Estimation of thermodynamic acidity constants of some penicillinase-resistant penicillins Fulltext Access 5 Pages 2014
Synthesis and antiproliferative activity of conjugates of adenosine with muramyl dipeptide and nor-muramyl dipeptide derivatives Fulltext Access 5 Pages 2014
Design and synthesis of novel azapeptide activators of apoptosis mediated by caspase-9 in cancer cells Fulltext Access 5 Pages 2014
Structure-guided discovery of 1,3,5-triazine-pyrazole conjugates as antibacterial and antibiofilm agent against pathogens causing human diseases with favorable metabolic fate Fulltext Access 5 Pages 2014
Discovery of furan-2-carbohydrazides as orally active glucagon receptor antagonists Fulltext Access 5 Pages 2014
Curcumin glucuronides: Assessing the proliferative activity against human cell lines Fulltext Access 5 Pages 2014
A bicyclic peptide scaffold promotes phosphotyrosine mimicry and cellular uptake Fulltext Access 5 Pages 2014
The potential role of nano- and micro-technology in the management of critical illnesses Fulltext Access 5 Pages 2014
Quantification of total and unbound tranexamic acid in human plasma by ultrafiltration liquid chromatography/tandem mass spectrometry: Application to pharmacokinetic analysis Fulltext Access 5 Pages 2014
Detection of sibutramine in adulterated dietary supplements using attenuated total reflectance-infrared spectroscopy Fulltext Access 5 Pages 2014
Assessment of drug entrapment within liposomes using photophysical probes Fulltext Access 5 Pages 2014
Adenosine dry powder inhalation for bronchial challenge testing, part 2: Proof of concept in asthmatic subjects Fulltext Access 5 Pages 2014
Modulation by kynurenine of extracellular kynurenate and glutamate in cerebral cortex of rats with acute liver failure Fulltext Access 5 Pages 2014
Mortality in hypertensive patients with coronary heart disease depends on chronopharmacotherapy and dipping status Fulltext Access 5 Pages 2014
Evaluation of the clinical indications, adverse drug reactions, and finasteride use in patients with benign prostatic hyperplasia in Poland Fulltext Access 5 Pages 2014
Recombinant human interleukin 24 reverses Adriamycin resistance in a human breast cancer cell line Fulltext Access 5 Pages 2014
Buthionine sulfoximine diverts the melanogenesis pathway toward the production of more soluble and degradable pigments Fulltext Access 5 Pages 2014
Specific enrichment of nonribosomal peptide synthetase module by an affinity probe for adenylation domains Fulltext Access 5 Pages 2014
Antitrypanosomal structure-activity-relationship study of synthetic cynaropicrin derivatives Fulltext Access 5 Pages 2014
Design and synthesis of guanylthiourea derivatives as potential inhibitors of Plasmodium falciparum dihydrofolate reductase enzyme Fulltext Access 5 Pages 2014
Synthesis of long-chain fatty acid derivatives as a novel anti-Alzheimer's agent Fulltext Access 5 Pages 2014
Regioselective synthesis of 3-benzyl substituted pyrimidino chromen-2-ones and evaluation of anti-microbial and anti-biofilm activities Fulltext Access 5 Pages 2014
Modulation of adipose tissue thermogenesis as a method for increasing energy expenditure Fulltext Access 5 Pages 2014
Synthesis of licochalcone analogues with increased anti-inflammatory activity Fulltext Access 5 Pages 2014
Synthesis and anticancer potential of benzothiazole linked phenylpyridopyrimidinones and their diones as mitochondrial apoptotic inducers Fulltext Access 5 Pages 2014
New titanocene derivatives with high antiproliferative activity against breast cancer cells Fulltext Access 5 Pages 2014
Discovery of substituted benzamides as follicle stimulating hormone receptor allosteric modulators Fulltext Access 5 Pages 2014
The pharmacokinetics and hypoglycaemic effect of sunitinib in the diabetic rabbits Fulltext Access 5 Pages 2014
Kojyl cinnamate ester derivatives promote adiponectin production during adipogenesis in human adipose tissue-derived mesenchymal stem cells Fulltext Access 5 Pages 2014
Synthesis and pharmacological evaluation of novel limonin derivatives as anti-inflammatory and analgesic agents with high water solubility Fulltext Access 5 Pages 2014
Synthesis and discovery of highly functionalized mono- and bis-spiro-pyrrolidines as potent cholinesterase enzyme inhibitors Fulltext Access 5 Pages 2014
Synthesis and biological evaluation of a series of benzoxazole/benzothiazole-containing 2,3-dihydrobenzo[b][1,4]dioxine derivatives as potential antidepressants Fulltext Access 5 Pages 2014
Synthesis and evaluation of new diaryl ether and quinoline hybrids as potential antiplasmodial and antimicrobial agents Fulltext Access 5 Pages 2014
Synthesis and evaluation of amide side-chain modified Agomelatine analogues as potential antidepressant-like agents Fulltext Access 5 Pages 2014
Inhibition of biofilm formation by conformationally constrained indole-based analogues of the marine alkaloid oroidin Fulltext Access 5 Pages 2014
Synthesis and biological evaluation of (+)-neopeltolide analogues: Importance of the oxazole-containing side chain Fulltext Access 5 Pages 2014
Anticancer phytochemical analogs 37: Synthesis, characterization, molecular docking and cytotoxicity of novel plumbagin hydrazones against breast cancer cells Fulltext Access 5 Pages 2014
The enone motif of (+)-grandifloracin is not essential for 'anti-austerity' antiproliferative activity Fulltext Access 5 Pages 2014
Fullerene derivatives as a new class of inhibitors of protein tyrosine phosphatases Fulltext Access 5 Pages 2014
Heterocyclic acyl-phosphate bioisostere-based inhibitors of Staphylococcus aureus biotin protein ligase Fulltext Access 5 Pages 2014
Synthesis and biological evaluation of isoprenylated coumarins as potential anti-pancreatic cancer agents Fulltext Access 5 Pages 2014
Beta-aminoketones as prodrugs for selective irreversible inhibitors of type-1 methionine aminopeptidases Fulltext Access 5 Pages 2014
Design, synthesis and biological evaluation of metronidazole–thiazole derivatives as antibacterial inhibitors Fulltext Access 5 Pages 2014
Synthesis and biological evaluation of a novel class of coumarin derivatives Fulltext Access 5 Pages 2014
Structure–activity relationship studies of antiplasmodial aminomethylthiazoles Fulltext Access 5 Pages 2014
Carbonic anhydrase inhibitory activity of sulfonamides and carboxylic acids incorporating cyclic imide scaffolds Fulltext Access 5 Pages 2014
Interaction kinetics of liposome-incorporated unsaturated fatty acids with fatty acid-binding protein 3 by surface plasmon resonance Fulltext Access 5 Pages 2014
Bicyclic brominated furanones: A new class of quorum sensing modulators that inhibit bacterial biofilm formation Fulltext Access 5 Pages 2014
Development of a new class of proteasome inhibitors with an epoxyketone warhead: Rational hybridization of non-peptidic belactosin derivatives and peptide epoxyketones Fulltext Access 5 Pages 2014
Inhibitory and mechanistic investigations of oxo-lipids with human lipoxygenase isozymes Fulltext Access 5 Pages 2014
Synthesis and structure–activity relationship of thiobarbituric acid derivatives as potent inhibitors of urease Fulltext Access 5 Pages 2014
The effect of assay type and sample matrix on detected cytokine concentrations in human blood serum and nasal lavage fluid Fulltext Access 5 Pages 2014
Gas chromatographic–mass spectrometric analysis and subsequent quality improvement of plastic infusion packaging materials Fulltext Access 5 Pages 2014
Identification and quantitation of the ingredients in a counterfeit Vietnamese herbal medicine against rheumatic diseases Fulltext Access 5 Pages 2014
Chromatographic separation and biological evaluation of benzimidazole derivative enantiomers as inhibitors of leukotriene biosynthesis Fulltext Access 5 Pages 2014
A carbon nanotubes based fluorescent aptasensor for highly sensitive detection of adenosine deaminase activity and inhibitor screening in natural extracts Fulltext Access 5 Pages 2014
A micellar liquid chromatography method for the quantification of abacavir, lamivudine and raltegravir in plasma Fulltext Access 5 Pages 2014
Separation and structural elucidation of a new tadalafil analogue diethylaminopretadalafil included as an adulterant in a dietary supplement Fulltext Access 5 Pages 2014
Rapid process development of chromatographic process using direct analysis in real time mass spectrometry as a process analytical technology tool Fulltext Access 5 Pages 2014
Chronic treatment with zinc hydroaspartate induces anti-inflammatory and anti-ulcerogenic activity in rats Fulltext Access 5 Pages 2014
Phenylbutazone and ketoprofen binding to serum albumin. Fluorescence study Fulltext Access 5 Pages 2014
Oral dosing in adult zebrafish: Proof-of-concept using pharmacokinetics and pharmacological evaluation of carbamazepine Fulltext Access 5 Pages 2014
Inhibition of sphingosine kinase-2 ablates androgen resistant prostate cancer proliferation and survival Fulltext Access 5 Pages 2014
Assessment of antioxidant supplementation on the neuropathic pain score and quality of life in diabetic neuropathy patients – A randomized controlled study Fulltext Access 5 Pages 2014
A new method for filtering of reactive “warheads” of transition-state analog protease inhibitors Fulltext Access 5 Pages 2014
Novel insights on the structural determinants of clozapine and olanzapine multi-target binding profiles Fulltext Access 5 Pages 2014
A one-pot approach to bio-synthesize globotriose and its derivatives from simpler substrates Fulltext Access 5 Pages 2014
Synthesis and evaluation of new 3-phenylcoumarin derivatives as potential antidepressant agents Fulltext Access 5 Pages 2014
The effect of short-term simvastatin treatment on plasma adipokine levels in patients with isolated hypercholesterolemia: A preliminary report Fulltext Access 5 Pages 2014
Synthesis and biological evaluation of new boron-containing chlorin derivatives as agents for both photodynamic therapy and boron neutron capture therapy of cancer Fulltext Access 5 Pages 2014
The survival times of malaria-infected mice are prolonged more by several new two-carbon-linked artemisinin-derived dimer carbamates than by the trioxane antimalarial drug artemether Fulltext Access 5 Pages 2014
Multisubstituted indole–acrylonitrile hybrids as potential cytotoxic agents Fulltext Access 5 Pages 2014
Synthesis and radical scavenging activity of phenol–imidazole conjugates Fulltext Access 5 Pages 2014
Synthesis and biological evaluation of compounds which contain pyrazole, thiazole and naphthalene ring as antitumor agents Fulltext Access 5 Pages 2014
Synthesis and biological activities of 2,3-dihydro-1,3,4-oxadiazole compounds and its derivatives as potential activator of ryanodine receptors Fulltext Access 5 Pages 2014
Design, synthesis, docking and anti-inflammatory evaluation of novel series of benzofuran based prodrugs Fulltext Access 5 Pages 2014
Substituted dithiazole piperazine benzamides as novel amyloid beta peptide reducing agents Fulltext Access 5 Pages 2014
Synthesis, antioxidant and photoprotection activities of hybrid derivatives useful to prevent skin cancer Fulltext Access 6 Pages 2014
Discovery of the rapanone and suberonone mixture as a motif for leishmanicidal and antifungal applications Fulltext Access 6 Pages 2014