Keywords: Biphalin; Opioid receptors; MOR/DOR/KOR agonist; Synergistic analgesic effect; Cyclic peptides; Acm; acetamidomethyl; ACN; acetonitrile; BBB; blood brain barrier; Boc; t-butyloxycarbonyl; BOP; (benzotriazol-1-yloxytris(dimethylamino)phosphonium hexafluoro
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Intelligent substance delivery into cells using cell-penetrating peptides
Keywords: CPP; cell-penetrating peptide; PTD; protein transduction domain; siRNA; small interfering ribonucleic acid; HIV-1; human immunodeficiency virus 1; Arg; arginine; Lys; lysine; Rn; polyarginine composed of n arginines, where n is natural number; a.a.; amino
Keywords: RNCGDQLZIATDOU-ZDRBWGSPSA-N; ICYPJNZJUFGALC-PDTBJYIYSA-N; PDRMAVOIWIVXKH-SFUSBHMVSA-N; ISADXJRTBSLWPX-ZDRBWGSPSA-N; NLBLLPROASDPSC-QWWZWVQMSA-N; XKMIKZDBUOHHDK-ZDRBWGSPSA-N; BTURADNXKHTWGA-IJOLSIAMSA-N; UEKHRDLXBMZMPD-ZYIYBEKCSA-N; UQCLCXDOXVZEOA-JARUQAPT
Keywords: Boc; t-butyloxycarbonyl; Boc-Lys(Boc)-Osu; Nα,Nε-di-Boc-l-lysine hydroxysuccinimide ester; BSA; bovine serum albumin; Cbz; carboxybenzyl; CLRs; C-type lectin receptors; CRD; carbohydrate-recognition domain; Con A; Concanavaline A; DBU; 1,8-diazabicyclo[
Keywords: Ac; acetyl; acac; acetylacetonate; AHPCS; allylhydridopolycarbosilane; Bn; benzyl; Boc; tert-butoxycarbonyl; BPR; back pressure regulator; bpy; 2,2â²-bipyridine; Bu; butyl; CFL; compact fluorescent lamp; DCB; 1,4-dicyanobenzene; de; diastereomeric excess
Keywords: SPPS; solid phase peptide synthesis; DMF; dimethyl formamide; DIPEA; diisopropylethylamine; DIPC; diisopropylcarbodiimide; HOBt; 1-hydroxybenzotriazole; Fmoc; 9-fluorenylmethyloxycarbonyl; HFIP; 1,1,1,3,3,3-hexafluoropropan-2-ol; TFA; trifluoroacetic acid
Development of potent and proteolytically stable human neuromedin U receptor agonists
Keywords: Neuromedin U (NMU); NMU-8; Neuromedin U receptor agonists; Plasma stability; 1â²Nal; 1â²-naphtylalanine; 2â²Nal; 2â²-naphtylalanine; 7-OH-Tic; 7-hydroxy-L-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid; ACN; acetonitrile; AUC; area under the curve;
Comparison of extracellular Cys/Trp motif between Schizosaccharomyces pombe Ctr4 and Ctr5
Keywords: Ctr; copper transporter; BCA; bicinchoninic acid; Fmoc; 9-fluorenylmethyloxycarbonyl; NMP; N-methylpyrrolidone; HBTU; 2-(1H-benzotriazol-1-yl)-1,1,3,3-tetramethyluronium hexafluorophosphate; HOBt; 1-hydroxybenzotriazol; DIEA; N,N-diisopropylethylamine; DM
Design of strategies to study the metabolic profile of highly polar compounds in plasma by reversed-phase liquid chromatography-high resolution mass spectrometry
Keywords: 9-Fluorenylmethyloxycarbonyl; Hydrophilic compounds; Liquid chromatography-high resolution mass spectrometry; Metabolic profile; Plasma; Ultrafiltration;
Ala5-galanin (2-11) is a GAL2R specific galanin analogue
Keywords: BBB; blood-brain barrier; CHO cells; Chinese hamster ovary cells; CNS; central nervous system; EDTA; ethylenediaminetetraacetic acid; FBS; fetal bovine serum; Fmoc; 9-fluorenylmethyloxycarbonyl; FSK; forskolin; GAL1R; Galanin receptor 1; GAL2R; Galanin re
Structure-activity relationship study of syringolin A as a potential anticancer agent
Keywords: Fmoc; 9-fluorenylmethyloxycarbonyl; EDCI; 1-ethyl-3-(3-dimethylaminopropyl)carboxamide; HOBt; 1-hydroxybenzotriazole; DMF; N,N-dimethylformamide; Proteasome inhibitor; Cancer; Structure-activity relationship;
Synthetic study of peptide aldehyde via acetal/thioacetal transformation: application for Lys/Ser-containing peptides
Keywords: Peptide aldehyde; Acetal; Thioacetal; Cysteine protease inhibitor; SPPS; solid phase peptide synthesis; NBS; N-bromo succinimide; SARS; severe acute respiratory syndrome; DMF; dimethyl formamide; DIPEA; diisopropylethylamine; DIPC; diisopropylcarbodiimide
A novel synthetic luteinizing hormone-releasing hormone (LHRH) analogue coupled with modified β-cyclodextrin: Insight into its intramolecular interactions
Keywords: BOP; benzotriazole-1-yl-oxy-tris-(dimethylamino)-phosphonium hexafluorophosphate; CLTR-Cl; 2-chlorotrityl chloride; DCC; N,Nâ²-dicyclohexylcarbodiimide; DMA; dimethylacetamide; DIC; N,Nâ²-diisopropylcarbodiimide; DIEA; diisopropylethylamine; DMF; N,N-di
Reevaluation of the rate constants for the reaction of hypochlorous acid (HOCl) with cysteine, methionine, and peptide derivatives using a new competition kinetic approach
Keywords: DTDPA; 3,3â²-dithiodipropionic acid; Fmoc; 9-fluorenylmethyloxycarbonyl; Fmoc-Met; 9-fluorenylmethyloxycarbonyl-tagged methionine; Fmoc-MetSO; 9-fluorenylmethyloxycarbonyl-tagged methionine sulfoxide; HOBr; the physiological mixture of hypobromous acid a
Potency optimization of Huwentoxin-IV on hNav1.7: A neurotoxin TTX-S sodium-channel antagonist from the venom of the Chinese bird-eating spider Selenocosmia huwena
Keywords: ACF; animal-component free; BSA; bovine serum albumin; CaCl2; calcium chloride; CD; circular dichroism spectroscopy; CHO; Chinese hamster ovary; CNS; central nervous system; CO2; carbon dioxide; CsF; cesium fluoride; CsOH; cesium hydroxide; DIC; diisoprop
Design, synthesis and evaluation of antimicrobial activity of N-terminal modified Leucocin A analogues
Keywords: AMP; antimicrobial peptide; CD; circular dichroism; DIC; 1,3-diisopropylcarbodiimide; Fmoc; 9-fluorenylmethyloxycarbonyl; HOBt; N-hydroxybenzotriazole; RP-HPLC; reversed phase high performance liquid chromatography; LAB; lactic acid bacteria; LeuA; Leucoc
Backbone cyclic helix mimetic of chemokine (C-C motif) receptor 2: A rational approach for inhibiting dimerization of G protein-coupled receptors
Keywords: ACN; acetonitrile allocallyloxycarbonyl; BBB; blood brain barrier; Boc; t-butyloxycarbonyl; BTC; bis(trichloromethyl)carbonate; CCR2; chemokine (C-C motif) receptor 2; CCR5; chemokine (C-C motif) receptor 5; CNS; central nervous system; DIPEA; diisopr
Conotoxin truncation as a post-translational modification to increase the pharmacological diversity within the milked venom of Conus magus
Keywords: Conotoxins; N-terminal modification; Milked venom; Post-translational modification; α-Conotoxin; Mass spectrometry; API; Atmospheric pressure ionization; Arg(Pbf); N-alpha-9-fluorenylmethoxycarbonyl-N-g-2,2,4,6,7-pentamethyldihydrobenzofuran-5-sulfonyl-l
Radiochemical and radiobiological assessment of a pyridyl-S-cysteine functionalized bombesin derivative labeled with the 99mTc(CO)3+ core
Keywords: Boc; t-butyloxycarbonyl; BSA; bovine serum albumin; Cys; cysteine; DIEA; N,N-diisopropylethylamine; DIC; diisopropylcarbamide; DMEM; Dulbecco's modified Eagle medium; DMF; dimethylformamide; EDTA; ethylenediaminetetraacetic acid; ESI-MS; electrospray io
A 'conovenomic' analysis of the milked venom from the mollusk-hunting cone snail Conus textile-The pharmacological importance of post-translational modifications
Keywords: αα; amino acid; CH3CN; acetonitrile; Acm; acetamidomethyl; API; atmospheric pressure ionization; DHB; dihydroxybenzoic acid; cDNA; complimentary DNA; CHCA; α-Cyano-4-hydroxycinnamic acid; CID; collision induced dissociation; DCM; dichloromethane; DIEA;
Colicin M hydrolyses branched lipids II from Gram-positive bacteria
Keywords: Branched lipid II; Chemo-enzymatic synthesis; Colicin M; Gram-positive bacteria; Peptidoglycan; A2pm; diaminopimelic acid; ColM; colicin M; Fmoc; 9-fluorenylmethyloxycarbonyl; HPLC; high-performance liquid chromatography; iAsn; isoasparagine; MALDI-TOF; m
Cyanoacetamide-based oxime carbonates: an efficient, simple alternative for the introduction of Fmoc with minimal dipeptide formation
Keywords: Amino acids; 9-Fluorenylmethyloxycarbonyl; Oxime; N-Protecting group; Peptide synthesis; Boc; tert-butoxycarbonyl; DCM; dichloromethane; ESI-MS; electrospray ionization mass spectrometry; Fmoc; fluorenylmethyloxycarbonyl; NMR; nuclear magnetic resonance;
Synthesis and comparative assessment of a labeled RGD peptide bearing two different 99mTc-tricarbonyl chelators for potential use as targeted radiopharmaceutical
Keywords: Arg/R; arginine; Asp/D; aspartic acid; Boc; t-butyloxycarbonyl; BSA; bovine serum albumin; CPA; 3-l-cysteine propionic acid; Cys; cysteine; d-Phe/f; d-phenylalanine; DIEA; N,N-diisopropylethylamine; DIPC; diisopropylcarbamide; DMEM; Dulbecco's modified
Functional and physical competition between phospholamban and its mutants provides insight into the molecular mechanism of gene therapy for heart failure
Keywords: Ca2+; divalent calcium ion; Dabcyl-SE; 4-((4-(dimethylamino)phenyl)azo)-benzoic acid succinimidyl ester; Fmoc; 9-fluorenylmethyloxycarbonyl; FRET; fluorescence resonance energy transfer; IAEDANS; 5-((((2-iodoacetyl)amino)ethyl)amino) naphthalene-1-sulfoni
Synthesis of a-factor peptide from Saccharomyces cerevisiae and photoactive analogues via Fmoc solid phase methodology
Keywords: Boc; tert-butyloxycarbonyl; Br-BC5; [(E)-(3-((4-bromo-2-methylbut-2-enyloxy)methyl)phenyl)-(phenyl)methanone]; Br-BC10; [(3-(((2E,6E)-8-bromo-2,6-dimethylocta-2,6-dienyloxy)methyl)-phenyl)(phenyl)methanone]; t-Bu; tert-butyl; CLEAR; cross-linked ethoxylat
Protection against malaria is conferred by passive transferring rabbit F(ab)2â² antibody fragments, induced by Plasmodium falciparum MSP-1 site-directed designed pseudopeptide-BSA conjugates assessed in a rodent model
Keywords: F(ab)â²2; antibody fragment for antigen binding; HABP; high activity binding peptide; Ï-[CH2NH]; reduced amide isoster bond; MHC; major histocompatibility complex; TCR; T-cell receptor; TCC; T-cell clone; APC; antigen presenting cell; CDR; complimentari
Rational conversion of noncontinuous active region in proteins into a small orally bioavailable macrocyclic drug-like molecule: The HIV-1 CD4:gp120 paradigm
Keywords: AcOH; acetic acid; Alloc; allyloxycarbonyl; Boc; t-butoxycarbonyl; BTC; bis(trichloromethyl)carbonate; DBU; 1,8-diazabicyclo[5.4.0]undec-7-ene; DCM; methylene chloride; DIC; N,Nâ²-diisopropylcarbodiimide; DIPEA; diisopropylethylamine; DMAP; dimethylamino
Photoaffinity labeling of Ras converting enzyme 1 (Rce1p) using a benzophenone-containing peptide substrate
Keywords: Abz; 2-aminobenzoyl; C5BP; 3-methylbenzophenone prenyl ether; CLEAR; crosslinked ethoxylate acrylate resin; Dde; 1-(4,4-dimethyl-2,6-dioxocyclohexylidene) ethyl; DI; deionized; DIEA; diisopropylethylamine; DMF; N,N-dimethylformamide; DMSO; dimethyl sulfox
Characterization of a conformationally sensitive TOAC spin-labeled substance P
Keywords: NK1r; neurokinin-1 receptor; SP; substance P; 4-TOAC SP; TOAC substance P with TOAC integrated at position 4; 9-TOAC SP; TOAC substance P with the TOAC spin label integrated at position 9; Nk1r; neurokinin-1 receptor; EPR; electron paramagnetic resonance
Synthesis of thiol-modified peptide nucleic acids designed for post-assembly conjugation reactions
Keywords: Peptide nucleic acid; Conjugation; Solid-phase synthesis; Boc; t-butyloxycarbonyl; Bhoc; benzhydryloxycarbonyl; DTT; dithiothreitol; Fmoc; 9-fluorenylmethyloxycarbonyl; PMB; para-methoxybenzyl; EDC; N-(3-dimethylaminopropyl)-Nâ²-ethylcarbodiimide hydroch
Importance of N- and C-terminal regions of gastrin-Gly for preferential binding to high and low affinity gastrin-Gly receptors
Keywords: BSA; bovine serum albumin; CCK-8; cholecystokinin-8; DIEA; N,N-diisopropylethylamine; DMF; N,N-dimethylformamide; DMSO; dimethylsulfoxide; ESI-MS; electrospray ionization mass spectrometry; FCS; fetal calf serum; Fmoc; 9-fluorenylmethyloxycarbonyl; G17; g
Targeting small-cell lung cancer with novel fluorescent analogs of somatostatin
Keywords: BSA; bovine serum albumin; CHO; Chinese hamster ovary; DABA; 2,4-diaminobutyric acid; DIEA; N,N-diisopropyl ethyl amine; DMSO; dimethyl sulfoxide; ESI-MS; electrospray ionization mass spectrometer; Fmoc; 9-fluorenylmethyloxycarbonyl; HPLC; high performanc