Keywords: ADME; absorption/distribution/metabolism/excretion; BBB; blood-brain barrier; CD3OD; tetradeuteromethanol; CDCl3; deuterochloroform; CH2Cl2; dichloromethane; C log D; distribution coefficient; C log P; calculated partition coefficient; CNS; central
مقالات ISI (ترجمه نشده)
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Anti-malarial synergy of secondary metabolites from Morinda lucida Benth
Keywords: 1D- and 2D; NMR one dimension and two dimension nuclear magnetic resonance; CC; Column chromatography; CQ; Chloroquine; CDCl3; Deuterated chloroform; DMSO-d6; Deuterated dimethyl sulfoxide; CD3OD; Deuterated methanol; DCM; Dichloromethane; DMSO; Dimethyl
Discovery of selective ATP-competitive eIF4A3 inhibitors
Keywords: RNA helicase; Eukaryotic initiation factor 4A3 (eIF4A3) inhibitors; Exon junction complex (EJC); ATP-competitive type inhibitors; Isothermal titration calorimetry (ITC); Surface plasmon resonance (SPR); BRR2; bad response to refrigeration 2 (an ATP-depend
Acetophenone derivatives from a freshwater fungal isolate of recently described Lindgomyces madisonensis (G416)
Keywords: CHCl3; chloroform; CH3OH; methanol; CH3CN; acetonitrile; NMR; nuclear magnetic resonance; HRESIMS; high-resolution electrospray ionization mass spectrometry; HPLC; high-performance liquid chromatography; HMBC; heteronuclear multiple bond coherence; HSQC;
Antinociceptive, anti-inflammatory and antioxidant activities of aqueous extract from Remirea maritima (Cyperaceae)
Keywords: AAPH; 2,2â²-azobis-2-methyl-propanimidamide,dihydrochloride; ASA; Acetylsalicylic acid; CD3OD; Deuterated methanol; CNS; Central nervous system; EDTA; Ethylenediamine tetraacetic acid; ERMA; Aqueous extract of Remirea maritima; ESI; Electrospray ionizati
The 3,7-diazabicyclo[3.3.1]nonane scaffold for subtype selective nicotinic acetylcholine receptor ligands. Part 2: Carboxamide derivatives with different spacer motifs
Keywords: BBB; blood-brain barrier; CD3OD; tetradeuteromethanol; CDCl3; deuterochloroform; CH2Cl2; dichloromethane; CNS; central nervous system; D2O; deuterium oxide; DCC; N,Nâ²-dicyclohexylcarbodiimide; DMAP; 4-(dimethylamino)pyridine; DME; 1,2-dimethoxyethane;
Origin of Nanodroplet Formation Upon Dissolution of an Amorphous Solid Dispersion: A Mechanistic Isotope Scrambling Study
Keywords: nanodroplet origin; dissolution mechanism; amorphous solid dispersions; amorphous solubility; AAPS; amorphous-amorphous phase separation; ASD; amorphous solid dispersion; Camorph; amorphous solubility; CD3OD; deuterated methanol; DL; drug loading; D-NFD;
Investigations into the millimeter and submillimeter-wave spectrum of perdeuterated methanol, CD3OD, in its ground and first excited torsional states
Keywords: Methanol; CD3OD; Rotational spectroscopy; Torsion-rotational spectroscopy; Submillimeter wave spectroscopy; Hamiltonian; Interstellar molecule;
Cryogenically cooled probes-a leap in NMR technology
Keywords: NMR (Nuclear Magnetic Resonance); Cryogenic probe technology; Sensitivity; Signal-to-noise ratio; 1D; 1-dimensional; 2D; 2-dimensional; 3D; 3-dimensional; ASTM; American Society for Testing and Materials; BPTI; bovine pancreatic trypsine inhibitor; CDCl3;