
Structure–intrinsic activity relationship studies in the group of 1-imido/amido substituted 4-(4-arylpiperazin-1-yl)cyclohexane derivatives; new, potent 5-HT1A receptor agents with anxiolytic- like activity
Keywords: Arylpiperazines; 5-HT1A receptor ligands; α1-Adrenergic receptor ligands; Conformational constraints; Structure–intrinsic activity relationships studies; 5-HT1A receptor antagonists