
Synthesis and biological evaluation of pyrido[2,3-d]pyrimidine-2,4-dione derivatives as eEF-2K inhibitors
Keywords: eEF-2K, eukaryotic elongation factor-2 kinase; 2-DOG, 2-deoxy-d-glucose; DMF, dimethylformamide; DMSO, dimethylsulfoxidePyrido[2,3-d]pyrimidine-2,4-dione; Uracil; eEF-2K inhibitor; Kinase inhibitor; Homology modeling