Keywords: گیرنده آدنوزین A3; Adenosine; Adenosine receptor; Drug target; Drug discovery; Pharmacology; Disease; T1D; type 1 diabetes; T2D; type 2 diabetes; A1AR; A1 adenosine receptor; A2AAR; A2A adenosine receptor; A2BAR; A2B adenosine receptor; A3AR; A3 adenosine receptor;
مقالات ISI گیرنده آدنوزین A3 (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: گیرنده آدنوزین A3; ATP; adenosine triphosphate; ECM; extracellular matrix; DAMPs; danger-associated molecular patterns; ENTPDase; ectonucleotidase triphosphate diphosphohydrolase; ENPPS; ectonucleotide pyrophosphatase/phosphodiesterase; RanBPM; ran binding protein; E-NTPDas
Anticancer activity study of A3 adenosine receptor agonists
Keywords: گیرنده آدنوزین A3; AC; adenylyl cyclase; A3AR; A3 Adenosine receptor; Caco-2; epithelial colorectal carcinoma; CHO; Chinese hamster ovary; Cl-IB-MECA; 2-chloro-N6-(3-iodobenzyl)-adenosine-5â²-N-methyluronamide; DMEM; Dulbecco's modified eagle medium; DMSO; dimethyl sulphox
Molecular dissection of the human A3 adenosine receptor coupling with β-arrestin2
Keywords: گیرنده آدنوزین A3; A3 adenosine receptor; β-Arrestin2; Nanoluciferase; Functional complementation; Live-cell reporter assay;
Probing structure-activity relationship in β-arrestin2 recruitment of diversely substituted adenosine derivatives
Keywords: گیرنده آدنوزین A3; G protein-coupled receptor; A3 adenosine receptor; β-arrestin2; Structure-activity relationship; Biased signaling;
Down-regulation of the A3 adenosine receptor in human mast cells upregulates mediators of angiogenesis and remodeling
Keywords: گیرنده آدنوزین A3; Mast cells; Adenosine; A3 adenosine receptor; HMC-1 cells; Tissue remodelingARs, adenosine receptors; A3R, adenosine-3-receptor; AREG, amphiregulin; Cl-IB-MECA, 2-chloro-N6-(3-iodobenzyl)-adenosine-5′-N-methyluronamide; Dex, dexamethasone; IL1β, Interleuk
Adenosine A3 receptor activation is neuroprotective against retinal neurodegeneration
Keywords: گیرنده آدنوزین A3; A3 adenosine receptor; Retinal ganglion cell; Neuroprotection; Excitotoxicity; Ischemia-reperfusion; Axon injury; A3R; A3 receptor; AMPA; α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid; CTZ; cyclothiazide; DARC; Detection of Apoptosing Retinal Cell
Simple synthesis of new carbon-11-labeled 1,2,4-triazolo[4,3-a]quinoxalin-1-one derivatives for PET imaging of A3 adenosine receptor
Keywords: گیرنده آدنوزین A3; Carbon-11-labeled 1,2,4-triazolo[4,3,a]quinoxalin-1-one derivatives; A3 adenosine receptor; Positron emission tomography (PET); Neurological disorders; Cardiac diseases; Cancer
Adenosine receptors and cancer
Keywords: گیرنده آدنوزین A3; A1 adenosine receptor; A2A adenosine receptor; A2B adenosine receptor; A3 adenosine receptor; Cancer; Molecular mechanism
The A3 adenosine receptor attenuates the calcium rise triggered by NMDA receptors in retinal ganglion cells
Keywords: گیرنده آدنوزین A3; A3 adenosine receptor; NMDA receptor; Glutamate; ATP; Purinergic signaling; Neuroprotection; Excitotoxicity; Retinal ganglion cells
Stimulation of the P2X7 receptor kills rat retinal ganglion cells in vivo
Keywords: گیرنده آدنوزین A3; P2X receptor; A3 adenosine receptor; purinergic signaling; retinal ganglion cells; neuroprotection; in vivo models
Synthesis and evaluation of new N6-substituted adenosine-5′-N-methylcarboxamides as A3 adenosine receptor agonists
Keywords: گیرنده آدنوزین A3; Adenosine agonist; A3 Adenosine receptor; Cardioprotection
Molecular docking study of A3 adenosine receptor antagonists and pharmacophore-based drug design
Keywords: گیرنده آدنوزین A3; A3 adenosine receptor; Antagonist; Docking; Pharmacophore-based virtual library screening
Structure–activity relationships of truncated adenosine derivatives as highly potent and selective human A3 adenosine receptor antagonists
Keywords: گیرنده آدنوزین A3; A3 Adenosine receptor; Antagonists; Truncated adenosine; Structure–activity relationships
The anti-inflammatory target A3 adenosine receptor is over-expressed in rheumatoid arthritis, psoriasis and Crohn’s disease
Keywords: گیرنده آدنوزین A3; A3 adenosine receptor; ADORA3; Crohn’s disease; Psoriasis; Rheumatoid arthritis; NF-κB; CREB; PI3K-PKB/Akt; Inflammation
Design and synthesis of N6-substituted-4′-thioadenosine-5′-uronamides as potent and selective human A3 adenosine receptor agonists
Keywords: گیرنده آدنوزین A3; A3 adenosine receptor; 4′-Thionucleosides; Agonist; Binding affinity
A novel adenosine analog, thio-Cl-IB-MECA, induces G0/G1 cell cycle arrest and apoptosis in human promyelocytic leukemia HL-60 cells
Keywords: گیرنده آدنوزین A3; A3AR; A3 adenosine receptor; thio-Cl-IB-MECA; 2-chloro-N6-(3-iodobenzyl)-4â²-thioadenosine-5â²-N-methyluronamide; A3 adenosine receptor agonist; Thio-Cl-IB-MECA; HL-60 cells; Cell cycle arrest; Apoptosis; Wnt signaling;
A3 adenosine receptor-mediated protection of the ischemic heart
Keywords: گیرنده آدنوزین A3; Adenosine; A3 adenosine receptor; Cardioprotection; Ischemia-reperfusion; Myocardial infarction; Stunning;