Keywords: حلالیت آب; Aqueous solubility; Disperse yellow 119; Reactivity; Substituents; Thermodynamic stability;
مقالات ISI حلالیت آب (ترجمه نشده)
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Keywords: حلالیت آب; Normal melting point; Aqueous solubility; Octanol/water partition coefficient; Group contribution method; Amino acids; AAE; average absolute error; ARE; average relative error [%]; ALogWs; adjustable parameter of Eq. (4); ALogkow; adjustable parameter of
Keywords: حلالیت آب; Anti-tuberculosis drug; Aqueous solubility; Drug stability; Mixed surfactant aggregates; Drug-surfactant interactions;
Keywords: حلالیت آب; Herbicide safeners; Aqueous solubility; Octanol-water partition coefficient; Adsorption; Oxidation; Environmental chemodynamics;
Quantification of apigenin trimethyl ether in rat plasma by liquid chromatography-tandem mass spectrometry: Application to a pre-clinical pharmacokinetic study
Keywords: حلالیت آب; Apigenin trimethyl ether; 5,7,4â²-Trimethoxyflavone; LC-MS/MS; Oral pharmacokinetics; Aqueous solubility;
Keywords: حلالیت آب; Halogenated benzenes; Vapor pressure; Hydration Gibbs energy; Aqueous solubility; Partition coefficient; Temperature of fusion;
Keywords: حلالیت آب; Aqueous solubility; Drug properties; General Solubility Equation (GSE); Hydrophobicity; Physicochemical properties;
Crystalline inclusion complexes formed between the drug diflunisal and block copolymers
Keywords: حلالیت آب; Pharmaceutical solid forms; Inclusion complexes; Drugs; Block copolymers; Thermal stability; Aqueous solubility; Dissolution profiles;
Keywords: حلالیت آب; Vascular adhesion protein-1; Diabetic nephropathy; Carbamimidoylcarbamate; Stability in plasma; Aqueous solubility;
Keywords: حلالیت آب; Carbazole sulfonamide derivatives; Synthesis; Antiproliferative activity; Aqueous solubility;
Keywords: حلالیت آب; Curcumin; Anticancer drug; Bioavailability; Aqueous solubility; Drug safety; Drug efficiency
Keywords: حلالیت آب; Mirtazapine salts; Molecular salt; Non-sublimating salts; Aqueous solubility; Single crystal structure;
Keywords: حلالیت آب; Diaryl amine; Kinesin spindle protein; Aqueous solubility
Keywords: حلالیت آب; SAR; structure-activity relationship; DPPH; 2,2-diphenyl-1-picrylhydrazyl; FRSA; free radical scavenging activity; Curcumin derivatives; Antitumor; Antioxidant activity; Aqueous solubility;
Keywords: حلالیت آب; QSPRs; Partial least-squares regression; Environmental contaminants; Aqueous solubility; Environmental mobility; Water quality;
Nano strategies for berberine delivery, a natural alkaloid of Berberis
Keywords: حلالیت آب; Aqueous solubility; Berberine; Bioavailability; Cancer therapy; Drug delivery; Nanocarriers;
Solution enhanced dispersion by supercritical fluids (SEDS): An approach in particle engineering to modify aqueous solubility of andrographolide from Andrographis paniculata extract
Keywords: حلالیت آب; SCFs; SEDS; sc-CO2; Andrographolide; Aqueous solubility; SEDS precipitated Andrographis paniculata powder;
An insight into effect of micelle-forming surfactants on aqueous solubilization and octanol/water partition coefficient of the drugs gemfibrozil and ibuprofen
Keywords: حلالیت آب; Ibuprofen; Gemfibrozil; Aqueous solubility; Partition coefficient; Micelle effect;
Preparation and characterization of dialdehyde β-cyclodextrin with broad-spectrum antibacterial activity
Keywords: حلالیت آب; Dialdehyde β-cyclodextrin; Periodate oxidation; Aqueous solubility; Antibacterial activity;
DMol3/COSMO-RS prediction of aqueous solubility and reactivity of selected Azo dyes: Effect of global orbital cut-off and COSMO segment variation
Keywords: حلالیت آب; Azo dye; Aqueous solubility; Reactivity; COSMO segment and global orbital cutoff;
Design, synthesis and biological evaluation of 7H-pyrrolo[2,3-d]pyrimidin-4-amine derivatives as selective Btk inhibitors with improved pharmacokinetic properties for the treatment of rheumatoid arthritis
Keywords: حلالیت آب; Btk; Inhibitor; Selectivity; Bioavailability; Aqueous solubility; Rheumatoid arthritis;
Structure-activity relationship studies on 1-(2-oxopropyl)indole-5-carboxylic acids acting as inhibitors of cytosolic phospholipase A2α: Effect of substituents at the indole 3-position on activity, solubility, and metabolic stability
Keywords: حلالیت آب; Cytosolic phospholipase A2α; Inhibitors; Indole derivatives; Metabolic stability; Ketone reduction; Glucuronidation; Aqueous solubility;
Novel hybrids of natural β-elemene bearing isopropanolamine moieties: Synthesis, enhanced anticancer profile, and improved aqueous solubility
Keywords: حلالیت آب; β-Elemene; Isopropanolamine; Dimer; Antitumor activity; Aqueous solubility;
Novel pyrazolo[1,5-a]pyridines with improved aqueous solubility as p110α-selective PI3 kinase inhibitors
Keywords: حلالیت آب; NKJYYWGDGSKPEW-LPYMAVHISA-N; AOXAAEQFLNMCLC-BUVRLJJBSA-N; WBWLQGYBHWVMKE-DHRITJCHSA-N; MXOGXVOOBVIVJW-YDZHTSKRSA-N; AZJHDRSPNKBZGF-MFKUBSTISA-N; QIGFDKVDGDNYSS-LGJNPRDNSA-N; QPTBMDPOZNSWEZ-WSDLNYQXSA-N; OCKIBXWFWFCVNS-YDZHTSKRSA-N; UZWYFVJGBGJHHK-OEAKJJBV
1-Heteroarylpropan-2-ones as inhibitors of fatty acid amide hydrolase: Studies on structure-activity relationships and metabolic stability
Keywords: حلالیت آب; Propan-2-one; Fatty acid amide hydrolase; Enzyme inhibition; Metabolic stability; Aqueous solubility;
Aqueous solubilities of five N-(diethylaminothiocarbonyl)benzimido derivatives at T = 298.15 K
Keywords: حلالیت آب; N-(diethylaminothiocarbonyl)benzimido derivatives; Aqueous solubility; COSMO-RS; Chemical space diagram
Aqueous solubility, vapor pressure and octanol-water partition coefficient of two phthalate isomers dibutyl phthalate and di-isobutyl phthalate contaminants of recycled food packages
Keywords: حلالیت آب; Aqueous solubility; Vapor pressures; Octanol-water partition coefficient; Dibutyl phthalate; Di-isobutyl phthalate;
Novel free fatty acid receptor 1 (GPR40) agonists based on 1,3,4-thiadiazole-2-carboxamide scaffold
Keywords: حلالیت آب; GPR40; Free fatty acid receptor 1; FFA1 agonists; Bioisosteric replacement; Total polar surface area; c Log P; Metabolic stability; Aqueous solubility
Synthesis and antitubercular evaluation of 4-carbonyl piperazine substituted 1,3-benzothiazin-4-one derivatives
Keywords: حلالیت آب; Tuberculosis; Benzothiazinones; Structure–activity relationships (SAR); Aqueous solubility
Discovery and SAR study of 2-(4-pyridylamino)thieno[3,2-d]pyrimidin-4(3H)-ones as soluble and highly potent PDE7 inhibitors
Keywords: حلالیت آب; Phosphodiesterase; Thienopyrimidinone; T-cell; Aqueous solubility
2-(Isopropylamino)thieno[3,2-d]pyrimidin-4(3H)-one derivatives as selective phosphodiesterase 7 inhibitors with potent in vivo efficacy
Keywords: حلالیت آب; Phosphodiesterase; Thienopyrimidinone; T-cell; Aqueous solubility; Anti-inflammation
β-cyclodextrin inclusion complexes containing Citrus sinensis (L.) Osbeck essential oil: An alternative to control Aedes aegypti larvae
Keywords: حلالیت آب; Citrus sinensis essential oil; β-cyclodextrin; Inclusion complexes; Aqueous solubility;
Parenterally administrable nano-micelles of 3,4-difluorobenzylidene curcumin for treating pancreatic cancer
Keywords: حلالیت آب; Pancreatic cancer; Nano-micelles; 3,4-Difluorobenzylidene curcumin; Styrene-maleic acid copolymer; Aqueous solubility; Nanoparticles;
Identification of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors with no evidence of CYP3A4 time-dependent inhibition and improved aqueous solubility
Keywords: حلالیت آب; Nicotinamide phosphoribosyltransferase; NAMPT; Cytochrome P450 time-dependent inhibition; CYP TDI; Aqueous solubility; Tumor metabolism
Externally predictive single-descriptor based QSPRs for physico-chemical properties of polychlorinated-naphthalenes: Exploring relationships of log SW, log KOA, and log KOW with electron-correlation
Keywords: حلالیت آب; QSPR; Persistent organic pollutants; Quantum chemical descriptors; Aqueous solubility; Partition-coefficients; Electron-correlation;
Synthesis and structure-activity relationships of 4-fluorophenyl-imidazole p38α MAPK, CK1δ and JAK2 kinase inhibitors
Keywords: حلالیت آب; VIZCCOPDAKHRKH-HNNXBMFYSA-N; JGMBDYVHJQPCAG-UHFFFAOYSA-N; PSOABNHNKXPGIE-UHFFFAOYSA-N; AWDXPJVBIPFUMF-UHFFFAOYSA-N; SCFAXAIGJNYTQW-UHFFFAOYSA-N; USGNAHFDLFPCMY-KFAMGINRSA-N; GXZIHMSRYZODGT-UHFFFAOYSA-N; KTAAEGBHFHOMIG-UHFFFAOYSA-L; WRUSSCKIDKSRLD-UHFFFAOY
Aqueous solubility (in the range between 298.15 and 338.15Â K), vapor pressures (in the range between 10â5 and 80Â Pa) and Henry's law constant of 1,2,3,4-dibenzanthracene and 1,2,5,6-dibenzanthracene
Keywords: حلالیت آب; Aqueous solubility; Vapor pressures; Partition coefficient air-water; Henry's constant; Polycyclic aromatic hydrocarbons;
solITC: A rapid method to determine solubility products and heats of solution of hydrophobic ionic liquids from in situ synthesis in isothermal titration calorimeter
Keywords: حلالیت آب; Electrolyte; Aqueous solubility; Solution thermodynamics; Calorimetry
Solubility prediction of indomethacin in PEG 400Â +Â water mixtures at various temperatures
Keywords: حلالیت آب; Indomethacin; Aqueous solubility; Mole fraction solubility; Polyethylene glycol 400; Thermodynamics; Modified Apelblat equation;
Solubilities of selected organic electronic materials in pressurized hot water and estimations of aqueous solubilities at 298.15Â K
Keywords: حلالیت آب; Aqueous solubility; OLED display; Hole transport material; Aromatic amine; Pressurized hot water;
Identification of 2,3-dihydro-1H-pyrrolo[3,4-c]pyridine-derived ureas as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT)
Keywords: حلالیت آب; Nicotinamide phosphoribosyltransferase; NAMPT; Aqueous solubility; X-ray crystal structure; Tumor metabolism;
Discovery of diarylurea P2Y1 antagonists with improved aqueous solubility
Keywords: حلالیت آب; P2Y1 antagonists; Diarylurea; Structure–activity relationship (SAR); Aqueous solubility; In vivo efficacy/bleeding model
Studies on aqueous solubility of 3,3′-diindolylmethane derivatives using cyclodextrin inclusion complexes
Keywords: حلالیت آب; Cyclodextrins; 3,3′-Diindolylmethane; Inclusion complex; Aqueous solubility; Supramolecular interaction
Solubility of fused silica in sub- and supercritical water: Estimation from a thermodynamic model
Keywords: حلالیت آب; Amorphous silica; Fused silica; Supercritical water; Near-critical water; Aqueous solubility; Thermodynamic model
Aqueous solubility: Simple predictive methods (in silico, in vitro and bio-relevant approaches)
Keywords: حلالیت آب; Aqueous solubility; Predicting solubility; In silico solubility; Solubility challenge; Kinetic solubility; Equilibrium solubility; Drug formulation
A novel, potent, and orally active VLA-4 antagonist with good aqueous solubility: trans-4-[1-[[2-(5-Fluoro-2-methylphenylamino)-7-fluoro-6-benzoxazolyl]acetyl]-(5S)-[methoxy(methyl)amino]methyl-(2S)-pyrrolidinylmethoxy]cyclohexanecarboxylic acid
Keywords: حلالیت آب; VLA-4; Eosinophil infiltration; Asthma; Aqueous solubility
Pyrazolopyridine inhibitors of B-RafV600E. Part 3: An increase in aqueous solubility via the disruption of crystal packing
Keywords: حلالیت آب; B-RafV600E; Aqueous solubility; Single-crystal X-ray; Crystal packing; Crystal lattice energy;
Synthesis and in vitro antitumor activity of asperphenamate derivatives as autophagy inducer
Keywords: حلالیت آب; Asperphenamate; Autophagy; Aqueous solubility; Structure–activity relationships; Inducer
Relevant parameters for assessing the environmental impact of some pyridinium, ammonium and pyrrolidinium based ionic liquids
Keywords: حلالیت آب; Aqueous solubility; Octanol/water partition coefficient; Relative lipophilicity; Infinite dilution diffusion coefficient; Ionic liquids; Functional group
Preparation and electrochemical behavior of water-soluble inclusion complex of ferrocene with β-cyclodextrin polymer
Keywords: حلالیت آب; Ferrocene; β-cyclodextrin polymer; Inclusion complex; Aqueous solubility; Electrochemistry;