
Preclinical pharmacology of FL442, a novel nonsteroidal androgen receptor modulator
Keywords: ADT, androgen-deprivation therapy; AF2, activation function 2; AhR, aryl hydrocarbon receptor; AR, androgen receptor; Bic, bicalutamide; CAR, constitutive androstane receptor; COS-1, African green monkey kidney cells; CRPC, castration resistant prostate c