Small molecule antagonists of the urokinase (uPA): urokinase receptor (uPAR) interaction with high reported potencies show only weak effects in cell-based competition assays employing the native uPAR ligand
Keywords: ATF, amino-terminal fragment of uPA; Boc, tert-butyloxycarbonyl; DCC, N,N′-dicyclohexylcarbodiimide; DIPEA, diisopropylethylamine; DMAP, 4-(N,N-dimethylamino)pyridine; EGF, epidermal growth factor; GPI, glycophosphatidylinositol; HBTU, O-benzotriazole-N,N