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Daneshyari Pharmaceutical Science Journas Latest Articles

Pharmaceutical Science Research Articles

Determination of bile salt critical micellization concentration on the road to drug discovery
Fulltext Access 20 Pages 2014
Hydrogels in a historical perspective: From simple networks to smart materials
Fulltext Access 20 Pages 2014
Stimuli-sensitive nanopreparations for combination cancer therapy
Fulltext Access 20 Pages 2014
Improving the efficacy of inhaled drugs in cystic fibrosis: Challenges and emerging drug delivery strategies
Fulltext Access 20 Pages 2014
Effective use of transdermal drug delivery in children
Fulltext Access 20 Pages 2014
Thiazolidine-2,4-diones as multi-targeted scaffold in medicinal chemistry: Potential anticancer agents
Fulltext Access 20 Pages 2014
Graphical contents list
Fulltext Access 20 Pages 2014
Preclinical pharmacokinetic evaluation of a new formulation of a bifendate solid dispersion using a supercritical fluid chromatography-tandem mass spectrometry method
Fulltext Access 20 Pages 2014
Solid-phase dispersive extraction method for analysis of benzodiazepine drugs in serum and urine samples
Fulltext Access 20 Pages 2014
Natural hydrazine-containing compounds: Biosynthesis, isolation, biological activities and synthesis
Fulltext Access 20 Pages 2014
Design, synthesis and biological evaluation of a series of pyrano chalcone derivatives containing indole moiety as novel anti-tubulin agents
Fulltext Access 20 Pages 2014
Intranasal delivery of systemic-acting drugs: Small-molecules and biomacromolecules
Fulltext Access 20 Pages 2014
Polymers in cell encapsulation from an enveloped cell perspective
Fulltext Access 20 Pages 2014
Synthesis, antibacterial activity, and biological evaluation of formyl hydroxyamino derivatives as novel potent peptide deformylase inhibitors against drug-resistant bacteria
Fulltext Access 20 Pages 2014
Graphical contents list
Fulltext Access 20 Pages 2014
Recent developments in biological activities of chalcones: A mini review
Fulltext Access 20 Pages 2014
An investigation of in vitro cytotoxicity and apoptotic potential of aromatic diselenides
Fulltext Access 20 Pages 2014
1,3,5-Triazine-based analogues of purine: From isosteres to privileged scaffolds in medicinal chemistry
Fulltext Access 20 Pages 2014
Studies on molecular properties prediction, antitubercular and antimicrobial activities of novel quinoline based pyrimidine motifs
Fulltext Access 20 Pages 2014
Graphical contents list
Fulltext Access 20 Pages 2014
The use of spirocyclic scaffolds in drug discovery
Fulltext Access 21 Pages 2014
Image-guided interventional therapy for cancer with radiotherapeutic nanoparticles
Fulltext Access 21 Pages 2014
Dry powders for oral inhalation free of lactose carrier particles
Fulltext Access 21 Pages 2014
Conventional and microwave assisted synthesis of pyrazolone Mannich bases possessing anti-inflammatory, analgesic, ulcerogenic effect and antimicrobial properties
Fulltext Access 21 Pages 2014
Engineered microenvironments provide new insights into ovarian and prostate cancer progression and drug responses
Fulltext Access 21 Pages 2014
The Biopharmaceutics Risk Assessment Roadmap for Optimizing Clinical Drug Product Performance
Fulltext Access 21 Pages 2014
Novel chromogenic aminopeptidase substrates for the detection and identification of clinically important microorganisms
Fulltext Access 21 Pages 2014
Synthesis and antiproliferative action of a novel series of maprotiline analogues
Fulltext Access 21 Pages 2014
A segmentation analysis for pharmacists' and patients' views of pharmacists' roles
Fulltext Access 21 Pages 2014
Recent advances in micro/nanoscale biomedical implants
Fulltext Access 21 Pages 2014
Acoustic behavior of microbubbles and implications for drug delivery
Fulltext Access 21 Pages 2014
Towards cytotoxic and selective derivatives of maslinic acid
Fulltext Access 22 Pages 2014
The use of skin models in drug development
Fulltext Access 22 Pages 2014
Understanding the relationship between wettability and dissolution of solid dispersion
Fulltext Access 23 Pages 2014
Amino derivatives of glycyrrhetinic acid as potential inhibitors of cholinesterases
Fulltext Access 23 Pages 2014
Next Generation Drying Technologies for Pharmaceutical Applications
Fulltext Access 23 Pages 2014
Design and synthesis of phenylisoxazole derivatives as novel human acrosin inhibitors
Fulltext Access 23 Pages 2014
Drug delivery design for intravenous route with integrated physicochemistry, pharmacokinetics and pharmacodynamics: Illustration with the case of taxane therapeutics
Fulltext Access 24 Pages 2014
Graphical contents list
Fulltext Access 24 Pages 2014
Inhibition of human thymidine phosphorylase by conformationally constrained pyrimidine nucleoside phosphonic acids and their “open-structure” isosteres
Fulltext Access 24 Pages 2014
Effectiveness of tobacco use cessation interventions delivered by pharmacy personnel: A systematic review
Fulltext Access 24 Pages 2014
Synthesis, structure-activity relationships and biological evaluation of barbigerone analogues as anti-proliferative and anti-angiogenesis agents
Fulltext Access 24 Pages 2014
Cancer nanotechnology: The impact of passive and active targeting in the era of modern cancer biology
Fulltext Access 24 Pages 2014
Enzyme-Transporter-Mediated Drug Interactions with Small Molecule Tyrosine Kinase Inhibitors
Fulltext Access 24 Pages 2014
Paediatric oral biopharmaceutics: Key considerations and current challenges
Fulltext Access 25 Pages 2014
Quantification of in situ granulation-induced changes in pre-compression, solubility, dose distribution and intrinsic in vitro release characteristics of ibuprofen-cationic dextran conjugate crystanules
Fulltext Access 25 Pages 2014
4-Thiazolidinones: The advances continue…
Fulltext Access 26 Pages 2014
Cancer nanomedicine and the complement system activation paradigm: Anaphylaxis and tumour growth
Fulltext Access 26 Pages 2014
Simultaneous determination of probe drugs, metabolites, inhibitors and inducer in human plasma by liquid chromatography/tandem mass spectrometry and its application to pharmacokinetic study
Fulltext Access 26 Pages 2014
Synthesis of novel, peptidic kinase inhibitors with cytostatic/cytotoxic activity
Fulltext Access 27 Pages 2014
Antibody-drug conjugates-A new wave of cancer drugs
Fulltext Access 27 Pages 2014
Critical practical aspects in the application of liquid chromatography–mass spectrometric studies for the characterization of impurities and degradation products
Fulltext Access 27 Pages 2014
Current applications of miniaturized chromatographic and electrophoretic techniques in drug analysis
Fulltext Access 27 Pages 2014
Early pharmaceutical profiling to predict oral drug absorption: Current status and unmet needs
Fulltext Access 27 Pages 2014
Lipid-based carriers for pulmonary products: Preclinical development and case studies in humans
Fulltext Access 28 Pages 2014
Natural product based leads to fight against leishmaniasis
Fulltext Access 28 Pages 2014
Structural and Dynamic Properties of Amorphous Solid Dispersions: The Role of Solid-State Nuclear Magnetic Resonance Spectroscopy and Relaxometry
Fulltext Access 28 Pages 2014
Is the full potential of the biopharmaceutics classification system reached?
Fulltext Access 28 Pages 2014
Present status of quinoxaline motifs: Excellent pathfinders in therapeutic medicine
Fulltext Access 28 Pages 2014
Cell-mediated delivery of nanoparticles: Taking advantage of circulatory cells to target nanoparticles
Fulltext Access 28 Pages 2014
Related impurities in peptide medicines
Fulltext Access 29 Pages 2014
Targeting the homologous recombination pathway by small molecule modulators
Fulltext Access 29 Pages 2014
Progress of the synthesis of condensed pyrazole derivatives (from 2010 to mid-2013)
Fulltext Access 30 Pages 2014
Gelatin carriers for drug and cell delivery in tissue engineering
Fulltext Access 31 Pages 2014
Synthesis of a novel legumain-cleavable colchicine prodrug with cell-specific toxicity
Fulltext Access 31 Pages 2014
High performance liquid chromatographic determination of ultra traces of two tricyclic antidepressant drugs imipramine and trimipramine in urine samples after their dispersive liquid-liquid microextraction coupled with response surface optimization
Fulltext Access 31 Pages 2014
Thermodynamic Investigation of Carbamazepine-Saccharin Co-Crystal Polymorphs
Fulltext Access 31 Pages 2014
A comprehensive review on synthetic approach for antimalarial agents
Fulltext Access 32 Pages 2014
Novel coumarin-dihydropyrazole thio-ethanone derivatives: Design, synthesis and anticancer activity
Fulltext Access 33 Pages 2014
Some molecular targets for antihyperlipidemic drug research
Fulltext Access 34 Pages 2014
Identification of forced degradation products of tamsulosin using liquid chromatography/electrospray ionization tandem mass spectrometry
Fulltext Access 34 Pages 2014
The implications of recent advances in carboxymethyl chitosan based targeted drug delivery and tissue engineering applications
Fulltext Access 34 Pages 2014
Flavones: An important scaffold for medicinal chemistry
Fulltext Access 34 Pages 2014
Polymer supported synthesis of a natural product-inspired oxepane library
Fulltext Access 35 Pages 2014
Targeted and heat-triggered doxorubicin delivery to tumors by dual targeted cationic thermosensitive liposomes
Fulltext Access 35 Pages 2014
Recent developments in tubulin polymerization inhibitors: An overview
Fulltext Access 36 Pages 2014
Preparation, anticholinesterase activity and molecular docking of new lupane derivatives
Fulltext Access 36 Pages 2014
Synthesis and antiproliferative effect of novel 4-thiazolidinone-, pyridine- and piperazine-based conjugates on human leukemic cells
Fulltext Access 36 Pages 2014
Changes in urinary metabolic profile after oral administration of curcuma extract in rats
Fulltext Access 38 Pages 2014
Encapsulated islets for diabetes therapy: History, current progress, and critical issues requiring solution
Fulltext Access 39 Pages 2014
Single compartment drug delivery
Fulltext Access 39 Pages 2014
Recent advances of resveratrol in nanostructured based delivery systems and in the management of HIV/AIDS
Fulltext Access 39 Pages 2014
Chemical biology on the genome
Fulltext Access 40 Pages 2014
Structure-activity relationships of substituted oxyoxalamides as inhibitors of the human soluble epoxide hydrolase
Fulltext Access 41 Pages 2014
Synthesis, molecular docking and biological evaluation of coumarin derivatives containing piperazine skeleton as potential antibacterial agents
Fulltext Access 41 Pages 2014
Ocular delivery of macromolecules
Fulltext Access 42 Pages 2014
Prospective therapeutic agents for obesity: Molecular modification approaches of centrally and peripherally acting selective cannabinoid 1 receptor antagonists
Fulltext Access 42 Pages 2014
Ropivacaine loaded microemulsion and microemulsion-based gel for transdermal delivery: Preparation, optimization, and evaluation
Fulltext Access 42 Pages 2014
Injectable controlled release depots for large molecules
Fulltext Access 45 Pages 2014
Scaffold biomaterials for nano-pathophysiology
Fulltext Access 46 Pages 2014
Nanoparticle targeting of anti-cancer drugs that alter intracellular signaling or influence the tumor microenvironment
Fulltext Access 46 Pages 2014
Highly cited research articles in Journal of Controlled Release: Commentaries and perspectives by authors
Fulltext Access 46 Pages 2014
Glycosylation-mediated targeting of carriers
Fulltext Access 50 Pages 2014
Antiproliferative novel isoxazoles: Modeling, virtual screening, synthesis, and bioactivity evaluation
Fulltext Access 52 Pages 2014
Recent advances in the structural library of functionalized quinazoline and quinazolinone scaffolds: Synthetic approaches and multifarious applications
Fulltext Access 52 Pages 2014
Designing and building the next generation of improved vaccine adjuvants
Fulltext Access 53 Pages 2014
Designer lipids for drug delivery: From heads to tails
Fulltext Access 56 Pages 2014
Synthesis and identification of chiral aminomethylpiperidine carboxamides as inhibitor of collagen induced platelet activation
Fulltext Access 63 Pages 2014
Synthesis, structure-activity relationship of iodinated-4-aryloxymethyl-coumarins as potential anti-cancer and anti-mycobacterial agents
Fulltext Access 63 Pages 2014
Rational approaches, design strategies, structure activity relationship and mechanistic insights for anticancer hybrids
Fulltext Access 66 Pages 2014
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