Practical and highly stereoselective technology for preparation of enantiopure sulfoxides and sulfinamides utilizing activated and functionally differentiated N-sulfonyl-1,2,3-oxathiazolidine-2-oxide derivatives Fulltext Access 23 Pages 2005
Carbamoylimidazolium and thiocarbamoylimidazolium salts: novel reagents for the synthesis of ureas, thioureas, carbamates, thiocarbamates and amides Fulltext Access 23 Pages 2005
Acyclic α-nitro ketones: a versatile class of α-functionalized ketones in organic synthesis Fulltext Access 23 Pages 2005
Regioselective cross-coupling reactions of multiple halogenated nitrogen-, oxygen-, and sulfur-containing heterocycles Fulltext Access 23 Pages 2005
Design, synthesis, and AMPA receptor antagonistic activity of a novel 6-nitro-3-oxoquinoxaline-2-carboxylic acid with a substituted phenyl group at the 7 position Fulltext Access 23 Pages 2005
Analysis of the role of 5-HT1A receptors in spatial and aversive learning in the rat Fulltext Access 23 Pages 2005
Synthesis and biological evaluation as AChE inhibitors of new indanones and thiaindanones related to donepezil Fulltext Access 24 Pages 2005
Tetrahedron report number 726Recent advances in the synthesis of 2H-1,4-benzoxazin-3-(4H)-ones and 3,4-dihydro-2H-1,4-benzoxazines Fulltext Access 24 Pages 2005
Syntheses of per-15N labeled etioporphyrins I-IV and a related tetrahydrobenzoporphyrin for applications in organic geochemistry and vibrational spectroscopy Fulltext Access 24 Pages 2005
Synthesis of substituted pyrrolidines and piperidines from endocyclic enamine derivatives. Synthesis of (±)-laburnamine Fulltext Access 24 Pages 2005
Microdialysis-theoretical background and recent implementation in applied life-sciences Fulltext Access 24 Pages 2005
Orally active CCR5 antagonists as anti-HIV-1 agents. Part 3: Synthesis and biological activities of 1-benzazepine derivatives containing a sulfoxide moiety Fulltext Access 24 Pages 2005
Structure-activity relationships for 1-alkyl-3-(1-naphthoyl)indoles at the cannabinoid CB1 and CB2 receptors: steric and electronic effects of naphthoyl substituents. New highly selective CB2 receptor agonists Fulltext Access 24 Pages 2005
Imperfect DNA mirror repeats in E. coli TnsA and other protein-coding DNA Fulltext Access 25 Pages 2005
Design and synthesis of novel platelet fibrinogen receptor antagonists with 2H-1,4-benzoxazine-3(4H)-one scaffold. A systematic study Fulltext Access 25 Pages 2005
Determination of the absolute stereochemistry and asymmetric total synthesis of madindolines A and B: a practical improvement to a second-generation approach from the first-generation Fulltext Access 25 Pages 2005
Recent advances in siloxane-based aryl-aryl coupling reactions: focus on heteroaromatic systems Fulltext Access 25 Pages 2005
Chiral ionic liquids, a renewal for the chemistry of chiral solvents? Design, synthesis and applications for chiral recognition and asymmetric synthesis Fulltext Access 25 Pages 2005
General Linearized Biexponential Model for QSAR Data Showing Bilinear-Type Distribution Fulltext Access 25 Pages 2005
Synthesis and biological evaluation of branched and conformationally restricted analogs of the anticancer compounds 3′-C-ethynyluridine (EUrd) and 3′-C-ethynylcytidine (ECyd) Fulltext Access 25 Pages 2005
Tissue-specific mRNA Expression Profiles of Human ATP-binding Cassette and Solute Carrier Transporter Superfamilies Fulltext Access 26 Pages 2005
The role of hydrophobic properties of chemicals in promoting allosteric reactions Fulltext Access 26 Pages 2005
Conformational control of stereochemistry in the non-concerted, degenerate rearrangement of a vinylcyclopropane Fulltext Access 26 Pages 2005
Synthesis of a novel class of chiral N,N,N-tridentate pyridinebisimidazoline ligands and their application in Ru-catalyzed asymmetric epoxidations Fulltext Access 26 Pages 2005
Naphtho[2,3-c]furan-4,9-diones and related compounds: theoretically interesting and bioactive natural and synthetic products Fulltext Access 26 Pages 2005
Experimental observation of thiamin diphosphate-bound intermediates on enzymes and mechanistic information derived from these observations Fulltext Access 26 Pages 2005
Ligand-based assessment of factor Xa binding site flexibility via elaborate pharmacophore exploration and genetic algorithm-based QSAR modeling Fulltext Access 27 Pages 2005
Synthesis of tri- and tetracyclic diterpenes. Cyclisations promoted by SmI2 Fulltext Access 27 Pages 2005
Benzotriazole mediated amino-, amido-, alkoxy- and alkylthio-alkylation Fulltext Access 27 Pages 2005
The rapid preparation of 2-aminosulfonamide-1,3,4-oxadiazoles using polymer-supported reagents and microwave heating Fulltext Access 27 Pages 2005
Design, synthesis, and biological activity of non-basic compounds as factor Xa inhibitors: SAR study of S1 and aryl binding sites Fulltext Access 28 Pages 2005
Permeability of Fluid-Phase Phospholipid Bilayers: Assessment and Useful Correlations for Permeability Screening and Other Applications Fulltext Access 28 Pages 2005
Synthesis of the EF-ring segment of ciguatoxin CTX1B based on novel regioselective reduction of unsaturated cyanohydrins and ring-closing olefin metathesis Fulltext Access 28 Pages 2005
Metal microcrystal pollutants; the heat resistant, transmissible nucleating agents that initiate the pathogenesis of TSEs? Fulltext Access 30 Pages 2005
Lead structures for applications in photodynamic therapy. Part 1: Synthesis and variation of m-THPC (Temoporfin) related amphiphilic A2BC-type porphyrins Fulltext Access 30 Pages 2005
Tetrahedron report number 727The Nazarov cyclization in organic synthesis. Recent advances Fulltext Access 30 Pages 2005
Stereospecific synthesis of 2,2,3-trisubstituted tetrahydroquinolines: application to the total syntheses of benzastatin E and natural virantmycin Fulltext Access 30 Pages 2005
Stereoselective synthesis of optically active 1-substituted-1-pyridyl-methylamines Fulltext Access 31 Pages 2005
Synthetic studies on oligosaccharides composed of 5-thioglucopyranose units Fulltext Access 32 Pages 2005
Thermodynamic and dynamic factors involved in the stability of native protein structure in amorphous solids in relation to levels of hydration Fulltext Access 32 Pages 2005
Palladium-catalysed reactions of alcohols. Part B: Formation of C-C and C-N bonds from unsaturated alcohols Fulltext Access 34 Pages 2005
Formation of five- and six-membered heterocyclic rings under radical cyclisation conditions Fulltext Access 40 Pages 2005
Palladium-catalysed reactions of alcohols. Part D: Rearrangements, carbonylations, carboxylations and miscellaneous reactions Fulltext Access 41 Pages 2005
Synthesis and applications of tetrathiafulvalenes and ferrocene-tetrathiafulvalenes and related compounds Fulltext Access 44 Pages 2005
Palladium-catalysed reactions of alcohols. Part C: Formation of ether linkages Fulltext Access 54 Pages 2005