Keywords: فعالیت ضد سرطان; Schiff base; Co(II); Ni(II), Cu(II) and Zn(II) complexes; DFT; Anticancer activity; BSA binding
مقالات ISI فعالیت ضد سرطان (ترجمه نشده)
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Keywords: فعالیت ضد سرطان; Benzofuran; N-Aryl piperazine; Hybrid compounds; Anticancer activity
Keywords: فعالیت ضد سرطان; Indolizine; Diversity-oriented synthesis; Anticancer activity; β-Catenin; p53
Keywords: فعالیت ضد سرطان; Iodine; Rearrangement; Pyran; Pyridone; Anticancer activity
Keywords: فعالیت ضد سرطان; anticancer activity; cytotoxicity; joboksansam; Panax ginseng; survival enzyme
Keywords: فعالیت ضد سرطان; Bis-thiazole; Anticancer activity; DNA synthesis inhibitory activity; Acetylcholinesterase; Butyrylcholinesterase
Keywords: فعالیت ضد سرطان; Securinine; Semisynthesis; Heck reaction; Anticancer activity; Plasmatic stability
Keywords: فعالیت ضد سرطان; Synthesis; Hydroxypyrazolines; Characterization; Anticancer activity; Antioxidant activity;
Keywords: فعالیت ضد سرطان; Conjugation; Hybrid compound; Anticancer activity; Antibacterial activityVKLNFXHMPBWPKG-YHXOGZJDSA-N; XCBUYIHKXYRZMH-SASGCTTMSA-N
Spectroscopic, structural and anticancer activity studies of (â)-cytisine halogenated N-benzyl derivatives
Keywords: فعالیت ضد سرطان; (-)-Cytisine; N-benzylcytisine derivatives; MS and NMR spectra analysis; X-ray diffraction; Alkaloids; Natural products; Anticancer activity;
A novel silver (I) complex of α-keto phosphorus ylide: Synthesis, characterization, crystal structure, biomolecular interaction studies, molecular docking and in vitro cytotoxic evaluation
Keywords: فعالیت ضد سرطان; Phosphorus ylides; BSA binding; CT-DNA binding; Anticancer activity; Molecular docking;
3D porous Mn(II) coordination polymer with left-handed 41 helical chains as building subunits: Selective gas adsorption of CO2 over CH4 and anticancer activity evaluation
Keywords: فعالیت ضد سرطان; Mn(II) compound; Homochiral framework; Porous framework; Gas adsorption; Anticancer activity;
New TRAP1 and Hsp90 chaperone inhibitors with cationic components: Preliminary studies on mitochondrial targeting
Keywords: فعالیت ضد سرطان; TRAP1 inhibitors; Mitochondrial targeting; Anticancer activity; Lipophilic cations; Apoptosis;
Reprint of: Antiproliferative activity of the Antrodia camphorata secondary metabolite 4,7-dimethoxy-5-methylbenzo[d][1,3]dioxole and analogues
Keywords: فعالیت ضد سرطان; Antrodia camphorata; 4,7-dimethoxy-5-methylbenzo[d][1,3]dioxole; anticancer activity; NCI-60 screen;
Synthesis and anticancer activity of novel NHC-gold(I)-sugar complexes
Keywords: فعالیت ضد سرطان; Anticancer activity; Thiosugar; NHC-gold complex; Thioredoxin reductase;
Investigation of chemical reactivity of 2-alkoxy-1,4-naphthoquinones and their anticancer activity
Keywords: فعالیت ضد سرطان; 2-Alkoxy-5-hydroxy-1,4-naphthoquinone; Anticancer activity; Chemical reactivity;
Synthesis, spectral- and theoretical study, x-ray analysis, and antiproliferative activity of 4,5-dihydrobenzoferroceno[1,2-d][1,2,3]selenadiazole and its benzo-fused analogue
Keywords: فعالیت ضد سرطان; 1,2,3-Selenadiazole; Ferrocene; Anticancer activity; X-ray diffraction;
Crystal structures and anticancer activities of five novel pyrazolone-enamine transition metal complexes with 4-benzoyl-3-methyl-1-phenyl-2-pyrazolin-5-one
Keywords: فعالیت ضد سرطان; Pyrazolone-enamine; Complex; Crystal structure; Fluorescence; Anticancer activity;
Structure and anticancer activity of native and modified polysaccharides from brown alga Dictyota dichotoma
Keywords: فعالیت ضد سرطان; Dictyota; Fucoidan; Laminaran; Structure; Anticancer activity; γ-radiation;
Novel 5H-[1,2,4]oxadiazolo[4,5-a]pyrimidin-5-one derivatives as antibacterial and anticancer agents: Synthesis and biological evaluation
Keywords: فعالیت ضد سرطان; Oxadiazole; Pyrimidine; Antibacterial activity; Anticancer activity;
One-pot reaction of amide functionalized Re(I) based dinuclear metallacycles: Synthesis, characterization and evaluation for anticancer potential
Keywords: فعالیت ضد سرطان; Self-assembly; Flexible pyridyl ligand; Amide functionality; Metallacycle; Anticancer activity;
Design and synthesis of aminocoumarin derivatives as DPP-IV inhibitors and anticancer agents
Keywords: فعالیت ضد سرطان; 3-Aminocoumarin derivatives; 7-Amino-4-methylcoumarin derivatives; DPP-IV inhibition; Anticancer activity;
Chemical composition, antioxidant and anticancer activity of licorice from Fruska Gora locality
Keywords: فعالیت ضد سرطان; AAE; ascorbic acid equivalents; BHA; butylated hydroxyanisole; BHT; butylated hydroxytoluene; DPPH; 2,2 diphenyl-1-picrylhydrazyl; dw; dry weight; EDTA; ethylenediamine tetraacetic acid; ESI; electrospray ionization; FC reagent; Folin-Ciocalteu reagent; F
Novel (S)-1,3,4,12a-tetrahydropyrazino[2,1-c][1,4]benzodiazepine-6,12(2H,11H)-dione derivatives: Selective inhibition of MV-4-11 biphenotypic B myelomonocytic leukemia cells' growth is accompanied by reactive oxygen species overproduction and apoptosis
Keywords: فعالیت ضد سرطان; Tricyclic benzodiazepines; Selective inhibition; Biphenotypic B myelomonocytic leukemia; Reactive oxygen species overproduction; Apoptosis; Anticancer activity;
New inhibitors of matrix metalloproteinases 9 (MMP-9): Lignans from Selaginella moellendorffii
Keywords: فعالیت ضد سرطان; Lignans; Selaginella moellendorffii; Matrix metalloproteinase; Migration; Anticancer activity;
Phytoconstituents from Vernonia glaberrima Welw. Ex O. Hoffm. leaves and their cytotoxic activities on a panel of human cancer cell lines
Keywords: فعالیت ضد سرطان; Vernonia glaberrima; Anticancer activity; 5-Methylcoumarin-4-β-glucoside; Molecular docking; Carbonic anhydrase IX;
Anticancer activity profiling of parthenolide analogs generated via P450-mediated chemoenzymatic synthesis
Keywords: فعالیت ضد سرطان; PTL; parthenolide; AML; acute myelogenous leukemia; CSCs; cancer stem cells; DMAPT; dimethylamino-parthenolide; PTDH; phosphite dehydrogenase; NADPH; nicotinamide adenine dinucleotide phosphate (reduced); IPTG; β-d-1-thiogalactopyranoside; δ-ALA; δ-ami
Green synthesis and characterization of hexagonal shaped MgO nanoparticles using insulin plant (Costus pictus D. Don) leave extract and its antimicrobial as well as anticancer activity
Keywords: فعالیت ضد سرطان; Costus pictus D. Don; MgO nanoparticles; Green chemistry; Antimicrobial activity; Anticancer activity;
Pyridazine-based heteroleptic copper(II) complexes as potent anticancer drugs by inducing apoptosis and S-phase arrest in breast cancer cell
Keywords: فعالیت ضد سرطان; DFT analysis; Docking studies; Anticancer activity; Apoptosis; Cell cycle arrest;
Preparation and functional analysis of gossypols having two carbohydrate appendages with enaminooxy linkages
Keywords: فعالیت ضد سرطان; Gossypol; Glycocluster; Chemoselective coupling; Anticancer activity; Drug delivery system;
Synthesis and investigations into the anticancer and antibacterial activity studies of β-carboline chalcones and their bromide salts
Keywords: فعالیت ضد سرطان; β-Carboline chalcones; β-Carbolinium chalcone bromides; Anticancer activity; Apoptosis; Antibacterial activity;
Optimal conditions for cordycepin production in surface liquid-cultured Cordyceps militaris treated with porcine liver extracts for suppression of oral cancer
Keywords: فعالیت ضد سرطان; 7,12-dimethylbenz[a]anthracene; anticancer activity; cordycepin; Cordyceps militaris; mycelial extract; oral cancer; porcine liver extracts; water extract;
Diferrocenyl(areno)oxazoles, spiro(arenooxazole)cyclopropenes, quinolines and areno[1,4-]oxazines: Synthesis, characterization and study of their antitumor activity
Keywords: فعالیت ضد سرطان; Diferrocenyl-cyclopropenium; Diferrocenyl-arenooxazoles; Ferrocenyl-oxazines; Diferrocenyl-spirooxazole-cyclopropene; Diferrocenyl-quinolines; Anticancer activity;
Apigenin: A dietary flavonoid with diverse anticancer properties
Keywords: فعالیت ضد سرطان; Apigenin; Anticancer activity; Apoptosis; Cell cycle arrest; Signalling pathways;
Anticancer effects of some novel dichloroacetophenones through the inhibition of pyruvate dehydrogenase kinase 1
Keywords: فعالیت ضد سرطان; PDK; pyruvate dehydrogenase kinase; PDC; pyruvate dehydrogenase complex; MMP; mitochondrial membrane potential; ROS; reactive oxygen species; OXPHOS; oxidative phosphorylation; TCA; tricarboxylic acid; PDPs; pyruvate dehydrogenase phosphatases; DCA; dichl
KT2 and RT2 modified antimicrobial peptides derived from Crocodylus siamensis Leucrocin I show activity against human colon cancer HCT-116 cells
Keywords: فعالیت ضد سرطان; Anticancer activity; Apoptosis; Colorectal cancer; Crocodile; Peptide;
A novel pH-sensitive liposome to trigger delivery of afatinib to cancer cells: Impact on lung cancer therapy
Keywords: فعالیت ضد سرطان; Afatinib; pH-sensitive liposomes; In vitro release; Anticancer activity; Lung cancers;
Picoplatin-based complexes with the bioactive orotate and 5-fluoroorotate ligands: Synthesis, DFT calculations, structure, spectroscopic characterization and in vitro cytotoxicity
Keywords: فعالیت ضد سرطان; Platinum(II) complexes; Picoplatin; Orotates; Vibrational spectra; DFT calculations; Anticancer activity;
Synthesis, structures and anticancer potentials of platinum(II) saccharinate complexes of tertiary phosphines with phenyl and cyclohexyl groups targeting mitochondria and DNA
Keywords: فعالیت ضد سرطان; Platinum(II); Saccharinate; Tertiary phosphine; Anticancer activity; Apoptosis;
Novel benzotriazole N-acylarylhydrazone hybrids: Design, synthesis, anticancer activity, effects on cell cycle profile, caspase-3 mediated apoptosis and FAK inhibition
Keywords: فعالیت ضد سرطان; Benzotriazole; N- acylarylhydrazone; Fragment-based design; Synthesis; Anticancer activity; FAK; Caspase-3; Cell cycle arrest profile; Apoptosis;
Anticancer activity of novel steroidal 6-substituted 4-en-3-one D-seco dinitriles
Keywords: فعالیت ضد سرطان; Steroids; Dinitriles; Anticancer activity; Apoptosis; Hormone-independent breast cancer; Cervix adenocarcinoma;
Pt(IV) complexes conjugating with chalcone analogue as inhibitors of microtubule polymerization exhibited selective inhibition in human cancer cells
Keywords: فعالیت ضد سرطان; Anticancer activity; Pt(IV) complex; Tubulin polymerization; Apoptosis;
Novel ciprofloxacin hybrids using biology oriented drug synthesis (BIODS) approach: Anticancer activity, effects on cell cycle profile, caspase-3 mediated apoptosis, topoisomerase II inhibition, and antibacterial activity
Keywords: فعالیت ضد سرطان; Ciprofloxacin; Biology oriented drug synthesis (BIODS); Anticancer activity; Topoisomerase II; Cell cycle arrest profile; Caspase-3; Apoptosis; Antibacterial activity;
Synthesis, anticancer activity and docking studies of N-phenyl-2-(2-((4-phenyl piperazin-1-yl) methyl)-1H-benzo [d] imidazol-1-yl) acetamides
Keywords: فعالیت ضد سرطان; o-phenylene diamine; Phenyl piperazines; Acid-amide coupling; Anticancer activity; Docking;
Catalytic cyclometallation in steroid chemistry V: Synthesis of hybrid molecules based on steroid oximes and (5Z,9Z)-tetradeca-5,9-dienedioic acid as potential anticancer agents
Keywords: فعالیت ضد سرطان; Cross-cyclomagnesiation; Grignard reagents; Steroid oximes; 5Z,9Z-Dienoic acids; Anticancer activity;
In vitro DNA binding, antioxidant, antimicrobial and anticancer assessment of amino acid functionalized magnetic nanoparticles
Keywords: فعالیت ضد سرطان; Magnetic nanoparticles; Amino acids; Surface functionalization; DNA binding; DPPH scavenging assay; Antimicrobial; Anticancer activity;
Modification of native fucoidan from Fucus evanescens by recombinant fucoidanase from marine bacteria Formosa algae
Keywords: فعالیت ضد سرطان; Marine bacteria; Fucoidanase; Fucoidan from Fucus evanescens; Fucoidan depolymerization; Anticancer activity; Endo-fucoidanase;
Silica nanoparticles with Tb(III)-centered luminescence decorated by Ag0 as efficient cellular contrast agent with anticancer effect
Keywords: فعالیت ضد سرطان; Silica nanoparticles; Lanthanide; Silver nanoparticles; Cytotoxicity; Cellular uptake; Anticancer activity;
Synthesis, characterisation and cytotoxic properties of N-heterocyclic carbene silver(I) complexes
Keywords: فعالیت ضد سرطان; Anticancer activity; N-heterocyclic carbene; Silver complex; Sulfonated N-heterocyclic carbene;
3-Nitroacridine derivatives arrest cell cycle at G0/G1 phase and induce apoptosis in human breast cancer cells may act as DNA-target anticancer agents
Keywords: فعالیت ضد سرطان; Acridine derivatives; Synthesis; DNA binding; Anticancer activity; Structure-activity relationship (SAR); Apoptosis;