
Synthesis and in vitro evaluation of bile acid prodrugs of floxuridine to target the liver
Keywords: 5-FU, 5-fluorouracil; Boc2O, di-tert-butyl dicarbonate; CDCA, chenodeoxycholic acid; DCC, N,N′-dicyclohexylcarbodiimide; DCM, dichloromethane; DMAP, 4-dimethylaminopyridine; DMEM, Dulbecco’s modified Eagle medium; DMF, dimethyl formamide; DMSO, dimethyl s