Stereoselective synthesis of optically active 1-substituted-1-pyridyl-methylamines

The stereoselective syntheses of chiral 1-substituted-1-(pyridyl)methylamines, bearing a stereogenic carbon bonded to the amino group and 2-, 3- or 4-position of the pyridine ring, are reviewed.

The stereoselective syntheses of chiral 1-substituted-1-(pyridyl)methylamines 1–3, bearing a chiral carbon bonded to the amino group and 2-, 3- or 4-position of the pyridine ring, are reviewed.Figure optionsDownload as PowerPoint slide