
Synthesis and biological evaluation of 2-anilino-4-substituted-7H-pyrrolopyrimidines as PDK1 inhibitors
Keywords: 3-Phosphoinositide-dependent kinase 1 (PDK1); 2-Anilino-4-substituted-pyrrolopyrimidines; Inhibitor; Suzuki cross-coupling; Buchwald–Hartwig cross-coupling