
A PET study comparing receptor occupancy by five selective cannabinoid 1 receptor antagonists in non-human primates
Keywords: Cannabinoid 1 receptor (CB1R) antagonists; Obesity; Positron emission tomography (PET); Receptor occupancy; [11C]SD5024; Rimonabant; TaranabantAZ, AstraZeneca; AUC, area under the curve; BBB, blood–brain barrier; CB1R, cannabinoid 1 receptor; CD, candidat