Keywords: پروتئین فعال 5-لیپوکسیژناز; Chromatographic enantioisolation; Polysaccharide-based stationary phases; 5-Lipoxygenase-activating protein; FLAP; Benzimidazole
مقالات ISI پروتئین فعال 5-لیپوکسیژناز (ترجمه نشده)
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Natural products as inhibitors of prostaglandin E2 and pro-inflammatory 5-lipoxygenase-derived lipid mediator biosynthesis
Keywords: پروتئین فعال 5-لیپوکسیژناز; AA; arachidonic acid; ABA; 3-O-acetyl-boswellic acid; AKBA; 3-O-acetyl-11-keto-boswellic acid; BA; boswellic acid; COX; cyclooxygenase; EGCG; epigallocatechin-3-gallate; FLAP; 5-lipoxygenase-activating protein; H(P)ETE; hydro(pero)xyeicosatetraenoic acid;
Identification of multi-target inhibitors of leukotriene and prostaglandin E2 biosynthesis by structural tuning of the FLAP inhibitor BRP-7
Keywords: پروتئین فعال 5-لیپوکسیژناز; 5-Lipoxygenase-activating protein; 5-Lipoxygenase; Microsomal prostaglandin E2 synthase-1; Leukotriene; Benzimidazole; Inflammation;
Too much of a good thing: How modulating LTB4 actions restore host defense in homeostasis or disease
Keywords: پروتئین فعال 5-لیپوکسیژناز; LT; leukotriene; PAMP; pathogen associated molecular patterns; PRR; pattern recognition receptor; AA; arachidonic acid; LO; lipoxygenase; cPLA2; cytosolic phospholipase A2; FLAP; 5-lipoxygenase-activating protein; cysLT; cysteinyl LT; BLT; B leukotriene r
Development of smart cell-free and cell-based assay systems for investigation of leukotriene C4 synthase activity and evaluation of inhibitors
Keywords: پروتئین فعال 5-لیپوکسیژناز; 5-LOX; 5-Lipoxygenase; AA; Arachidonic acid; FLAP; 5-Lipoxygenase-activating protein; GSH; Glutathione; LT; Leukotriene; LTA4H; Leukotriene A4 hydrolase; cys-LTs; Cysteinyl leukotrienes; MAPEG; Membrane-associated protein in eicosanoid and glutathione met
4,5-Diarylisoxazol-3-carboxylic acids: A new class of leukotriene biosynthesis inhibitors potentially targeting 5-lipoxygenase-activating protein (FLAP)
Keywords: پروتئین فعال 5-لیپوکسیژناز; Inflammation; Leukotrienes; 5-lipoxygenase; 5-lipoxygenase-activating protein; Isoxazole
Synthesis and biological evaluation of C(5)-substituted derivatives of leukotriene biosynthesis inhibitor BRP-7
Keywords: پروتئین فعال 5-لیپوکسیژناز; Leukotriene; 5-Lipoxygenase-activating protein; FLAP; Benzimidazole; BRP-7
BRP-187: A potent inhibitor of leukotriene biosynthesis that acts through impeding the dynamic 5-lipoxygenase/5-lipoxygenase-activating protein (FLAP) complex assembly
Keywords: پروتئین فعال 5-لیپوکسیژناز; 5-LO; 5-lipoxygenase; AA; arachidonic acid; COX; cyclooxygenase; cPLA2; cytosolic phospholipase A2; FLAP; 5-lipoxygenase-activating protein; fMLP; N-formyl-methionyl-leucyl-phenylalanine; H(P)ETE; hydro(pero)oxyeicosatetraenoic acid; HHT; hydroxyheptadeca
Characterization of the interaction of human 5-lipoxygenase with its activating protein FLAP
Keywords: پروتئین فعال 5-لیپوکسیژناز; 5-H(p)ETE; 5S-hydro(pero)xy-6,8,11,14(E,Z,Z,Z)-eicosatetraenoic acid; 6-trans-LTB4; 5S,12R-dihydroxy-6,8,10,14(E,E,E,Z)-eicosatetraenoic acid; 6-trans-12-epi-LTB4; 5S,12S-dihydroxy-6,8,10,14-(E,E,E,Z)-eicosatetraenoic acid; Aa; amino acid; AA; arachidonic
Identification of novel benzimidazole derivatives as inhibitors of leukotriene biosynthesis by virtual screening targeting 5-lipoxygenase-activating protein (FLAP)
Keywords: پروتئین فعال 5-لیپوکسیژناز; AA; arachidonic acid; cPLA2; cytosolic phospholipase A2; FLAP; 5-lipoxygenase-activating protein; 5-HpETE; 5-hydroperoxyeicosatetraenoic acid; 5-LO; 5-lipoxygenase; LT; leukotriene; PGC buffer; phosphate-buffered saline pH 7.4 containing 1Â mg/mL glucose
Development of 5-lipoxygenase inhibitors-lessons from cellular enzyme regulation
Keywords: پروتئین فعال 5-لیپوکسیژناز; AA; arachidonic acid; cPLA2; cytosolic phospholipase A2; FLAP; 5-lipoxygenase-activating protein; fMLP; N-formyl-methionyl-leucyl-phenylalanin; GM-CSF; granulocyte macrophage colony-stimulating factor; GPx; glutathione peroxidase; LPS; lipopolysaccharide;
Attenuation of breast tumor cell growth by conjugated linoleic acid via inhibition of 5-lipoxygenase activating protein
Keywords: پروتئین فعال 5-لیپوکسیژناز; AA; arachidonic acid; CLA; conjugated linoleic acid; t10, c12-CLA; trans10, cis12-CLA; c9, t11-CLA; cis9, trans11-CLA; DMEM; Dulbecco's modified eagle media; 5-HETE; 5-hydroxyeicosatetraenoic acid; 13-HODE; 13-hydroxyoctadecadienoic acid; COX-2; cyclooxyg