Keywords: Tricyclic multiple(urea); Bn-protected; Crystal structure; DIBAL-H; Selective reduction;
مقالات ISI (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: ADME-Tox; absorption, distribution, metabolism, excretion, and toxicity; CYP2C19; hepatic cytochrome P450 2C19; CYP3A4; hepatic cytochrome P450 3A4; DSC; differential scanning calorimetry; DIBAL-H; diisobutylaluminium hydride; DME; 1,2-dimethoxyethane; DM
Keywords: Benzimidazoles; o-Phenylenediamine; Polyazacycloalkanes; Dihydrobenzimidazoles; DIBAL-H;
Keywords: Ac; acetyl; acac; acetylacetonate; 9-BBN; 9-borabicyclo[3.3.1]nonane; Bn; benzyl; Boc; tert-butyloxycarbonyl; BOM; benzyloxymethyl; brsm; based on recovered starting material; Bz; benzoyl; CAN; ammonium cerium(IV) nitrate; Cbz; benzyloxycarbonyl; CD; circ
Peramivir conjugates as orally available agents against influenza H275Y mutant
Keywords: Peramivir; Caffeic acid; Conjugate; Neuraminidase; Inhibitor; Influenza; Drug resistance; Ala; alanine; All; allyl; Asn; asparagine; Asp; aspartic acid; CDI; 1,1â²-carbonyl diimidazole; DIBAL-H; diisobutylaluminium hydride; DMAP; 4-dimethylaminopyridine;
Facile reductive oxy-Nazarov cyclization of 2-methoxy-2, 4-hexadienoates
Keywords: Reduction; Dibal-H; Oxy-Nazarov; 5-Hydroxyl cyclopentenone;
Discovery of novel somatostatin receptor subtype 5 (SSTR5) antagonists: Pharmacological studies and design to improve pharmacokinetic profiles and human Ether-a-go-go-related gene (hERG) inhibition
Keywords: Boc; tert-butoxycarbonyl; Pd(OAc)2; palladium acetate; PBu3; tributylphosphine; DIBAL-H; diisobutylaluminum hydride; S-phos; 2-dicyclohexylphosphino-2â²,6â²-dimethoxybiphenyl; Pd2(dba)3; tris(dibenzylideneacetone) dipalladium; NaH; sodium hydride; LiAlH
An update on the stereoselective synthesis of γ-amino acids
Keywords: ABO; 2,7,8-trioxabicyclo[3.2.1]octane; Ac; acetyl; ACPECA; 4-aminocyclopent-2-ene-1-carboxylic acid; AHPPA; 4-amino-3-hydroxy-5-phenylpentanoic acid; AMCP; 2-(aminomethyl)-cyclopentanecarboxylic acid; APCH; 2-(1-aminopropyl)cyclohexanecarboxylic acid; APT
Stereoselective synthesis of 3-hydroxy-3-methylglutaryl-coenzyme A reductase inhibitors
Keywords: HMG-CoA reductase inhibitors; Statins; Chiral β-hydroxy-δ-lactone; Chiral 3,5-syn-diol acid; Asymmetric synthesis; Ac; acetyl; Ar; aryl; Bn; benzyl; Bz; benzoyl; n-Bu; butyl; t-Bu; tert-butyl; CDI; 1,1â²-carbonyldiimidazole; BINOL; 1,1â²-bi-2-naphthol
Aromatic abietane diterpenoids: total syntheses and synthetic studies
Keywords: Diterpene; Abietane; Total synthesis; Semisynthesis; AcCl; acetyl chloride; Ac2O; acetic anhydride; BnCl; benzyl chloride; n-BuLi; n-butyllithium; DCC; N,Nâ²-dicyclohexylcarbodiimide; DCM; dichloromethane; DDQ; 2,3-dichloro-5,6-dicyano-1,4-benzoquinone;
An update on the stereoselective synthesis of α-aminophosphonic acids and derivatives
Keywords: α-Aminophosphonic acids; α-Aminophosphonates; Stereoselective synthesis; Three-component reaction; ABSA; 4-acetamidobenzenesulfonyl azide; Abu; aminobutyric acid; Ac; acetyl; ACE; angiotensin-converting enzyme; Ala; alanine; Ar; aryl; BINAP; 2,2â²-bis(
Total synthesis of glycomaurrol and eustifoline-C by DIBAL-H promoted reductive ring opening of pyrano[2,3-c]carbazoles
Keywords: Carbazole; Pyranocarbazole; DIBAL-H; Reduction; Ring opening;
Chemical synthesis of tetracyclic terpenes and evaluation of antagonistic activity on endothelin-A receptors and voltage-gated calcium channels
Keywords: 2D NOESY; two-dimensional nuclear Overhauser effect spectroscopy; Dibal-H; diisobutylaluminum hydride; DRG; dorsal root ganglion; ee; enantiomeric excess; ET-1; endothelin-1; ETA; endothelin A receptors; EGTA; ethylene glycol tetraacetic acid; EC50; media
Tetrahedron report number 1022Recent developments of the Stille reaction as a revolutionized method in total synthesis
Keywords: Stille coupling; Natural product; Palladium; Total synthesis; Cross coupling; CuTC; copper(I) thiophene-2-carboxylate; DIBAL-H; diisobutylaluminum hydride; DIPEA; diisopropylethylamine; DMF; dimethylformamide; MOM; methoxymethyl; NMP; N-methylpyrrolidone;
Synthesis of four mono-functionalized α-cyclodextrin derivatives for further confirming DIBAL-H-promoted bis-de-O-methylation mechanism
Keywords: α-Cyclodextrin; DIBAL-H; Mechanism; Synthesis;
Synthesis and evaluation of heteroaryl substituted diazaspirocycles as scaffolds to probe the ATP-binding site of protein kinases
Keywords: AGC; protein kinases A G and C; ATP; adenosine triphosphate; 9-BBN; 9-borabicyclo[3.1.1.]nonane Boc tert-butyloxycarbonyl; CAMK; calcium/calmodulin-dependent kinases; Cbz; benzyloxycarbonyl; DFG; aspartate-phenylalanine-glycine sequence; DIBAL-H; diis
Synthesis of two mono-deoxy β-cyclodextrin derivatives as useful tools for confirming DIBAL-H promoted bis-de-O-methylation mechanism
Keywords: Cyclodextrin (CD); DIBAL-H; Deoxy; Synthesis; Mechanism
Facile preparation of two tetrols from permethylated α-cyclodextrin and unambiguous NMR analysis
Keywords: Cyclodextrin; Tetrol; DIBAL-H; De-O-methylation; Regioselectivity;
Preparation of 1-C-glycosyl aldehydes by reductive hydrolysis
Keywords: Glycosyl cyanides; 1-C-Glycosyl aldehydes; DIBAL-H; β-Elimination; 1,3-Imidazolidine derivative;
Design and synthesis of 3-pyridylacetamide derivatives as dipeptidyl peptidase IV (DPP-4) inhibitors targeting a bidentate interaction with Arg125
Keywords: DPP-4; Dipeptidyl peptidase IV; GLP-1; Glucagon-like peptide 1; SAR; Structure-activity relationship; AcOH; Acetic acid; DIBAL-H; Diisobutylaluminum hydride; Boc; tert-Butoxy carbonyl; TMSCN; Trimethylsilyl cyanide; TBAF; Tetrabutylammonium fluoride; mC
Tetrahedron report number 878Synthesis of unusually strained spiroheterocyclic ring systems and their exploits in synthesis
Keywords: acac; acetylacetonate; Bz; benzoyl; cod; 1,5-cyclooctadiene; DBU; 1,8-diazabicyclo[5.4.0]undec-7-ene; DET; diethyl tartrate; DIBAL-H; diisobutylaluminum hydride; DMDO; dimethyl dioxirane; DMSO; dimethylsulfoxide; EtOAc; ethyl acetate; EWG; electron-withdr
Regioselective ring opening of benzylidene acetal protecting group(s) of hexopyranoside derivatives by DIBAL-H
Keywords: Deprotection; Benzylidene acetal; DIBAL-H; Solvent effect; Reduction
Synthesis of (Z)-alkene-containing cis-proline dipeptide mimetics using samarium(II) diiodide (SmI2)-mediated reductive alkylation reaction
Keywords: Samarium diiodide; Reductive alkylation reaction; Dipeptide mimetic; Proline; Ns; 2-nitrobenzenesulfonyl; Bn; benzyl; TBS; tert-butyldimethylsilyl; DIBAL-H; diisobutylaluminumhydride; Tf2NPh; N-phenylbis(trifluoromethanesulfonimide); TBAF; tetrabutylammon
Tetrahedron report number 821Total syntheses and synthetic studies of spongiane diterpenes
Keywords: Diterpenes; Spongiane; Marine natural products; Synthesis; AcCl; acetyl chloride; Ac2O; acetic anhydride; AIBN; azobisisobutyronitrile; BuLi; buthyllithium; DIBAL-H; diisobutylaluminum hydride; DHP; dihydropyrane; DMAD; dimethyl acetylenedicarboxylate; DM
Advances in the Baylis-Hillman reaction-assisted synthesis of cyclic frameworks
Keywords: Baylis-Hillman reaction; Cyclic compounds; Heterocycles; Nucleophilic substitution; Ac; acetyl; AIBN; 2,20-azobisisobutyronitrile; Aq; aqueous; Ar; aryl; 9BBN; 9-borabicyclo[3.3.1]nonane; BINAP; 2,20-bis(diphenylphosphanyl)-1,10-binaphthyl; BF3·Et2O; b
Application of hydrolytic kinetic resolution (HKR) in the synthesis of bioactive compounds
Keywords: Hydrolytic kinetic resolution; Terminal epoxides; Bis-epoxides; meso-Epoxides; Natural products; Synthesis; Biological activity; Ac; acetyl; AD; asymmetric dihydroxylation; AE; asymmetric epoxidation; Bn; benzyl; NBS; N-bromosuccinimide; Boc; t-butoxycarb
Recent advances in the chemistry of macroline, sarpagine and ajmaline-related indole alkaloids
Keywords: Ac; acetyl; AD; asymmetric dihydroxylation; AIBN; 2,2â²-azobisisobutyronitrile; Ar; aryl; 9-BBN; 9-borabicyclo[3.3.1]nonane; Bn; benzyl; Boc; tert-butoxycarbonyl; Bu; butyl; Bz; benzoyl; cat; catalytic; CBz; benzyloxycarbonyl; CLB; chlorobenzoyl; Cy; cyc
Naphtho[2,3-c]furan-4,9-diones and related compounds: theoretically interesting and bioactive natural and synthetic products
Keywords: Naphtho[2,3-c]furan-4,9-diones; Naphtho[2,3-c]furan-4(9H)-ones; Naphtho[2,3-c]furan; Isofuranonaphthoquinones; Ac; acetyl; AIBN; 2â²-azobis(isobutyronitrile); Ar; aryl; Bn; benzyl; BOM; benzyloxymethyl; But; tert-butyl; CSA; camphor-10-sulfonic acid; DBU