Design, synthesis and evaluation of MCH receptor 1 antagonists-Part I: Optimization of HTS hits towards an in vivo efficacious tool compound BI 414

Design, synthesis and evaluation of MCH receptor 1 antagonists-Part I: Optimization of HTS hits towards an in vivo efficacious tool compound BI 414

Database: Elsevier - ScienceDirect (ساینس دایرکت)
Journal: Bioorganic & Medicinal Chemistry Letters - Volume 25, Issue 16, 15 August 2015, Pages 3264-3269

Stephan G. Müller, Armin Heckel, Jörg T. Kley, Thorsten Lehmann, Philipp Lustenberger, Thorsten Oost, Gerald J. Roth, Klaus Rudolf, Kirsten Arndt, Martin Lenter, Ralf R.H. Lotz, Gerd-Michael Maier, Michael Markert, Marcus Schindler, Dirk Stenkamp,