کد مقاله کد نشریه سال انتشار مقاله انگلیسی نسخه تمام متن
1361315 981460 2012 4 صفحه PDF دانلود رایگان
عنوان انگلیسی مقاله ISI
Phosphonium lipocations as antiparasitic agents
موضوعات مرتبط
مهندسی و علوم پایه شیمی شیمی آلی
پیش نمایش صفحه اول مقاله
Phosphonium lipocations as antiparasitic agents
چکیده انگلیسی

Phosphonium lipocations were synthesized and evaluated for inhibition of the development of Plasmodium falciparum and Trypanosoma cruzi, etiological agents of malaria and Chagas disease, respectively. Optimal phthalimides and 1,4-naphthoquinone-based lipocations were active in vitro at mid-high nM concentrations against P. falciparum and low μM concentrations against T. cruzi.

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ناشر
Database: Elsevier - ScienceDirect (ساینس دایرکت)
Journal: Bioorganic & Medicinal Chemistry Letters - Volume 22, Issue 8, 15 April 2012, Pages 2976–2979
نویسندگان
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