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Daneshyari Pharmaceutical Science Journas Latest Articles

Pharmaceutical Science Research Articles

Solid lipid nanoparticles for pulmonary delivery of insulin
Fulltext Access 12 Pages 2008
Effect of Nonsteroidal Anti-Inflammatory Drugs on the Cellular Membrane Fluidity
Fulltext Access 12 Pages 2008
Calorimetric Relaxation and the Glass-Liquid Temperature Range of Acetaminophen-Nifedipine Alloys
Fulltext Access 12 Pages 2008
Lateral and Rotational Mobility of Some Drug Molecules in a Poly(Ethylene Glycol) Diacrylate Hydrogel and the Effect of Drug-Cyclodextrin Complexation
Fulltext Access 12 Pages 2008
Design and Characterization of a New Miniaturized Rotating Disk Equipment for In Vitro Dissolution Rate Studies
Fulltext Access 12 Pages 2008
Drug Release Phenomena Within a Hydrophobic Starch Acetate Matrix: FTIR Mapping of Tablets After In Vitro Dissolution Testing
Fulltext Access 12 Pages 2008
Process Analytical Technology: Nondestructive Evaluation of Cyclosporine A and Phospholipid Solid Dispersions by Near Infrared Spectroscopy and Imaging
Fulltext Access 12 Pages 2008
Parenteral microemulsions: An overview
Fulltext Access 12 Pages 2008
Mechanistic Study of Electroosmotic Transport Across Hydrated Nail Plates: Effects of pH and Ionic Strength
Fulltext Access 12 Pages 2008
Correlation of Annealing with Chemical Stability in Lyophilized Pharmaceutical Glasses
Fulltext Access 12 Pages 2008
PLGA nanospheres for the ocular delivery of flurbiprofen: Drug release and interactions
Fulltext Access 12 Pages 2008
Effect of O-acylmenthol on transdermal delivery of drugs with different lipophilicity
Fulltext Access 12 Pages 2008
Determination of intraliposomal pH and its effect on membrane partitioning and passive loading of a hydrophobic camptothecin, DB-67
Fulltext Access 12 Pages 2008
Physicochemical, in silico and in vivo evaluation of a danazol–β-cyclodextrin complex
Fulltext Access 12 Pages 2008
Development of a reaction-limited model of dissolution: Application to official dissolution tests experiments
Fulltext Access 12 Pages 2008
Allosteric kinetics of human carboxylesterase 1: Species differences and interindividual variability
Fulltext Access 12 Pages 2008
Carboxylated high amylose starch as pharmaceutical excipients: Structural insights and formulation of pancreatic enzymes
Fulltext Access 12 Pages 2008
Moisture sorption, compressibility and caking of lactose polymorphs
Fulltext Access 12 Pages 2008
Using a Modified Shepards Method for Optimization of a Nanoparticulate Cyclosporine A Formulation Prepared by a Static Mixer Technique
Fulltext Access 12 Pages 2008
A new biocompatible nanoparticle delivery system for the release of fibrinolytic drugs
Fulltext Access 12 Pages 2008
State of the art and perspectives for the delivery of antisense oligonucleotides and siRNA by polymeric nanocarriers
Fulltext Access 12 Pages 2008
Cospray-dried unfractionated heparin with L-leucine as a dry powder inhaler mucolytic for cystic fibrosis therapy
Fulltext Access 12 Pages 2008
Use of hydrodynamic flow focusing for the generation of biodegradable camptothecin‐loaded polymer microspheres
Fulltext Access 12 Pages 2008
Are pharmaceutics really going supercritical?
Fulltext Access 12 Pages 2008
High bioavailability from nebulized itraconazole nanoparticle dispersions with biocompatible stabilizers
Fulltext Access 12 Pages 2008
Non-destructive acoustic defect detection in drug tablets
Fulltext Access 12 Pages 2008
Top-down production of drug nanocrystals: Nanosuspension stabilization, miniaturization and transformation into solid products
Fulltext Access 12 Pages 2008
Efficacy of the Injectable Calcium Phosphate Ceramics Suspensions Containing Magnesium, Zinc and Fluoride on the Bone Mineral Deficiency in Ovariectomized Rats
Fulltext Access 12 Pages 2008
Oral Delivery of Antisense Oligonucleotides in Man
Fulltext Access 12 Pages 2008
On the Volume of Distribution at Steady State and Its Relationship With Two‐Compartmental Models
Fulltext Access 12 Pages 2008
Dirhenium decacarbonyl-loaded PLLA nanoparticles: Influence of neutron irradiation and preliminary in vivo administration by the TMT technique
Fulltext Access 12 Pages 2008
Injectable block copolymer hydrogels for sustained release of a PEGylated drug
Fulltext Access 12 Pages 2008
Enhancement of dissolution rate and bioavailability of aceclofenac: A chitosan-based solvent change approach
Fulltext Access 12 Pages 2008
Combination Particles Containing Salmeterol Xinafoate and Fluticasone Propionate: Formulation and Aerodynamic Assessment
Fulltext Access 12 Pages 2008
Clusterin antisense complexed with chitosan for controlled intratumoral delivery
Fulltext Access 12 Pages 2008
Modifications in Low-Density Lipoprotein Receptor Expression Affects Cyclosporin A Cellular Uptake and Cytotoxicity
Fulltext Access 12 Pages 2008
Effect of Anesthetic Structure on Inhalation Anesthesia: Implications for the Mechanism
Fulltext Access 12 Pages 2008
Biowaiver Monographs for Immediate Release Solid Oral Dosage Forms: Pyrazinamide**
Fulltext Access 12 Pages 2008
Passive Transfer of Polyethylene Glycol to Liposomal-Recombinant Human FVIII Enhances its Efficacy in a Murine Model for Hemophilia A
Fulltext Access 12 Pages 2008
Correlation Between Molecular Mobility and Crystal Growth of Amorphous Phenobarbital and Phenobarbital with Polyvinylpyrrolidone and L‐proline
Fulltext Access 12 Pages 2008
Enhanced antitumor activity of combinations of free and HPMA copolymer-bound drugs
Fulltext Access 12 Pages 2008
Quality by Design, Part I: Application of NIR Spectroscopy to Monitor Tablet Manufacturing Process
Fulltext Access 12 Pages 2008
Screening poly(ethyleneglycol) micro- and nanogels for drug delivery purposes
Fulltext Access 12 Pages 2008
Solubilization of hydrophobic drugs by methoxy poly(ethylene glycol)‐block‐polycaprolactone diblock copolymer micelles: Theoretical and experimental data and correlations
Fulltext Access 12 Pages 2008
Degradation of paclitaxel and related compounds in aqueous solutions I: Epimerization
Fulltext Access 12 Pages 2008
Characteristics of hydrogen bond formation between sugar and polymer in freeze‐dried mixtures under different rehumidification conditions and its impact on the glass transition temperature
Fulltext Access 12 Pages 2008
Wet granulation as innovative and fast method to prepare controlled release granules based on an ion‐exchange resin
Fulltext Access 12 Pages 2008
Topical Corticosteroids, Structure-Activity and the Glucocorticoid Receptor: Discovery and Development-A Process of ''Planned Serendipity''
Fulltext Access 12 Pages 2008
The effect of water solubility of solutes on their flux through human skin in vitro: A prodrug database integrated into the extended Flynn database
Fulltext Access 12 Pages 2008
Drug–polymer interaction and its significance on the physical stability of nifedipine amorphous dispersion in microparticles of an ammonio methacrylate copolymer and ethylcellulose binary blend
Fulltext Access 12 Pages 2008
Enhanced Efficiency of Thermally Targeted Taxanes Delivery in a Human Xenograft Model of Gastric Cancer
Fulltext Access 12 Pages 2008
Effects of repeated callbacks on response rate and nonresponse bias: Results from a 17-state pharmacy survey
Fulltext Access 13 Pages 2008
Rational Estimation of the Optimum Amount of Non‐Fibrous Disintegrant Applying Percolation Theory for Binary fast Disintegrating Formulation
Fulltext Access 13 Pages 2008
Silicone Elastomer Uptake Method for Determination of Free 1‐Alkyl‐2‐Pyrrolidone Concentration in Micelle and Hydroxypropyl‐β‐Cyclodextrin Systems Used in Skin Transport Studies
Fulltext Access 13 Pages 2008
A mechanistic Study on the Chemical and Enzymatic Degradation of PEG‐Oligo(ε‐caprolactone) Micelles
Fulltext Access 13 Pages 2008
Release Kinetics of Benzoic Acid and its Sodium Salt From a Series of Poly(N‐Isopropylacrylamide) Matrices with Various Percentage Crosslinking
Fulltext Access 13 Pages 2008
Effect of P‐Glycoprotein Expression Levels on the Concentration‐Dependent Permeability of Drugs to the Cell Membrane
Fulltext Access 13 Pages 2008
The surface characterisation and comparison of two potential sub-micron, sugar bulking excipients for use in low-dose, suspension formulations in metered dose inhalers
Fulltext Access 13 Pages 2008
Compaction properties, drug release kinetics and fronts movement studies from matrices combining mixtures of swellable and inert polymers: Effect of HPMC of different viscosity grades
Fulltext Access 13 Pages 2008
How to achieve sustained and complete protein release from PLGA-based microparticles?
Fulltext Access 13 Pages 2008
Selectivity of folate conjugated polymer micelles against different tumor cells
Fulltext Access 13 Pages 2008
Pharmacokinetics of raloxifene in male Wistar–Hannover rats: Influence of complexation with hydroxybutenyl-beta-cyclodextrin
Fulltext Access 13 Pages 2008
Pilot study of a hierarchical Bayes method for utility estimation in a choice-based conjoint analysis of prescription benefit plans including medication therapy management services
Fulltext Access 13 Pages 2008
A modified model of pharmacists' job stress: The role of organizational, extra-role, and individual factors on work-related outcomes
Fulltext Access 13 Pages 2008
Effect of Thermodynamic Activities of the Unionized and Ionized Species on Drug Flux across Buccal Mucosa
Fulltext Access 13 Pages 2008
Physicochemical Characterisation of a Novel Thermogelling Formulation for Percutaneous Penetration of 5-Aminolevulinic Acid
Fulltext Access 13 Pages 2008
Functionality of magnesium stearate derived from bovine and vegetable sources: Dry granulated tablets
Fulltext Access 13 Pages 2008
Biowaiver Monographs for Immediate Release Solid Oral Dosage Forms: Aciclovir
Fulltext Access 13 Pages 2008
Spontaneous Crystallinity Loss of Drugs in the Disordered Regions of Poly(Ethylene Oxide) in the Presence of Water
Fulltext Access 13 Pages 2008
Role of Agglomeration in the Dispersion of Salmeterol Xinafoate from Mixtures for Inhalation with Differing Drug to Fine Lactose Ratios
Fulltext Access 13 Pages 2008
Potential Use of Polyamidoamine Dendrimer/α-Cyclodextrin Conjugate (Generation 3, G3) as a Novel Carrier for Short Hairpin RNA-Expressing Plasmid DNA
Fulltext Access 13 Pages 2008
Characterization of the “hygroscopic” properties of active pharmaceutical ingredients
Fulltext Access 13 Pages 2008
A Comparison of the Effect of Chitosan and Chitosan-Coated Vesicles on Monolayer Integrity and Permeability Across Caco-2 and 16HBE14o-Cells
Fulltext Access 13 Pages 2008
An Investigation into the Mechanisms of Drug Release From Taste-Masking Fatty Acid Microspheres
Fulltext Access 13 Pages 2008
Site-specific drug delivery to the middle-to-lower region of the small intestine reduces food-drug interactions that are responsible for low drug absorption in the fed state
Fulltext Access 13 Pages 2008
Stabilization of Low Glass Transition Temperature Indomethacin Formulations: Impact of Polymer-Type and Its Concentration
Fulltext Access 13 Pages 2008
Inhibition of Aggregation of Aluminum Hydroxide Adjuvant During Freezing and Drying
Fulltext Access 13 Pages 2008
Pharmacokinetic/Pharmacodynamic Modeling of Corticosterone Suppression and Lymphocytopenia by Methylprednisolone in Rats
Fulltext Access 13 Pages 2008
N-in-1 Dosing Pharmacokinetics in Drug Discovery: Experience, Theoretical and Practical Considerations
Fulltext Access 13 Pages 2008
Quality-by-Design (QbD): Effects of Testing Parameters and Formulation Variables on the Segregation Tendency of Pharmaceutical Powder Measured by the ASTM D 6940-04 Segregation Tester
Fulltext Access 13 Pages 2008
Role of Mechanical Stress in Crystallization and Relaxation Behavior of Amorphous Indomethacin
Fulltext Access 13 Pages 2008
Moisture Sorption and Permeability Characteristics of Polymer Films: Implications for Their Use as Barrier Coatings for Solid Dosage Forms Containing Hydrolyzable Drug Substances
Fulltext Access 13 Pages 2008
Structure-Permeability Relationship Analysis of the Permeation Barrier Properties of the Stratum Corneum and Viable Epidermis/Dermis of Rat Skin
Fulltext Access 13 Pages 2008
Ordering and disordering of molecular solids upon mechanical milling: The case of fananserine
Fulltext Access 13 Pages 2008
Effect of propylene glycol on ibuprofen absorption into human skin in vivo
Fulltext Access 13 Pages 2008
Porcine Vagina Ex Vivo as a Model for Studying Permeability and Pathogenesis in Mucosa
Fulltext Access 13 Pages 2008
PLGA Nanoparticles for Oral Delivery of Hydrophobic Drugs: Influence of Organic Solvent on Nanoparticle Formation and Release Behavior In Vitro and In Vivo Using Estradiol as a Model Drug
Fulltext Access 13 Pages 2008
Contribution of Variable Domains to the Stability of Humanized IgG1 Monoclonal Antibodies
Fulltext Access 13 Pages 2008
Phosphatidylserine Containing Liposomes Reduce Immunogenicity of Recombinant Human Factor VIII (rFVIII) in a Murine Model of Hemophilia A*
Fulltext Access 13 Pages 2008
The Development of Thermally Assisted Particle Manipulation and Thermal Nanointeraction Studies as a Means of Investigating Drug‐polymer Interactions
Fulltext Access 13 Pages 2008
Fluoxetine Pretreatment Effects Pharmacokinetics of 3,4‐Methylenedioxymethamphetamine (MDMA, ECSTASY) in Rat
Fulltext Access 13 Pages 2008
Effects of E. Coli lipopolysaccharide on the pharmacokinetics of ipriflavone and its metabolites, M1 and M5, after intravenous and oral administration of ipriflavone to rats: Decreased metabolism of ipriflavone due to decreased expression of hepatic CYP1A
Fulltext Access 13 Pages 2008
Correlation between Chemical Reactivity and the Hammett Acidity Function in Amorphous Solids Using Inversion of Sucrose as a Model Reaction
Fulltext Access 13 Pages 2008
Development of a liquid enzyme-based ceruminolytic product
Fulltext Access 13 Pages 2008
Peptide-mediated lipofection is governed by lipoplex physical properties and the density of surface-displayed amines
Fulltext Access 13 Pages 2008
pH-Dependent Interactions of Indinavir and Lipids in Nanoparticles and Their Ability to Entrap a Solute
Fulltext Access 13 Pages 2008
Evaluation of Hydrophilic Permeant Transport Parameters in the Localized and Non-Localized Transport Regions of Skin Treated Simultaneously With Low-Frequency Ultrasound and Sodium Lauryl Sulfate
Fulltext Access 13 Pages 2008
Transungual Iontophoretic Transport of Polar Neutral and Positively Charged Model Permeants: Effects of Electrophoresis and Electroosmosis
Fulltext Access 13 Pages 2008
Interactions of pluronic block copolymers on P‐gp efflux activity: Experience with HIV‐1 protease inhibitors
Fulltext Access 13 Pages 2008
Changes in metformin pharmacokinetics after intravenous and oral administration to rats with short‐term and long‐term diabetes induced by streptozotocin
Fulltext Access 13 Pages 2008
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