Synthesis of oxetane-3-carboxaldehyde and methyl oxetane-3-carboxylate via homologation of oxetane-3-one Fulltext Access 6 Pages 2016
Computational Models of Neurological DisorderVirtual Brain for neurological disease modeling Fulltext Access 6 Pages 2016
Synthesis of original phosphine-sulfoxide ligands for asymmetric allylic alkylation Fulltext Access 6 Pages 2016
Novel chiral thiourea organocatalysts for the catalytic asymmetric oxaziridination Fulltext Access 6 Pages 2016
A novel host material with high thermal stability for green electrophosphorescent device Fulltext Access 6 Pages 2016
A novel colorimetric and fluorescent probe for detecting fluoride anions: from water and toothpaste samples Fulltext Access 6 Pages 2016
Simple approach to modular chiral scaffolds: binding functional sulfur nucleophiles to Cinchona alkaloids Fulltext Access 6 Pages 2016
Rational construction of macrocycles consisting of methylene bridged ureas Fulltext Access 6 Pages 2016
Reversible capture and release of aromatic amines by vicinal tricarbonyl compound Fulltext Access 6 Pages 2016
A convenient one-pot process for the synthesis of 2,4-dihydroxy-6-phenylethylenyl-8-deazapteridine derivatives Fulltext Access 6 Pages 2016
Translational PharmacologyTranslational pharmacokinetic/pharmacodynamic analysis in cancer pharmacology: a tool to maximize the value of antitumor efficacy from tumor bearing mice Fulltext Access 6 Pages 2016
Poly[(9,9-dioctyl-fluorenyl-2,7-diyl)-co-fluorenone]-based orange fluorescence probe for cellular imaging Fulltext Access 6 Pages 2016
Novel efficient functionalized tetrapyrazolic macrocycle for the selective extraction of lithium cations Fulltext Access 6 Pages 2016
A new ratiometric two-photon fluorescent probe for imaging of lysosomes in living cells and tissues Fulltext Access 6 Pages 2016
1,2,4-Triazole derivatives as host materials for blue and green phosphorescent organic light-emitting devices Fulltext Access 6 Pages 2016
Compositional analysis of pretreated (beech) wood using differential scanning calorimetry and multivariate data analysis Fulltext Access 6 Pages 2016
Hydrophobic microenvironment optimization for efficient immobilization of lipases on octadecyl functionalised resins Fulltext Access 6 Pages 2016
Enzymatic profiling in prostate and breast cancer cells: phosphate hydrolysis and alcohol oxidation Fulltext Access 6 Pages 2016
Expanding substrate scope of lipase-catalyzed transesterification by the utilization of liquid carbon dioxide Fulltext Access 6 Pages 2016
General synthesis, structure, and optical properties of benzothiophene-fused benzoheteroles containing Group 15 and 16 elements Fulltext Access 6 Pages 2016
Virtual liver models in pre-surgical planning, intra-surgical navigation and prognosis analysis Fulltext Access 6 Pages 2016
Characterization of antibody-drug conjugates by mass spectrometry: advances and future trends Fulltext Access 6 Pages 2016
Electron affinity of tricyclic, bicyclic, and monocyclic compounds containing cyanoenones correlates with their potency as inducers of a cytoprotective enzyme Fulltext Access 6 Pages 2016
Synthesis of novel flavone derivatives possessing substituted benzamides and their biological evaluation against human cancer cells Fulltext Access 6 Pages 2016
Development and structural analysis of adenosine site binding tankyrase inhibitors Fulltext Access 6 Pages 2016
Kinetic controlled affinity labeling of target enzyme with thioester chemistry Fulltext Access 6 Pages 2016
Design, synthesis, and biological evaluation of new arylamide derivatives possessing sulfonate or sulfamate moieties as steroid sulfatase enzyme inhibitors Fulltext Access 6 Pages 2016
High-yield preparation of new crown ether-based cryptands and improving complexation with paraquat, paraquat derivatives and diquat Fulltext Access 6 Pages 2016
Azide-enolate 1,3-dipolar cycloaddition in the synthesis of novel triazole-based miconazole analogues as promising antifungal agents Fulltext Access 6 Pages 2016
Strategies for improving the solubility and metabolic stability of griseofulvin analogues Fulltext Access 6 Pages 2016
Synthesis and cytotoxicity of novel artemisinin derivatives containing sulfur atoms Fulltext Access 6 Pages 2016
Discovery of novel free fatty acid receptor 1 agonists bearing triazole core via click chemistry Fulltext Access 6 Pages 2016
Synthesis and biological evaluation of novel hydrogen sulfide releasing nicotinic acid derivatives Fulltext Access 6 Pages 2016
Regulatory Incentives for Antibiotic Drug Development: A Review of Recent Proposals Fulltext Access 6 Pages 2016
The emergence and evolution of antimicrobial resistance: Impact on a global scale Fulltext Access 6 Pages 2016
Simulations reveal increased fluctuations in estrogen receptor-alpha conformation upon antagonist binding Fulltext Access 6 Pages 2016
Preparation and characterization of the pH and thermosensitive magnetic molecular imprinted nanoparticle polymer for the cancer drug delivery Fulltext Access 6 Pages 2016
Design and synthesis of selective, dual fatty acid binding protein 4 and 5 inhibitors Fulltext Access 6 Pages 2016
Discovery of anabaenopeptin 679 from freshwater algal bloom material: Insights into the structure-activity relationship of anabaenopeptin protease inhibitors Fulltext Access 6 Pages 2016
Synthesis and biological evaluation of lovastatin-derived aliphatic hydroxamates that induce reactive oxygen species Fulltext Access 6 Pages 2016
AntihypoxamiR functionalized gramicidin lipid nanoparticles rescue against ischemic memory improving cutaneous wound healing Fulltext Access 6 Pages 2016
Benzylamide antagonists of protease activated receptor 2 with anti-inflammatory activity Fulltext Access 6 Pages 2016
Design and synthesis of novel hydroxypyridinone derivatives as potential tyrosinase inhibitors Fulltext Access 6 Pages 2016
Cholinesterase inhibitory activity of chlorophenoxy derivatives—Histamine H3 receptor ligands Fulltext Access 6 Pages 2016
Synthesis of linear and cyclic peptide–PEG–lipids for stabilization and targeting of cationic liposome–DNA complexes Fulltext Access 6 Pages 2016
Simple Nε-thioacetyl-lysine-containing cyclic peptides exhibiting highly potent sirtuin inhibition Fulltext Access 6 Pages 2016
Quantitative relationships between structure and cytotoxic activity of flavonoid derivatives. An application of Hirshfeld surface derived descriptors Fulltext Access 6 Pages 2016
Design and synthesis of fluorescent glycolipid photoaffinity probes and their photoreactivity Fulltext Access 6 Pages 2016
2-Phenylbenzofuran derivatives as butyrylcholinesterase inhibitors: Synthesis, biological activity and molecular modeling Fulltext Access 6 Pages 2016
Seeking potent anti-tubercular agents: Design, synthesis, anti-tubercular activity and docking study of various ((triazoles/indole)-piperazin-1-yl/1,4-diazepan-1-yl)benzo[d]isoxazole derivatives Fulltext Access 6 Pages 2016
An evaluation of synthetic indole derivatives as inhibitors of monoamine oxidase Fulltext Access 6 Pages 2016
Design and synthesis of novel quinoxaline derivatives as potential candidates for treatment of multidrug-resistant and latent tuberculosis Fulltext Access 6 Pages 2016
Dioxol and dihydrodioxin analogs of 2- and 3-phenylacetonitriles as potent anti-cancer agents with nanomolar activity against a variety of human cancer cells Fulltext Access 6 Pages 2016
Click-based synthesis and antitubercular evaluation of dibenzofuran tethered thiazolyl-1,2,3-triazolyl acetamides Fulltext Access 6 Pages 2016
Identification of novel 2-aminothiazole conjugated nitrofuran as antitubercular and antibacterial agents Fulltext Access 6 Pages 2016
Synthesis and antitubercular activity of new 1,3,4-oxadiazoles bearing pyridyl and thiazolyl scaffolds Fulltext Access 6 Pages 2016
New insights into 3-(aminomethyl)naphthoquinones: Evaluation of cytotoxicity, electrochemical behavior and search for structure–activity correlation Fulltext Access 6 Pages 2016
New antibacterial isocoumarin glycosides from a wetland soil derived fungal strain Metarhizium anisopliae Fulltext Access 6 Pages 2016
Copper-mediated alkylation of furan and thiophene derivatives with cyclic ethers Fulltext Access 6 Pages 2016
Determination on temperature gradient of different polar reactants in reaction mixture under microwave irradiation with molecular probe Fulltext Access 6 Pages 2016
Lipase-initiated one-pot synthesis of spirooxazino derivatives: redesign of multicomponent reactions to expand substrates scope and application potential Fulltext Access 6 Pages 2016
An alternative approach to the synthesis of peptides containing a cystathionine bridge Fulltext Access 6 Pages 2016
Diarylation of chalcogen elements using arylboronic acids via copper- or palladium-catalyzed oxidative coupling Fulltext Access 6 Pages 2016
Nitrosocarbonyl release from O-substituted hydroxamic acids with pyrazolone leaving groups Fulltext Access 6 Pages 2016
Direct, visible light-sensitized benzylic CH fluorination of peptides using dibenzosuberenone: selectivity for phenylalanine-like residues Fulltext Access 6 Pages 2016
Base- and acid-catalyzed intramolecular oxy-Michael reaction for the synthesis of tetrahydrofuran ring Fulltext Access 6 Pages 2016
Base-promoted domino reaction for the synthesis of 2,3-disubstituted indoles from 2-aminobenzaldehyde/2-amino aryl ketones, tosylhydrazine, and aromatic aldehydes Fulltext Access 6 Pages 2016
Hemithioketal formation of vicinal tricarbonyl compound with thiols and their recovery Fulltext Access 6 Pages 2016
New insights in the mechanism of the microwave-assisted Pauson-Khand reaction Fulltext Access 6 Pages 2016
Highly selective oxidation of unsaturated hydrocarbons to carbonyl compounds by two-phase catalysis Fulltext Access 6 Pages 2016
Design and synthesis of thiourea derivatives with sulfur-containing heterocyclic scaffolds as potential tyrosinase inhibitors Fulltext Access 6 Pages 2016
Photochemical functionalization of diazines: metal-free vinylation and phosphonylation Fulltext Access 6 Pages 2016
Design of high-performance dye-sensitized solar cells by variation of the dihedral angles of dyes Fulltext Access 6 Pages 2016
Novel substituted aminothiazoles as potent and selective anti-hepatocellular carcinoma agents Fulltext Access 6 Pages 2016
Novel bicyclo[3.1.0]hexane analogs as antagonists of metabotropic glutamate 2/3 receptors for the treatment of depression Fulltext Access 6 Pages 2016
Synthesis and biological evaluation of chalcone derivatives containing aminoguanidine or acylhydrazone moieties Fulltext Access 6 Pages 2016
Increasing metabolic stability via the deuterium kinetic isotope effect: An example from a proline-amide-urea aminothiazole series of phosphatidylinositol-3 kinase alpha inhibitors Fulltext Access 6 Pages 2016