Enantio-differential approach to identify the target cell for glucosyl jasmonate-type leaf-closing factor, by using fluorescence-labeled probe compounds Fulltext Access 9 Pages 2006
The Ugi reaction with 2-substituted cyclic imines. Synthesis of substituted proline and homoproline derivatives Fulltext Access 9 Pages 2006
Three different fluorescent responses to transition metal ions using receptors based on 1,2-bis- and 1,2,4,5-tetrakis-(8-hydroxyquinolinoxymethyl)benzene Fulltext Access 9 Pages 2006
α-Aminoisobutyric acid modified protected analogues of β-amyloid residue 17-20: a change from sheet to helix Fulltext Access 9 Pages 2006
Acid-catalyzed rearrangement of 1-benzyl-2-methyl-3-piperidone to 1-benzyl-2-acetylpyrrolidine Fulltext Access 9 Pages 2006
Sequential addition reaction of lithium acetylides and Grignard reagents to thioiminium salts from thiolactams leading to 2,2-disubstituted cyclic amines Fulltext Access 9 Pages 2006
Asymmetric syntheses of N-substituted α-amino esters via dynamic kinetic resolution of α-haloacyl diacetone-d-glucose Fulltext Access 9 Pages 2006
Synthesis of a hydrophilic and non-ionic anthracene derivative, the N,Nâ²-di-(2,3-dihydroxypropyl)-9,10-anthracenedipropanamide as a chemical trap for singlet molecular oxygen detection in biological systems Fulltext Access 9 Pages 2006
Dark singlet oxygenation of organic substrates in single-phase and multiphase microemulsion systems Fulltext Access 9 Pages 2006
Reactions of urocanic acid (UCA) methyl esters with singlet oxygen and 4-methyl-1,2,4-triazoline-3,5-dione (MTAD) Fulltext Access 9 Pages 2006
Reaction of (1,3-dioxo-2,3-dihydro-1H-inden-2-ylidene)propanedinitrile with N-arylisoindolines Fulltext Access 9 Pages 2006
A novel tert-butoxycarbonylation reagent: 1-tert-butoxy-2-tert-butoxycarbonyl-1,2-dihydroisoquinoline (BBDI) Fulltext Access 9 Pages 2006
A free radical Mannich type reaction: selective α-CH aminomethylation of ethers by Ti(III)/t-BuOOH system under aqueous acidic conditions Fulltext Access 9 Pages 2006
A homologous series of eunicellin-based diterpenes from Acalycigorgia sp. characterised by tandem mass spectrometry Fulltext Access 9 Pages 2006
Studies toward the construction of substituted piperidine-2-ones and pyridine-2-ones from Baylis-Hillman adducts: discovery of a facile synthesis of 5-methyl-4-oxo-6-aryl-3-aza-bicyclo[3.1.0]hexane-1-carboxylates Fulltext Access 9 Pages 2006
Palladium-catalyzed carbon dioxide elimination-fixation reaction of 6-methoxycarbonyloxy-2,4-hexadien-1-ols Fulltext Access 9 Pages 2006
Design and synthesis of fluconazole/bile acid conjugate using click reaction Fulltext Access 9 Pages 2006
Synthesis, in vitro antiproliferative activities, and Chk1 inhibitory properties of dipyrrolo[3,4-a:3,4-c]carbazole-triones Fulltext Access 9 Pages 2006
Synthesis and conformational analysis of naphth[1â²,2â²:5,6][1,3]oxazino[3,2-c][1,3]benzoxazine and naphth[1â²,2â²:5,6][1,3]oxazino[3,4-c][1,3]benzoxazine derivatives Fulltext Access 9 Pages 2006
Foldamer-based pyridine-fullerene tweezer receptors for enhanced binding of zinc porphyrin Fulltext Access 9 Pages 2006
Remote stereocontrol by the sulfinyl group: Mukaiyama aldol reactions of (S)-2-[2-(p-tolylsulfinyl)phenyl]acetaldehyde in the asymmetric synthesis of β-hydroxyacids and 1,3-diols Fulltext Access 9 Pages 2006
5,6-Bis(dimethylamino)acenaphthylene as an activated alkene and 'proton sponge' in halogenation reactions Fulltext Access 9 Pages 2006
Musk or violet? Design, synthesis and odor of seco-derivates of a musky carotol lead Fulltext Access 9 Pages 2006
Synthesis of glutamic acid and glutamine peptides possessing a trifluoromethyl ketone group as SARS-CoV 3CL protease inhibitors Fulltext Access 9 Pages 2006
Synthesis and some transformations of new 9-furylnaphtho[2,3-b]furan derivatives Fulltext Access 9 Pages 2006
Facile and catalytic degradation method of DDT using Pd/C-Et3N system under ambient pressure and temperature Fulltext Access 9 Pages 2006
Chiral ligand-controlled asymmetric conjugate amination of enoates with lithium mesitylmethyl(trimethylsilyl)amide Fulltext Access 9 Pages 2006
Reaction between glutaric anhydride and N-benzylidenebenzylamine, and further transformations to new substituted piperidin-2-ones Fulltext Access 9 Pages 2006
Cobalt-mediated solid phase synthesis of 3-O-alkynylbenzyl galactosides and their evaluation as galectin inhibitors Fulltext Access 9 Pages 2006
Regioselectivity in acylation of oligosaccharides catalyzed by the metalloprotease thermolysin Fulltext Access 9 Pages 2006
An efficient solid-phase synthesis of 2-alkyl-4,6-diaminopyrimidines and 2,4,6-triaminopyrimidines Fulltext Access 9 Pages 2006
A new approach towards 2-amino-1-aryloxy-3-methoxypropanes from 1-arylmethyl-2-(bromomethyl)aziridines Fulltext Access 9 Pages 2006
Study on the reactions of ethyl 4,4,4-trifluoro-3-oxobutanoate with arylidenemalononitriles Fulltext Access 9 Pages 2006
Synthesis of dihydrodehydrodiconiferyl alcohol and derivatives through intramolecular C-H insertion Fulltext Access 9 Pages 2006
New dioxadiaza-, trioxadiaza- and hexaaza-macrocycles containing dibenzofuran units Fulltext Access 9 Pages 2006
Photodegradation of some 14,15-bisnorlabdene-13-ones, derived from larixol. Synthesis of drimanic dienes with functional groups at C-6 Fulltext Access 9 Pages 2006
Synthesis of aminimides derived from oleic acid: a new family of drag-reducing surfactants Fulltext Access 9 Pages 2006
Synthesis of enantiopure bis-aziridines, bis-epoxides, and aziridino-epoxides from d-mannitol Fulltext Access 9 Pages 2006
Sodium dithionite initiated regio- and stereoselective radical addition of polyfluoroalkyl iodide with norbornene analogs Fulltext Access 9 Pages 2006
Self-assembly of aromatic sulfonamide–amide hybridized molecules: formation of 2D layers and 3D microporous networks in the solid state Fulltext Access 9 Pages 2006
Catalytic enantioselective [2+2]-cycloaddition reaction of 2-methoxycarbonyl-2-cyclopenten-1-one by chiral copper catalyst Fulltext Access 9 Pages 2006
Synthesis of 6- to 10-membered ring (E)-hydroxyiminohydroazaazoniabenzocycloalkenes derivative from cyclization of 2-nitromethylene-1-(Ï-phenylalkyl)imidazolidine or 2-nitromethylene-1-(Ï-phenylalkyl)hexahydropyrimidine in trifluoromethanesulfonic acid Fulltext Access 9 Pages 2006
An efficient synthesis of (E)-α,β-unsaturated ketones and esters with total stereoselectivity by using chromium dichloride Fulltext Access 9 Pages 2006
Enantioselective total and formal syntheses of paroxetine (PAXIL) via phosphine-catalyzed enone α-arylation using arylbismuth(V) reagents: a regiochemical complement to Heck arylation Fulltext Access 9 Pages 2006
Longipedlactones A-I, nine novel triterpene dilactones possessing a unique skeleton from Kadsura longipedunculata Fulltext Access 9 Pages 2006
Synthesis, antitumor and anti-HIV activities of benzodithiazine-dioxides Fulltext Access 9 Pages 2006
Synthesis and evaluation of azaindole-α-alkyloxyphenylpropionic acid analogues as PPARα/γ agonists Fulltext Access 9 Pages 2006
Synthesis of functionalised 2-aryl-5-nitro-1H-indoles and their activity as bacterial NorA efflux pump inhibitors Fulltext Access 9 Pages 2006
Improved synthesis of 2′-amino-2′-deoxyguanosine and its phosphoramidite Fulltext Access 9 Pages 2006
Anti-tubercular agents. Part 3. Benzothiadiazine as a novel scaffold for anti-Mycobacterium activity Fulltext Access 9 Pages 2006
Polymeric grape-seed procyanidins, but not monomeric catechins and oligomeric procyanidins, impair degranulation and membrane ruffling in RBL-2H3 cells Fulltext Access 9 Pages 2006
Design, synthesis, and pharmacological evaluation of new neuroactive pyrazolo[3,4-b]pyrrolo[3,4-d]pyridine derivatives with in vivo hypnotic and analgesic profile Fulltext Access 9 Pages 2006
Phenazine-1-carboxamides: Structure–cytotoxicity relationships for 9-substituents and changes in the H-bonding pattern of the cationic side chain Fulltext Access 9 Pages 2006
Development and optimization of a useful assay for determining Hsp90’s inherent ATPase activity Fulltext Access 9 Pages 2006
Microwave-assisted synthesis of antimicrobial dihydropyridines and tetrahydropyrimidin-2-ones: Novel compounds against aspergillosis Fulltext Access 9 Pages 2006
3D QSAR on a library of heterocyclic diamidine derivatives with antiparasitic activity Fulltext Access 9 Pages 2006
Site-specific recombination of asymmetric lox sites mediated by a heterotetrameric Cre recombinase complex Fulltext Access 9 Pages 2006
Three-dimensional quantitative structure–activity relationship (3 D-QSAR) and docking studies on (benzothiazole-2-yl) acetonitrile derivatives as c-Jun N-terminal kinase-3 (JNK3) inhibitors Fulltext Access 9 Pages 2006
Steric interactions and the activity of fentanyl analogs at the μ-opioid receptor Fulltext Access 9 Pages 2006
Selection of a 2-azabicyclo[2.2.2]octane-based α4β1 integrin antagonist as an inhaled anti-asthmatic agent Fulltext Access 9 Pages 2006
New derivatives of xanthenone-4-acetic acid: Synthesis, pharmacological profile and effect on TNF-α and NO production by human immune cells Fulltext Access 9 Pages 2006
Studies on quinones. Part 41: Synthesis and cytotoxicity of isoquinoline-containing polycyclic quinones Fulltext Access 9 Pages 2006
Cytoprotective effect of caffeic acid phenethyl ester (CAPE) and catechol ring-fluorinated CAPE derivatives against menadione-induced oxidative stress in human endothelial cells Fulltext Access 9 Pages 2006
Novel antibiotics: C-2 symmetrical macrocycles inhibiting Holliday junction DNA binding by E. coli RuvC Fulltext Access 9 Pages 2006
Homology model of RSK2 N-terminal kinase domain, structure-based identification of novel RSK2 inhibitors, and preliminary common pharmacophore Fulltext Access 9 Pages 2006
Influence of rhamnose substituents on the potency of SL0101, an inhibitor of the Ser/Thr kinase, RSK Fulltext Access 9 Pages 2006
Efficient microwave enhanced regioselective synthesis of a series of benzimidazolyl/triazolyl spiro [indole-thiazolidinones] as potent antifungal agents and crystal structure of spiro[3H-indole-3,2′-thiazolidine]-3′(1,2,4-triazol-3-yl)-2,4′(1H)-dione Fulltext Access 9 Pages 2006
Synthesis and anti-HIV activity of new alkenyldiarylmethane (ADAM) non-nucleoside reverse transcriptase inhibitors (NNRTIs) incorporating benzoxazolone and benzisoxazole rings Fulltext Access 9 Pages 2006
Synthesis and characterization of novel hydrazide–hydrazones and the study of their structure–antituberculosis activity Fulltext Access 9 Pages 2006
Synthesis and biological properties of new α-methylene-γ-butyrolactones and α,β-unsaturated δ-lactones Fulltext Access 9 Pages 2006
Antibacterial and antifungal activity of acyclic and macrocyclic uracil derivatives with quaternized nitrogen atoms in spacers Fulltext Access 9 Pages 2006
Synthesis and in vitro activity of a series 1β-methylcarbapenem derivatives Fulltext Access 9 Pages 2006
Design and evaluation of “3 + 1” mixed ligand oxorhenium and oxotechnetium complexes bearing a nitroaromatic group with potential application in nuclear medicine oncology Fulltext Access 9 Pages 2006
In vitro mutagenicity of anti-inflammatory parsalmide analogues PA7, PA10, and PA31 triggered by biotransformation into hydroxy derivatives Fulltext Access 9 Pages 2006
Synthesis and antiproliferative activity of benzo[d]isothiazole hydrazones Fulltext Access 9 Pages 2006
Cytotoxic 5-aryl-1-(4-nitrophenyl)-3-oxo-1,4-pentadienes mounted on alicyclic scaffolds Fulltext Access 9 Pages 2006
Design, synthesis and antiproliferative activity of some new azapyranoxanthenone aminoderivatives Fulltext Access 9 Pages 2006
Synthesis and evaluation of 7-amino-2-(2(3)-furyl)-5-phenylethylamino-oxazolo[5,4-d]pyrimidines as potential A2A adenosine receptor antagonists for positron emission tomography (PET) Fulltext Access 9 Pages 2006
In vivo antitumor, in vitro antibacterial activity and alkylating properties of phosphorohydrazine derivatives of coumarin and chromone Fulltext Access 9 Pages 2006
Synthesis, characterization, antimicrobial and single crystal X-ray crystallographic studies of some new sulfonyl, 4-chloro phenoxy benzene and dibenzoazepine substituted benzamides Fulltext Access 9 Pages 2006
Nitrofurylsemicarbazone Rhenium and Ruthenium Complexes as Anti-trypanosomal Agents Fulltext Access 9 Pages 2006
Synthesis, structure, toxicological and pharmacological investigations of 4-hydroxycoumarin derivatives Fulltext Access 9 Pages 2006
Syntheses and odor of “bulky group”-modified sandalwood odorants: isophorono-β-santalol analogues Fulltext Access 9 Pages 2006
Air to fat and blood to fat distribution of volatile organic compounds and drugs: Linear free energy analyses Fulltext Access 9 Pages 2006
Structural modifications of benzanilide derivatives, effective potassium channel openers. X. Fulltext Access 9 Pages 2006
Antihelminthic activity of some newly synthesized 5(6)-(un)substituted-1H-benzimidazol-2-ylthioacetylpiperazine derivatives Fulltext Access 9 Pages 2006
Synthesis, crystal structure and anticancer activity of novel derivatives of ethyl 1-(4-oxo-8-aryl-4,6,7,8-tetrahydroimidazo[2,1-c][1,2,4]triazin-3-yl)formate Fulltext Access 9 Pages 2006
Air to brain, blood to brain and plasma to brain distribution of volatile organic compounds: linear free energy analyses Fulltext Access 9 Pages 2006
Synthesis and structure–activity relationships of retro bis-aminopyrrolidine urea (rAPU) derived small-molecule antagonists of the melanin-concentrating hormone receptor-1 (MCH-R1). Part 2 Fulltext Access 9 Pages 2006
Quantitative structure–activity analysis of 5-arylidene-2,4-thiazolidinediones as aldose reductase inhibitors Fulltext Access 9 Pages 2006
Identification of phosphodiesterase-1 and 5 dual inhibitors by a ligand-based virtual screening optimized for lead evolution Fulltext Access 9 Pages 2006