Crystal structure of the Eg5 - K858 complex and implications for structure-based design of thiadiazole-containing inhibitors
Keywords: داروهای ضد سرطان; 1,3,4-thiadiazole; K858 enantiomers; Eg5; Antimitotic drugs; Eg5-K858 complex; Rational drug design; KSP; Kinesin spindle protein; MT; Microtubule; PDB; Protein Data Bank; PK; Pyruvate kinase; LDH; Lactate dehydrogenase; ITC; Isothermal titration calorime