Keywords: 5-HT; 5-Hydroxytryptamine or serotonin; AA-5-HT; N-arachidonoyl-serotonin; ACEA; arachidonoyl 2â²-chloroethylamide; AEA; N-arachidonoylethanolamine; 2-AG; 2-arachidonoylglycerol; AM251; N-(piperidin-1-yl)-5-(4-iodophenyl)-1-(2,4-dichlorophenyl)-4-methyl-
مقالات ISI (ترجمه نشده)
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SGIP1 alters internalization and modulates signaling of activated cannabinoid receptor 1 in a biased manner
Keywords: Seven transmembrane receptors; G-protein coupled receptors; Cannabinoid receptor 1; Protein-protein interactions; Bias signaling; Receptor endocytosis; SGIP1; src homology 3-domain growth factor receptor-bound 2-like (endophilin) interacting protein 1; CC
Evaluation of the abuse potential of AM281, a new synthetic cannabinoid CB1 receptor antagonist
Keywords: AM281; Cannabinoid antagonist; Abuse potential; Conditioned place preference; Self-administration
The non-selective cannabinoid receptor agonist WIN 55,212-2 attenuates responses of C-fiber nociceptors in a murine model of cancer pain
Keywords: ANOVA; analysis of variance; CM; C-mechanonociceptors; CMH; C-mechanoheat nociceptors; CV; conduction velocity; DRG; dorsal root ganglion; IQR; interquartile range; PBS; phosphate-buffered saline; PID; post-implantation day; TRP; transient receptor potent
Role of endocannabinoid and glutamatergic systems in DOI-induced head-twitch response in mice
Keywords: ADHD; Attention-deficit/hyperactivity disorder; AM281; N-(piperidin-1-yl)-5-(4-iodophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide; AM404; N-(4-hydroxyphenyl)arachidonylamide; AMPA; α-amino-3-hydroxy-5-methyl-4-isoxazolepropionate; Anan
Synthesis and preliminary biological evaluation of [123I]Me2Pyr, a new potential ligand for imaging of central cannabinoid CB1 receptors
Keywords: Iodine-123, -125; Cannabinoid CB1 receptors; SR141716A; Diaryl pyrazoles; Tributylstannyl precursors; Radioiododestannylation; AM281
Effects of cannabinoids on nitric oxide production by chondrocytes and proteoglycan degradation in cartilage
Keywords: AM281; 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-4-morpholinyl-1H-pyrazole-3-carboxamide; AM630; 6-iodo-2-methyl-1-[2-(4-morpholinyl) ethyl]-1H-indol-3-yl](4-methoxyphenyl)methanone; anandamide; N-(2-hydroxyethyl)-5Z,8Z,11Z,14Z-eicosatetraenamide
Inverse agonism and neutral antagonism at cannabinoid CB1 receptors
Keywords: CB1 receptors; Inverse agonism; SR141716A; AM251; AM281; LY320135; Neutral antagonists; Anandamide; Endocannabinoids; Autoprotection;