Keywords: دامنه خارج سلولی; GHR; growth hormone receptor; GHRtm; recombinant fragment GHR254-294; JAK2; Janus kinase 2; RTK; receptor tyrosine kinase; TMD; transmembrane domain; ECD; extracellular domain; ICD; intracellular domain; JM; juxtamembrane; ecJM; extracellular juxtamembr
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Keywords: دامنه خارج سلولی; aa; amino acid; ADMA; asymmetric dimethylarginine; AF; atrial fibrillation; ALP; alkaline phosphatase; BMI; body mass index; BMP; bone morphogenetic protein; Cys; cysteine; CAD; coronary artery disease; CKD; chronic kidney disease; CRD; cysteine rich doma
Keywords: دامنه خارج سلولی; Ache; acetylcholinesterase; AD; Alzheimer's disease; Adra2a, Adra2b, Adra1b; adrenoceptor alpha 2a, alpha 2b, beta 1; Akt1; Akt serine/threonine protein kinase 1/protein kinase B; ApoE; apolipoprotein E; Bche; butyrylcholinesterase; BDNF; brain derived ne
Keywords: دامنه خارج سلولی; 2â²-F-Py; 2â²-fluoro-pyrimidines; 3D; three-dimensional; 3WJ; three-way junction; AMD; age-related macular degeneration; AuNPs; gold nanoparticles; BBB; blood-brain barrier; Bcl-2; B-cell lymphoma 2; BM; bone marrow; CCL2; chemokine C-C motif ligand 2;
Keywords: دامنه خارج سلولی; AC; adenylate cyclase; Actn4; α-Actinin-4; ARF6; ADP-ribosylation factor 6; ATD; amino terminal domain; CAIN; calcineurin inhibitor protein; CaM; calmodulin; CaMKII; Ca2+/calmodulin-dependent protein kinase II; Cbln1; cerebellin 1 precursor; CC; coiled-c
Keywords: دامنه خارج سلولی; Myasthenia gravis; Nicotinic acetylcholine receptor; Immunoadsorption; Therapy; Experimental autoimmune myasthenia gravis; MG; myasthenia gravis; EAMG; experimental autoimmune MG; AChR; nicotinic acetylcholine receptor; ECD; extracellular domain; MIR; mai
Keywords: دامنه خارج سلولی; ACh; acetylcholine; α-BTX; α-bungarotoxin; Carb; carbamylcholine; Chol; cholesterol; ECD; extracellular domain; ELIC; Erwinia ligand-gated ion channel; GLIC; Gloebacter ligand-gated ion channel; nAChR; nicotinic acetylcholine receptor; PA; 1-palmitoyl-2
Keywords: دامنه خارج سلولی; BP; bitopic protein; RTK; receptor tyrosine kinase; TMD; transmembrane domain; JM; juxtamembrane; ECD; extracellular domain; ICD; intracellular domain; NMR; nuclear magnetic resonance; MD; molecular dynamics; LID; “ligand-induced dimerization” mechani
Keywords: دامنه خارج سلولی; 5HT3R; 5-hydroxytryptamine receptor, subtype 3; ATP; Adenosine triphosphate; BK; big potassium channels; Cho; cholesterol; CTD; C-terminal domain; ECD; extracellular domain; ELIC; Erwinia chrysanthemi ligand-gated ion channel; GABAAR; gamma-aminobutyric a
Keywords: دامنه خارج سلولی; 1,25-D3; 1,25-Dihydroxy vitamin D3; ACF; Aberrant crypt foci; AC; Adenylate cyclase; ADH; Autosomal dominant hypocalcaemia; CaSR; Calcium-sensing receptor; cAMP; Cyclic adenosine 3â²,5â²-monophosphate; Cai2+; Â Intracellular free ionised calcium; Cao2+;
Keywords: دامنه خارج سلولی; HCC; hepatocellular carcinoma; DDS; drug delivery system; ECM; extracellular matrix; MVD; microvessel density; EPR; enhanced permeability and retention; ASGP-R; asialoglycoprotein receptor; GPC3; glypican 3; HS chain; heparin sulfate chain; GA; glycyrrhet
Keywords: دامنه خارج سلولی; MG; myasthenia gravis; AChR; nicotinic acetylcholine receptor; ECD; extracellular domain; MIR; main immunogenic region; AChBP; acetylcholine binding protein; α-Btx; α-bungarotoxin.; Nicotinic acetylcholine receptor; Extracellular domain; Myasthenia grav
Keywords: دامنه خارج سلولی; AFM; atomic force microscopy; BSA; bovine serum albumin; CHO-cells; Chinese hamster ovary cells; DMEM; Dulbecco's modified Eagle's medium; Dsc; desmocollin; Dsg; desmoglein; E-Cadherin; epithelial cadherin; EC; extracellular domain; EGTA; ethylene glycol
Keywords: دامنه خارج سلولی; ECD; extracellular domain; ER; endoplasmic reticulum; FL; full-length; (P)RR; (pro)renin receptor; s(P)RR; soluble (pro)renin receptor; (Pro)renin receptor; ATP6AP2; Dimerization; Extracellular domain; Retention;
Stoichiometry dependent inhibition of rat α3β4 nicotinic acetylcholine receptor by the ribbon isomer of α-conotoxin AuIB
Keywords: دامنه خارج سلولی; ACh; acetylcholine; AChBP; acetylcholine-binding protein; ECD; extracellular domain; gAuIB; globular AuIB; ICD; intracellular domain; nAChR; nicotinic acetylcholine receptor; rAuIB; ribbon AuIB; SAR; structure-activity relationship; TMD; transmembrane dom
Molecular and in silico analyses validates pathogenicity of homozygous mutations in the NPR2 gene underlying variable phenotypes of Acromesomelic dysplasia, type Maroteaux
Keywords: دامنه خارج سلولی; AMDM; Acromesomelic dysplasia, Maroteaux type; ECD; extracellular domain; GC; guanylate cyclase; CNP; C-type natriuretic peptide; PDB; protein databank; PDF; probability density function; DOPE; discrete optimized protein energy; MD; molecular dynamics; Hs
GLA supplementation regulates PHD2 mediated hypoxia and mitochondrial apoptosis in DMBA induced mammary gland carcinoma
Keywords: دامنه خارج سلولی; AA; arachidonic acid; AB; alveolar bud; AAA; aromatic amino acid; BCAA; branched chain amino acid; BSA; bovine serum albumin; BMRB; biological magnetic resonance databank; CEC; cuboidal epithelial cell; CPMG; carr-purcell-meiboom-gill; DMBA; 7, 12-d
Dually modified transmembrane proteoglycans in development and disease
Keywords: دامنه خارج سلولی; ActR; activin type receptor; ALK; activin receptor like kinase; AV; atrioventricular cushion; BMP; bone morphogenetic protein; BMPR; bone morphogenetic protein receptor; C1; conserved domain 1; C2; conserved domain 2; Cdc42; control protein 42 homolog; CS
GABAA receptor: Positive and negative allosteric modulators
Keywords: دامنه خارج سلولی; γ-Aminobutyric acid type A receptors; Inhibitory neurotransmission; CNS depressant drug target; Anxiolytics/sedatives/general anesthetics; Ethanol; GABA; γ-aminobutyric acid; GABAAR; GABAA receptors; LGIC; ligand-gated ion channels; PLGIC; pentameric LG
Toll-receptor 9 gene in the black tiger shrimp (Penaeus monodon) induced the activation of the TLR-NF-κB signaling pathway
Keywords: دامنه خارج سلولی; Pm or P. monodon; Penaeus monodon; TLR; Toll-like receptor; PRR; pathogen recognition receptors; TIR; Toll/interleukin-1 receptor; ECD; extracellular domain; PAMP; Pathogen Associated Molecular Patterns; LRR; leucine-rich repeat; LRR-NT; leucine-rich repe
Identification of small molecule activators for ErbB 4 receptor to enhance oligodendrocyte regeneration by in silico approach
Keywords: دامنه خارج سلولی; ADMET; adsorption distribution metabolism excretion toxicity; BBB; blood brain barrier; BS; bioavailability score; CNS; central nervous system; CT; C-terminal tail; ECD; extracellular domain; EGF; epidermal growth factor; ESOL; estimated solubility; EV; E
Regulation of granulocyte colony-stimulating factor receptor-mediated granulocytic differentiation by C-mannosylation
Keywords: دامنه خارج سلولی; C-mannosylation; Glycosylation; Granulocyte colony-stimulating factor receptor (G-CSFR); Mass spectrometry; Myeloid differentiation; TSR; thrombospondin type 1 repeat; G-CSF; granulocyte colony-stimulating factor; G-CSFR; granulocyte colony-stimulating fa
HER2-targeted gold nanoparticles potentially overcome resistance to trastuzumab in gastric cancer
Keywords: دامنه خارج سلولی; Gold nanoparticle; Trastuzumab resistance; HER2; Gastric cancer; Autophagy; Tmab; trastuzumab; HER2; human epidermal growth factor receptor 2; AuNP; gold nanoparticle; ECD; extracellular domain; ADCC; antibody-dependent cellular cytotoxicity; PTEN; phosph
Evolutionary history of the podoplanin gene
Keywords: دامنه خارج سلولی; BLAST; Basic Local Alignment Search Tool; CT; cytoplasmic domain; EC; extracellular domain; NCBI; National Center for Biotechnology Information; PDPN; podoplanin; SRA; Sequence Read Archive; TAE; Tris Acetate-EDTA buffer; PCR; polymerase chain reaction; U
Tricyclic antidepressants inhibit hippocampal α7* and α9α10 nicotinic acetylcholine receptors by different mechanisms
Keywords: دامنه خارج سلولی; AChR; nicotinic acetylcholine receptor; ACh; acetylcholine; TCAs; tricyclic antidepressants; α-BTx; α-bungarotoxin; MLA; methyllycaconitine; RT; room temperature; IC50; ligand concentration that produces 50% inhibition (of binding or of agonist activati
Sequence defined antibodies improve the detection of cadherin 2 (N-cadherin) during zebrafish development
Keywords: دامنه خارج سلولی; mAb; monoclonal antibody; Cdh2; cadherin-2; zCdh2; zebrafish Cadherin-2; ECD; extracellular domain; Ig; immunoglobulin; CNS; central nervous system; crybb1; crystallin Beta B1; pac; parachute; Tg; transgenic; BAC; bacterial artificial chromosome; GFP; gre
Functional properties and mechanism of action of PPTQ, an allosteric agonist and low nanomolar positive allosteric modulator at GABAA receptors
Keywords: دامنه خارج سلولی; Ago-PAM; allosteric agonist and positive allosteric modulator; C/R; concentration-response; ECD; extracellular domain; FMP; FLIPR Membrane Potential Blue; GABA; γ-Aminobutyric acid; GABAAR; GABAA receptor; methaqualone; 2-methyl-3-(o-tolyl)-quinazolin-4(
Cell adhesion and matricellular support by astrocytes of the tripartite synapse
Keywords: دامنه خارج سلولی; β (Greek Small Letter Beta): 03B2; α (Greek Small Letter Alpha): 03B1; δ (Greek Small Letter Delta): 03B4; γ (Greek Small Letter Gamma): 03B3; ACM; astrocyte-conditioned medium; AMIGO; adhesion molecule with IG-like domain; AMOG; A Molecule On Glia; A
Mouse Model of Alagille Syndrome and Mechanisms of Jagged1 Missense Mutations
Keywords: دامنه خارج سلولی; Notch; Jagged1; Alagille; Heart; Liver; Kidney; Vertebrae; Development; ALGS; Alagille syndrome; ECD; extracellular domain; EGF; epidermal growth factor; FACS; fluorescence-activated cell sorting; GSEA; gene set enrichment analyses; HPA; Human Protein Atl
Genotype-functional-phenotype correlations in photoreceptor guanylate cyclase (GC-E) encoded by GUCY2D
Keywords: دامنه خارج سلولی; Cyclic GMP; Genotype-phenotype correlation; Guanylate cyclase; GUCY2D; Mutation; Photoreceptor; Retinal diseases; AAV; adeno-associated virus; ad; autosomal dominant; ar; autosomal recessive; BSP; bone spicule-like pigmentation; CCD; cyclase catalytic dom
Objective, domain-specific HER2 measurement in uterine and ovarian serous carcinomas and its clinical significance
Keywords: دامنه خارج سلولی; HER2; Intracellular domain; Extracellular domain; Serous carcinoma; Quantitative immunofluorescence; Targeted therapy;
Crystal structure of tissue factor in complex with antibody 10H10 reveals the signaling epitope
Keywords: دامنه خارج سلولی; CDR; complementarity determining region; CHES; N-cyclohexyl-2-aminoethanesulfonic acid; ECD; extracellular domain; EDTA; ethylenediaminetetraacetic acid; FVII; coagulation factor VII; FX; coagulation factor X; HEPES; 4-(2-hydroxyethyl)-1-piperazineethanes
Structural insights into the interaction of a monoclonal antibody and Nodal peptides by STD-NMR spectroscopy
Keywords: دامنه خارج سلولی; ActRIIA; activin type II receptor A; ActRIIB; activin type II receptor B; ALK; activin receptor-like kinase; CFC; Cripto-1/FLR1/cryptic; ECD; extracellular domain; EGF; epidermal growth factor; GEM; Group epitope mapping; mAb; monoclonal antibody; SMAD; S
Construction of high level prokaryotic expression and purification system of PD-L1 extracellular domain by using Escherichia coli host cell machinery
Keywords: دامنه خارج سلولی; PCR; polymerase chain reaction; ECD; extracellular domain; TM; trans-membrane; CD; cytoplasmic domain; PD-L1; programmed cell death ligand 1; PDL1-ECD; programmed cell death ligand 1- extracellular domain; ERS; enzyme restriction sites; Ori; origin of rep
Characterization of a reproducible rat EAMG model induced with various human acetylcholine receptor domains
Keywords: دامنه خارج سلولی; MG; myasthenia gravis; AChR; nicotinic acetylcholine receptor; ECD; extracellular domain; MIR; main immunogenic region; AChBP; acetylcholine binding protein; α-Btx; α-bungarotoxin; EAMG; experimental autoimmune myasthenia gravis; EMG; electromyography;
Functional characterization of two naturally occurring mutations V221G and T449N in the follicle stimulating hormone receptor
Keywords: دامنه خارج سلولی; Extracellular domain; FSH receptor; Naturally occurring mutations; Ovarian hyperstimulation syndrome; Primary amenorrhea;
Targeting GPNMB with glembatumumab vedotin: Current developments and future opportunities for the treatment of cancer
Keywords: دامنه خارج سلولی; AE; Adverse Event; α-MSH; alpha-Melanocyte Stimulating Hormone; ADC; Antibody-Drug Conjugate; ASPS; Alveolar Soft Part Sarcoma; ASPSCR1; Alveolar Soft Part Sarcoma Chromosome Region Candidate 1; BMP-2; Bone Morphogenetic Protein-2; BRK; Breast Tumor Kina
The effects of RAMPs upon cell signalling
Keywords: دامنه خارج سلولی; Receptor activity modifying protein; G protein-coupled receptor; Signalling; Trafficking; Coupling; AM; adrenomedullin; AMY; amylin; CaSR; calcium-sensing receptor; CGRP; calcitonin gene-related peptide; CHO; chinese hamster ovary; CLR; calcitonin recepto
Functional characterization of two prokaryotic pentameric ligand-gated ion channel chimeras - role of the GLIC transmembrane domain in proton sensing
Keywords: دامنه خارج سلولی; 5HT3R; serotonin receptor; α-BTX; α-bungarotoxin; AChBP; acetylcholine-binding protein; ECD; extracellular domain; ELIC; Erwinia ligand-gated ion channel; GLIC; Gloebacter ligand-gated ion channel; GlyR; glycine receptor; nAChR; nicotinic acetylcholine
The roles of subcellularly located EGFR in autophagy
Keywords: دامنه خارج سلولی; AMPK; AMP-activated protein kinase; ATG; autophagy-related; BCL2; B-cell lymphoma 2; BCL2L1; BCL2 like 1; BNIP3; BCL2/Adenovirus E1B-binding protein Nip3; CME; clathrin-mediated endocytosis; cytoSTAT3; cytoplasmic STAT3; Dsbs; double strand breaks; ECD; e
The role of carbohydrate component of recombinant α7 nicotinic acetylcholine receptor extracellular domain in its immunogenicity and functional effects of resulting antibodies
Keywords: دامنه خارج سلولی; α7 nicotinic acetylcholine receptor; Antibody; Carbohydrate component; Inflammation; Amyloid-beta; Alzheimer disease; nAChR; nicotinic acetylcholine receptor; Aβ; amyloid-beta; ECD; extracellular domain; LCH; Lens culinaris hemagglutinin; LPS; lipopolys
Original ArticleKeratinocytes/EpidermisMembrane-Tethered Intracellular Domain of Amphiregulin Promotes Keratinocyte Proliferation
Keywords: دامنه خارج سلولی; aa; amino acid; Ab; antibody; AREG; amphiregulin; CTD; C-terminal domain; DAPI; 4â²,6-diamidino-2-phenylindole; ECD; extracellular domain; EGFR; epidermal growth factor receptor; rh; recombinant human; sAREG; soluble/shed AREG; Tet; tetracycline;
Bupropion and its photoreactive analog (±)-SADU-3-72 interact with luminal and non-luminal sites at human α4β2 nicotinic acetylcholine receptors
Keywords: دامنه خارج سلولی; Human α4β2 nicotinic acetylcholine receptor; Bupropion; (±)-SADU-3-72; Molecular docking; Luminal and non-luminal sites; Ca2+ influx; AChR; nicotinic acetylcholine receptor; NCA; noncompetitive antagonist; (±)-BP; (±)-bupropion [(±)-2-(tert-butylami
Positive allosteric modulators of α7 nicotinic acetylcholine receptors affect neither the function of other ligand- and voltage-gated ion channels and acetylcholinesterase, nor β-amyloid content
Keywords: دامنه خارج سلولی; 5-HT; 5-hydroxytryptamine (serotonin); m5-HT3AR; murine serotonin type 3A receptor; AChR; nicotinic acetylcholine receptor; ACh; acetylcholine; NMDAR; N-methyl-D-aspartate receptor; AMPAR; α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor; NI
Molecular basis for high affinity and selectivity of peptide antagonist, Bantag-1, for the orphan BB3 receptor
Keywords: دامنه خارج سلولی; Bantag-1; Boc-Phe-His-4-amino-5-cyclohexyl-2,4,5-trideoxypentonyl-Leu-(3-dimethylamino) benzylamide N-methylammonium trifluoroacetate, BB3 receptor antagonist; BB3 receptor or BB3; bombesin receptor subtype-3; BB3â receptor or BB3â; His294 in BB3 rece
Adhesion GPCRs in immunology
Keywords: دامنه خارج سلولی; GPCR; G protein-coupled receptor; aGPCR; adhesion G protein-coupled receptor; ADGR; general adhesion GPCR name followed by class and subtype specific code; 7TM; 7 transmembrane; VLGR1; very large G protein-coupled receptor 1; ECD; extracellular domain; GP
Exploring the positive allosteric modulation of human α7 nicotinic receptors from a single-channel perspective
Keywords: دامنه خارج سلولی; Cys-loop receptors; Nicotinic receptors; Patch-clamp; Single-channel recordings; Positive allosteric modulators; nAChR; nicotinic acetylcholine receptor; ACh; acetylcholine; 5-HT3A; serotonin type 3A receptor; PAM; positive allosteric modulator; PAM-2; 3-
A pharmacological assessment of agonists and modulators at α4β2γ2 and α4β2δ GABAA receptors: The challenge in comparing apples with oranges
Keywords: دامنه خارج سلولی; GABAAR; γ-amino butyric acid receptor type A; DS1 and DS2; Delta selective agents 1 and 2; ECD; extracellular domain; ICL; intracellular loop between TM3 and TM4; PAM; positive allosteric modulator; TMD; transmembrane domain; wt.; wild-type; GABAA recept
Selective and differential interactions of BNN27, a novel C17-spiroepoxy steroid derivative, with TrkA receptors, regulating neuronal survival and differentiation
Keywords: دامنه خارج سلولی; Neurotrophins; Nerve growth factor (NGF); TrkA; Neurodegeneration; Neurotrophin receptors signaling; Neuronal apoptosis; Steroid; STD NMR; Molecular modeling; NGF; nerve growth factor; BDNF; brain-derived neurotrophic factor; NT-3; neurotrophin-3; CYP17;
Identification of the tethered peptide agonist of the adhesion G protein-coupled receptor GPR64/ADGRG2
Keywords: دامنه خارج سلولی; GPR64; GPCR; G protein; Molecular pharmacology; Signal transduction; Peptide agonist; 7TM; seven-transmembrane spanning domain; CTF; C-terminal fragment; ECD; extracellular domain; eV; empty vector; DMEM; dulbecco minimum essential medium; ELISA; enzyme-l