
1,2,4-Triazolsulfone: A novel isosteric replacement of acylsulfonamides in the context of NaV1.7 inhibition
Keywords: آکیل سولفون آمید; 3-(Sulfonyl)-1,2,4-triazole; Triazolesulfone; Bioisostere; Acylsulfonamide; pKa; Sodium channel; NaV1.7; NaV1.5; Pain;