational design and synthesis of novel anti-prostate cancer agents bearing a 3,5-bis-trifluoromethylphenyl moiety Fulltext Access 5 Pages 2016
Synthesis of lignan conjugates via cyclopropanation: Antimicrobial and antioxidant studies Fulltext Access 5 Pages 2016
Synthesis and cytotoxic activities of semisynthetic zearalenone analogues Fulltext Access 5 Pages 2016
Design, synthesis, and evaluation of water-soluble morpholino-decorated paclitaxel prodrugs with remarkably decreased toxicity Fulltext Access 5 Pages 2016
An evolved oxazolidinone with selective potency against Mycobacterium tuberculosis and gram positive bacteria Fulltext Access 5 Pages 2016
Synthesis, characterization and anti-cancer activity of a peptide nucleolipid bioconjugate Fulltext Access 5 Pages 2016
Identification of new quinic acid derivatives as histone deacetylase inhibitors by fluorescence-based cellular assay Fulltext Access 5 Pages 2016
The natural flavone fukugetin as a mixed-type inhibitor for human tissue kallikreins Fulltext Access 5 Pages 2016
Carbohydrate-based inducers of cellular stress for targeting cancer cells Fulltext Access 5 Pages 2016
Anti-inflammatory and antioxidant properties of a novel resveratrol–salicylate hybrid analog Fulltext Access 5 Pages 2016
Antibacterial and antifungal activities of 2,3-pyrrolidinedione derivatives against oral pathogens Fulltext Access 5 Pages 2016
Functional foldamers that target bacterial membranes: The effect of charge, amphiphilicity and conformation Fulltext Access 5 Pages 2016
Incorporation of fluorophore–cholesterol conjugates into liposomal and mycobacterial membranes Fulltext Access 5 Pages 2016
Synthesis and asymmetric resolution of a dopaminergic compound: 2-amino-5-methoxyindane Fulltext Access 5 Pages 2016
Synthesis and study of the structural properties of oxa[5]helicene derivatives Fulltext Access 5 Pages 2016
A chiral, bis-anthraquinone-bridged cyclophane with a large specific rotation Fulltext Access 5 Pages 2016
Chiral copper-catalyzed asymmetric monoarylation of vicinal diols with diaryliodonium salts Fulltext Access 5 Pages 2016
Pyridazinone substituted benzenesulfonamides as potent carbonic anhydrase inhibitors Fulltext Access 5 Pages 2016
Biological evaluation and molecular docking studies of new curcuminoid derivatives: Synthesis and characterization Fulltext Access 5 Pages 2016
Optimization of isoxazoline amide benzoxaboroles for identification of a development candidate as an oral long acting animal ectoparasiticide Fulltext Access 5 Pages 2016
Synthesis and anti-proliferative activity of fluoro-substituted chalcones Fulltext Access 5 Pages 2016
Sequential one-pot synthesis of bis(indolyl)glyoxylamides: Evaluation of antibacterial and anticancer activities Fulltext Access 5 Pages 2016
Quinazolinones–Phenylquinoxaline hybrids with unsaturation/saturation linkers as novel anti-proliferative agents Fulltext Access 5 Pages 2016
Solubility-driven lead optimisation: Recent examples and personal perspectives Fulltext Access 5 Pages 2016
Synthesis, biological evaluation and molecular docking of 2-phenyl-benzo[d]oxazole-7-carboxamide derivatives as potential Staphylococcus aureus Sortase A inhibitors Fulltext Access 5 Pages 2016
Cationic lioposomes with folic acid as targeting ligand for gene delivery Fulltext Access 5 Pages 2016
Antioxidant properties of thio-caffeine derivatives: Identification of the newly synthesized 8-[(pyrrolidin-1-ylcarbonothioyl)sulfanyl]caffeine as antioxidant and highly potent cytoprotective agent Fulltext Access 5 Pages 2016
Synthesis and evaluation of novel 1,2,3-triazole-based acetylcholinesterase inhibitors with neuroprotective activity Fulltext Access 5 Pages 2016
Polycyclic amines as chloroquine resistance modulating agents in Plasmodium falciparum Fulltext Access 5 Pages 2016
Synthesis and activity of benzimidazole-1,3-dioxide inhibitors of separase Fulltext Access 5 Pages 2016
Synthesis and in vitro evaluation of water-soluble 1,4-diphenethylpiperazine analogs as novel inhibitors of the vesicular monoamine transporter-2 Fulltext Access 5 Pages 2016
Design, synthesis, and protein methyltransferase activity of a unique set of constrained amine containing compounds Fulltext Access 5 Pages 2016
Development of indole sulfonamides as cannabinoid receptor negative allosteric modulators Fulltext Access 5 Pages 2016
Suppression of store overload-induced calcium release by hydroxylated metabolites of carvedilol Fulltext Access 5 Pages 2016
Diversification of edaravone via palladium-catalyzed hydrazine cross-coupling: Applications against protein misfolding and oligomerization of beta-amyloid Fulltext Access 5 Pages 2016
Synthesis and biological evaluation of a novel artesunate–podophyllotoxin conjugate as anticancer agent Fulltext Access 5 Pages 2016
Synthesis, crystal structures, molecular docking, and in vitro biological activities of transition metals with 4-(2,3-dichlorophenyl)piperazine-1-carboxylic acid Fulltext Access 5 Pages 2016