Effect of fluoro substituents and central atom nature on chiral derivatives of bisdiphenylborates and isoelectronic structures Fulltext Access 6 Pages 2005
Synthesis and biocatalytic resolution of a new atropisomeric thiobiphenyl: (2,2â²,6,6â²-tetramethoxybiphenyl-3,3â²-diyl)dimethanethiol Fulltext Access 6 Pages 2005
Chemoenzymatic preparation of the enantiomers of β-tryptophan ethyl ester and the β-amino nitrile analogue Fulltext Access 6 Pages 2005
Synthesis and olfactory evaluation of the enantiomerically enriched forms of 7,11-epoxymegastigma-5(6)-en-9-one and 7,11-epoxymegastigma-5(6)-en-9-ols isomers, identified in Passiflora edulis Fulltext Access 6 Pages 2005
Dirhodium catalyzed intramolecular enantioselective C-H insertion reaction of N-cumyl-N-(2-p-anisylethyl)diazoacetamide: synthesis of (â)-Rolipram Fulltext Access 6 Pages 2005
Enzyme-assisted synthesis of (S)-1,3-dihydroxy-3,7-dimethyl-6-octen-2-one, the male-produced aggregation pheromone of the Colorado potato beetle, and its (R)-enantiomer Fulltext Access 6 Pages 2005
The first asymmetric catalytic halo aldol reaction of β-iodo allenoates with aldehydes by using chiral salen catalyst Fulltext Access 6 Pages 2005
Advances in analysis and synthesis of myo-inositol-derivatives through resolution by crystallisation Fulltext Access 6 Pages 2005
Synthesis of enantiomerically pure glycidol via a fully enantioselective lipase-catalyzed resolution Fulltext Access 6 Pages 2005
Stereoselective synthesis of (2R,3S,4S,5R)-trans-3,4-dihydroxy-5-(4-fluorophenoxymethyl)-2-(1-N-hydroxyureidyl-3-butyn-4-yl)tetrahydrofuran and (2R,3S,4S,5R)-trans-5-ethynyl-2-(4-fluorophenoxymethyl)-3,4-O-isopropylidene tetrahydrofuran from mannose diace Fulltext Access 6 Pages 2005
Thiourea-based non-nucleoside inhibitors of HIV reverse transcriptase as bifunctional organocatalysts in the asymmetric Strecker synthesis Fulltext Access 6 Pages 2005
Synthesis, characterisation and cytotoxicity of chloro derivatives of prenylnaphthohydroquinone Fulltext Access 6 Pages 2005
Structure–affinity relationships of halogenated predicentrine and glaucine derivatives at D1 and D2 dopaminergic receptors: halogenation and D1 receptor selectivity Fulltext Access 6 Pages 2005
Studies on interaction of an intramolecular charge transfer fluorescence probe: 4′-Dimethylamino-2,5-dihydroxychalcone with DNA Fulltext Access 6 Pages 2005
Human recombinant monoamine oxidase B as reliable and efficient enzyme source for inhibitor screening Fulltext Access 6 Pages 2005
Irreversibly inhibitory kinetics of 3,5-dihydroxyphenyl decanoate on mushroom (Agaricus bisporus) tyrosinase Fulltext Access 6 Pages 2005
Cyclopentenediones, inhibitors of farnesyl protein transferase and anti-tumor compounds, isolated from the fruit of Lindera erythrocarpa Makino Fulltext Access 6 Pages 2005
Synthesis and atropisomeric stability of 2,2â²-bis(ferrocenylhydroxymethyl)-1,1â²-biphenyl Fulltext Access 6 Pages 2005
Synthesis of a peptidocalix[4]arene library and identification of compounds with hydrolytic activity Fulltext Access 6 Pages 2005
Synthesis of complex carbobicyclic compounds from sugar allyltins: functionalization of the allylic position in bicyclo[4.3.0]nonene derivatives Fulltext Access 6 Pages 2005
Neo-glycoconjugates: stereoselective synthesis of α-glycosyl amides via Staudinger ligation reactions Fulltext Access 6 Pages 2005
Evaluation of substituent effects on activity and enantioselectivity in the enzymatic reduction of aryl ketones Fulltext Access 6 Pages 2005
Syntheses of chiral hybrid O,N-donor ligands for the investigation of lanthanide complex reactivities in direct aldol condensations Fulltext Access 6 Pages 2005
First synthesis of 5,6-branched galacto-hexasaccharide, the dimer of the trisaccharide repeating unit of the cell-wall galactans of Bifidobacterium catenulatum YIT 4016 Fulltext Access 6 Pages 2005
Palladium-catalyzed asymmetric hydrovinylation under mild conditions using monodentate chiral spiro phosphoramidite and phosphite ligands Fulltext Access 6 Pages 2005
Synthesis, NMR conformational studies and host-guest behaviour of new (+)-tartaric acid derivatives Fulltext Access 6 Pages 2005
Enzymatic resolution of N-protected-β3-amino methyl esters, using lipase B from Candida antarctica Fulltext Access 6 Pages 2005
Polymer-supported chiral phosphinooxathiane ligands for palladium-catalyzed asymmetric allylations Fulltext Access 6 Pages 2005
Enantiopure erythro- and threo-1-aryl-1-[2-pyrrolidyl]-methanols: synthesis from l-proline Fulltext Access 6 Pages 2005
3-N,N-Dimethylamino-3-deoxy lincomycin: A structure-based hybrid between lincomycin and the desosamine unit of erythromycin Fulltext Access 6 Pages 2005
S-Oxidation products of (+)-thiomicamine-derived oxazolines-promising substrates in the synthesis of alkyl methyl sulfoxides Fulltext Access 6 Pages 2005
Enzymatic synthesis of N-glycoprotein linkage region disaccharide mimetics using β-N-acetylhexosaminidases from Aspergillus oryzae and Vigna radiata Fulltext Access 6 Pages 2005
Syntheses of sugar-related pyrrolidine derivatives by reductive amination reactions Fulltext Access 6 Pages 2005
Transglycosylation of tagatose with maltotriose by Bacillus stearothermophilus maltogenic amylase (BSMA) Fulltext Access 6 Pages 2005
Synthesis of diastereo- and enantiomerically pure anti-3-methyl-1,4-pentanediol via lipase catalysed acylation Fulltext Access 6 Pages 2005
Metal promoted asymmetry in the 1,2-diboroethylarene synthesis: diboration versus dihydroboration Fulltext Access 6 Pages 2005
New unsymmetrical hybrid ferrocenylphosphine-phosphoramidite ligands derived from H8-BINOL for highly efficient Rh-catalyzed enantioselective hydrogenation Fulltext Access 6 Pages 2005
Asymmetric induction in the conjugate addition of thioacetic acid to methacrylamides with chiral auxiliaries Fulltext Access 6 Pages 2005
Synthesis of the (1S,2S)- and (1R,2S)-stereoisomers of the respective E- and Z-isomers of ethyl 4-[(2-hydroxycyclohexyl)methyl]phenoxy-3-methyl-2-butenoate using yeast whole cell bioreduction of the parent ketones Fulltext Access 6 Pages 2005
Tunable dendritic ligands of chiral 1,2-diamine and their application in asymmetric transfer hydrogenation Fulltext Access 6 Pages 2005
Enantioselective reduction of benzofuryl halomethyl ketones: asymmetric synthesis of (R)-bufuralol Fulltext Access 6 Pages 2005
Amination/annulation of chlorobutenones with chiral amine compounds: synthesis of 1,2,4-trisubstituted pyrroles Fulltext Access 6 Pages 2005
(1S,2S)-1-Amino-2-hydroxy-1,2,3,4-tetrahydronaphthalene: a new chiral auxiliary for asymmetric Reformatsky reactions Fulltext Access 6 Pages 2005
The synthesis of oximes and nitroalkanes bearing a chiral auxiliary unit: convenient substrates for the preparation of enantiomerically pure nitrile oxides Fulltext Access 6 Pages 2005
The first simple and efficient synthesis of the unusual dipeptide part of Phomopsin A Fulltext Access 6 Pages 2005
The high-pressure [4+2]cycloaddition of 1-methoxybuta-1,3-diene to the glycolaldehyde-derived heterodienophiles, catalyzed by chiral metallosalen complexes Fulltext Access 6 Pages 2005
Synthesis of Rosavin and its analogues based on a Mizoroki-Heck type reaction Fulltext Access 6 Pages 2005
Chemoenzymatic synthesis of calcilytic agent NPS-2143 employing a lipase-mediated resolution protocol Fulltext Access 6 Pages 2005
Enantioselective microbial reduction of 6-oxo-8-[4-[4-(2-pyrimidinyl)-1-piperazinyl]butyl]-8-azaspiro[4.5]decane-7,9-dione Fulltext Access 6 Pages 2005
The dynamic kinetic resolution of 3-oxo-4-phenyl-β-lactam by recombinant E. coli overexpressing yeast reductase Ara1p Fulltext Access 6 Pages 2005
Preparation of (R)- and (S)-6-hydroxybuspirone by enzymatic resolution or hydroxylation Fulltext Access 6 Pages 2005
Palladium/chiral phosphine–olefin complexes: X-ray crystallographic analysis and the use in catalytic asymmetric allylic alkylation Fulltext Access 6 Pages 2005
5-Methyl-4H-1,3-dioxins, new chiral building blocks: transformation into (R)- and (S)-4-hydroxymethyl-4-methyl-1,3-dioxolanes via oxidation and rearrangement and determination of the absolute configuration Fulltext Access 6 Pages 2005
Solid state properties of 1,2-epoxy-3-(2-methoxyphenyloxy)-propane-valuable intermediate in non-racemic drug synthesis Fulltext Access 6 Pages 2005
Studies on the construction of abutasterone-type and 24-epi-abutasterone-type side chains employing asymmetric dihydroxylation of (E)-20(22),24-cholestadiene Fulltext Access 6 Pages 2005
Enantioselective aza-Michael reactions catalyzed by samarium iodobinaphtholate Fulltext Access 6 Pages 2005
Theoretical study revealing the functioning of a novel combination of catalytic motifs in histone deacetylase Fulltext Access 6 Pages 2005
Symbioimine and neosymbioimine, amphoteric iminium metabolites from the symbiotic marine dinoflagellate Symbiodinium sp. Fulltext Access 6 Pages 2005
On the mechanism of isomerization of all-trans-retinol esters to 11-cis-retinol in retinal pigment epithelial cells: 11-Fluoro-all-trans-retinol as substrate/inhibitor in the visual cycle Fulltext Access 6 Pages 2005
New 1,2,3,4-tetrahydro-1-aza-anthraquinones and 2-aminoalkyl compounds from norlapachol with molluscicidal activity Fulltext Access 6 Pages 2005
3D-QSAR analysis on benzazole derivatives as eukaryotic topoisomerase II inhibitors by using comparative molecular field analysis method Fulltext Access 6 Pages 2005
Xanthones induce cell-cycle arrest and apoptosis in human colon cancer DLD-1 cells Fulltext Access 6 Pages 2005
QSAR studies of paeonol analogues for inhibition of platelet aggregation Fulltext Access 6 Pages 2005
Inclusion complexes of azadirachtin with native and methylated cyclodextrins: solubilization and binding ability Fulltext Access 6 Pages 2005
Classical and dynamic resolution of 1-amino-3-methyl-1,3,4,5-tetrahydrobenzo[d]azepin-2-one Fulltext Access 6 Pages 2005
Synthesis and antimycobacterial evaluation of certain fluoroquinolone derivatives Fulltext Access 6 Pages 2005
N,N′-Bis(3-aminopropyl)-2,7-diamino-1,8-naphthyridine stabilized a single pyrimidine bulge in duplex DNA Fulltext Access 6 Pages 2005
Steroid-derived phospholipid scramblases induce exposure of phosphatidylserine on the surface of red blood cells Fulltext Access 6 Pages 2005
‘Green’ methodology for efficient and selective benzoylation of nucleosides using benzoyl cyanide in an ionic liquid Fulltext Access 6 Pages 2005
Synthesis and structure-activity relationships of 2-alkylidenethiazolidine-4,5-diones as antibiotic agents Fulltext Access 6 Pages 2005
Cancer preventive agents, Part 2: Synthesis and evaluation of 2-phenyl-4-quinolone and 9-oxo-9,10-dihydroacridine derivatives as novel antitumor promoters Fulltext Access 6 Pages 2005
Synthesis of new phorbol derivatives having ethereal side chain and evaluation of their anti-HIV activity Fulltext Access 6 Pages 2005
Heterogeneous catalysis of the asymmetric aldol reaction by solid-supported proline-terminated peptides Fulltext Access 6 Pages 2005