Keywords: DNA گیراز; Quinolone; Free radical process; DNA gyrase; Antibacterial; Electron microscope;
مقالات ISI DNA گیراز (ترجمه نشده)
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Keywords: DNA گیراز; Quinoline; Isatoic anhydride; Anthranilamide Schiff bases; Antitubercular activity; DNA gyrase;
Keywords: DNA گیراز; Chemical space; Middle space; Bacterial permeability; Fluoroquinolone; DNA gyrase; Antibacterial; Antibiotic; Dimer
Keywords: DNA گیراز; Fluoroquinolone; Flavonoid; Hybrid; DNA gyrase; Efflux pump; Inhibitor
Regulation of the gyr operon of Mycobacterium tuberculosis by overlapping promoters, DNA topology, and reiterative transcription
Keywords: DNA گیراز; Mycobacterium; DNA gyrase; Relaxation stimulated transcription; Overlapping promoters; Topology; Reiterative transcription; RST; Relaxation stimulated transcription; ITR; Initial transcribed region; RT; Reiterative transcription;
A novel synthesis of 2-arylbenzimidazoles in molecular sieves-MeOH system and their antitubercular activity
Keywords: DNA گیراز; Arylbenzimidazoles; Chemoselectivity; Molecular sieves; Antitubercular; DNA gyrase; Acute oral toxicity;
Design, synthesis and antibacterial properties of pyrimido[4,5-b]indol-8-amine inhibitors of DNA gyrase
Keywords: DNA گیراز; ESKAPE pathogens; Anti-infectives; Topoisomerases; DNA gyrase; Pyrimido[4,5-b]indol-8-amine;
Design, synthesis, and evaluation of novel N-1 fluoroquinolone derivatives: Probing for binding contact with the active site tyrosine of gyrase
Keywords: DNA گیراز; Bacterial resistance; Fluoroquinolone; DNA gyrase; Topoisomerase;
Drug efficacy of novel 3-O-methoxy-4-halo disubstituted 5,7-dimethoxy chromans; evaluated via DNA gyrase inhibition, bacterial cell wall lesion and antibacterial prospective
Keywords: DNA گیراز; Antibacterial; Disubstituted-5,7-dimethoxy chromans; DNA gyrase; Lipinski's filter; Molecular docking;
DNA gyrase inhibitors: Progress and synthesis of potent compounds as antibacterial agents
Keywords: DNA گیراز; DNA gyrase; DNA gyrase inhibitors; Quinolones; Spiropyrimidinetriones; Coumarins; Chebulinic acid;
Synthesis, structural and antimicrobial studies of type II topoisomerase-targeted copper(II) complexes of 1,3-disubstituted thiourea ligands
Keywords: DNA گیراز; Copper complexes; Thiourea; DNA gyrase; FTIR; Docking;
Design and synthesis of novel 1H-tetrazol-5-amine based potent antimicrobial agents: DNA topoisomerase IV and gyrase affinity evaluation supported by molecular docking studies
Keywords: DNA گیراز; 1H-tetrazol-5-amine; Antimicrobial activity; Topoisomerase type IV; DNA gyrase; Cytotoxicity; Molecular docking;
In vitro antiplasmodial efficacy of synthetic coumarin-triazole analogs
Keywords: DNA گیراز; Coumarin; Plasmodium falciparum; Antiplasmodial; DNA gyrase;
New N-phenylpyrrolamide DNA gyrase B inhibitors: Optimization of efficacy and antibacterial activity
Keywords: DNA گیراز; Antibacterial; DNA gyrase; GyrB; Inhibitor; N-phenylpyrrolamide; ParE; Topoisomerase IV; ATCC; American type culture collection; ATR; attenuated total reflectance; CDI; 1,1â²-carbonyldiimidazole; CFU; colony-forming unit; CLSI; Clinical and Laboratory St
PLGA nanoformulation of sparfloxacin enhanced antibacterial activity with photoprotective potential under ambient UV-R exposure
Keywords: DNA گیراز; Sparfloxacin; DNA gyrase; DNA damage; Apoptosis; Photostability;
In vitro and in vivo evaluation of fluoroquinolone resistance associated with DNA gyrase mutations in Francisella tularensis, including in tularaemia patients with treatment failure
Keywords: DNA گیراز; Francisella tularensis; Tularaemia; Fluoroquinolones; Antibiotic resistance; DNA gyrase; Treatment failure; FQ; fluoroquinolone; QRDR; quinolone-resistance determining region;
3,4-Dihydropyrimidinone-coumarin analogues as a new class of selective agent against S. aureus: Synthesis, biological evaluation and molecular modelling study
Keywords: DNA گیراز; Coumarin; Matrix metalloproteinases; S. aureus; DNA gyrase; Gelatin zymography;
New 1,4-dihydro[1,8]naphthyridine derivatives as DNA gyrase inhibitors
Keywords: DNA گیراز; Fluoroquinolones; DNA gyrase; Antibacterial activity; ATP luminescence; NIH/3T3; Ames MPF;
Design, synthesis and biological evaluation of 4,5-dibromo-N-(thiazol-2-yl)-1H-pyrrole-2-carboxamide derivatives as novel DNA gyrase inhibitors
Keywords: DNA گیراز; Antibacterial; DNA gyrase; Docking; Inhibitor; Thiazole;
Fragment-based discovery of DNA gyrase inhibitors targeting the ATPase subunit of GyrB
Keywords: DNA گیراز; DNA gyrase; GyrB; Fragment-based screening; NMR; Structure-based design
Identification of 5,6-dihydroimidazo[2,1-b]thiazoles as a new class of antimicrobial agents
Keywords: DNA گیراز; Heterocyclic; Antimicrobial; MRSA; DNA gyrase; Imidazothiazole;
Development of acridine derivatives as selective Mycobacterium tuberculosis DNA gyrase inhibitors
Keywords: DNA گیراز; Tuberculosis; DNA gyrase; Acridine derivatives
Discovery and structure-activity relationships of a novel isothiazolone class of bacterial type II topoisomerase inhibitors
Keywords: DNA گیراز; ESKAPE pathogens; Anti-infectives; Topoisomerases; DNA gyrase; Isothiazolone;
Replacement of cardiotoxic aminopiperidine linker with piperazine moiety reduces cardiotoxicity? Mycobacterium tuberculosis novel bacterial topoisomerase inhibitors
Keywords: DNA گیراز; DNA gyrase; Topoisomerase; Tuberculosis; 1,5-Naphthyridin-2(1H)-one; zERG toxicity
Engineering another class of anti-tubercular lead: Hit to lead optimization of an intriguing class of gyrase ATPase inhibitors
Keywords: DNA گیراز; Medium throughput virtual screening; Mycobacterium tuberculosis; DNA gyrase; Differential scanning fluorimetry
Proposal of Helicobacter canicola sp. nov., previously identified as Helicobacter cinaedi, isolated from canines
Keywords: DNA گیراز; Canine; DNA-DNA hybridization; In silico DNA similarity analysis; Average nucleotide identity (ANI); DNA gyrase; Heat shock protein; 16S rRNA; 23S rRNA;
Fluoroquinolones stimulate the DNA cleavage activity of topoisomerase IV by promoting the binding of Mg2Â + to the second metal binding site
Keywords: DNA گیراز; Divalent metal ion; DNA gyrase; Fluoroquinolone; Quinazolinedione; Topoisomerase IV;
Emergence of fluoroquinolone-resistant Propionibacterium acnes caused by amino acid substitutions of DNA gyrase but not DNA topoisomerase IV
Keywords: DNA گیراز; Propionibacterium acnes; Fluoroquinolone resistance; DNA gyrase; Amino acid substitution;
Ambient UV-B exposure reduces the binding of ofloxacin with bacterial DNA gyrase and induces DNA damage mediated apoptosis
Keywords: DNA گیراز; OFLX; UV-B; DNA gyrase; DNA damage; Apoptosis;
Identification of a novel mutation at the primary dimer interface of GyrA conferring fluoroquinolone resistance in Clostridium difficile
Keywords: DNA گیراز; Clostridium difficile; DNA gyrase; Fluoroquinolone resistance; Genomics
Chemical conjugation of 2-hexadecynoic acid to C5-curcumin enhances its antibacterial activity against multi-drug resistant bacteria
Keywords: DNA گیراز; C5-curcuminoids synthesis; Antibacterial agents; MRSA; Antagonism; DNA gyrase;
Characterization of Campylobacter jejuni DNA gyrase as the target of quinolones
Keywords: DNA گیراز; DNA gyrase; Quinolones; Campylobacter jejuni;
Characterisation of the DNA gyrase from the thermophilic eubacterium Thermus thermophilus
Keywords: DNA گیراز; DNA gyrase; Drug screening; Gyrase-DNA ternary complex; Structure-directed drug discovery;
Benzothiazinone-piperazine derivatives as efficient Mycobacterium tuberculosis DNA gyrase inhibitors
Keywords: DNA گیراز; Tuberculosis; DNA gyrase; Supercoiling; Minimum inhibitory concentration
Design and synthesis of novel quinoline–aminopiperidine hybrid analogues as Mycobacterium tuberculosis DNA gyraseB inhibitors
Keywords: DNA گیراز; Tuberculosis; DNA gyrase; Quinoline; Aminopiperidine
Development of 2-amino-5-phenylthiophene-3-carboxamide derivatives as novel inhibitors of Mycobacterium tuberculosis DNA GyrB domain
Keywords: DNA گیراز; Tuberculosis; DNA gyrase; Antimycobacterial; Cytotoxicity;
Comparison of rpoB gene sequencing, 16S rRNA gene sequencing, gyrB multiplex PCR, and the VITEK2 system for identification of Acinetobacter clinical isolates
Keywords: DNA گیراز; Sequence analysis; DNA; RNA; Ribosomal; 16S; Acinetobacter; rpoB; DNA Gyrase; Genes; Identification; PCR
Pyridine-3-carboxamide-6-yl-ureas as novel inhibitors of bacterial DNA gyrase: Structure based design, synthesis, SAR and antimicrobial activity
Keywords: DNA گیراز; Bacterial resistance; DNA gyrase; Pyridine-3-carboxamide; Molecular modelling
Discovery and in vivo evaluation of alcohol-containing benzothiazoles as potent dual-targeting bacterial DNA supercoiling inhibitors
Keywords: DNA گیراز; DNA gyrase; Topoisomerase; Antibacterial; Synthesis; In vivo; Dual-targeting;
Novel 3-arylfuran-2(5H)-one-fluoroquinolone hybrid: Design, synthesis and evaluation as antibacterial agent
Keywords: DNA گیراز; 3-Arylfuran-2(5H)-one; Fluoroquinolone; Hybrid; Multi-target; TyrRS; DNA gyrase
Development of novel N-linked aminopiperidine-based mycobacterial DNA gyrase B inhibitors: Scaffold hopping from known antibacterial leads
Keywords: DNA گیراز; Tuberculosis; DNA gyrase; GyrB domain; Aminopiperidine
Thiazolopyridone ureas as DNA gyrase B inhibitors: Optimization of antitubercular activity and efficacy
Keywords: DNA گیراز; Tuberculosis; DNA gyrase; Thiazolopyridone ureas; GyrB;
Extending the N-linked aminopiperidine class to the mycobacterial gyrase domain: Pharmacophore mapping from known antibacterial leads
Keywords: DNA گیراز; DNA gyrase; Tuberculosis; Aminopiperidine; Antimycobacterial; Supercoiling; Cytotoxicity
An efficient synthesis and biological screening of benzofuran and benzo[d]isothiazole derivatives for Mycobacterium tuberculosis DNA GyrB inhibition
Keywords: DNA گیراز; Tuberculosis; Antitubercular; DNA gyrase; Benzofuran; Benzo[d]isothiazole; Cytotoxicity;
Flavone-based analogues inspired by the natural product simocyclinone D8 as DNA gyrase inhibitors
Keywords: DNA گیراز; Simocyclinone D8; DNA gyrase; Antibiotics; Natural product; Flavone; Quercetin;
Design, synthesis and biological evaluation of α-substituted isonipecotic acid benzothiazole analogues as potent bacterial type II topoisomerase inhibitors
Keywords: DNA گیراز; DNA gyrase; Topoisomerase; Antibacterial;
In vitro anti-Helicobacter pylori activity of a flavonoid rich extract of Glycyrrhiza glabra and its probable mechanisms of action
Keywords: DNA گیراز; PPI; Proton pump inhibitor; DGL; Deglycyrrhizinated licorice; MAG; Monoammonium glycyrrhizinate; DMSO; Dimethyl sulfoxide; FBS; Fetal bovine serum; MIC; Minimum inhibitory concentration; DHFR; Dihydrofolate reductase; PBS; Phosphate buffered saline; FITC;
Novel quinoline derivatives as inhibitors of bacterial DNA gyrase and topoisomerase IV
Keywords: DNA گیراز; Antibacterial; DNA gyrase; Dual-targeting; Inhibitor; Topoisomerase IV;
Novel DNA gyrase inhibitors: Microbiological characterisation of pyrrolamides
Keywords: DNA گیراز; Antibacterial; Pyrrolamide; DNA gyrase;
Thiazole-aminopiperidine hybrid analogues: Design and synthesis of novel Mycobacterium tuberculosis GyrB inhibitors
Keywords: DNA گیراز; Tuberculosis; DNA gyrase; GyrB subunit; Thiazole; Amino piperidine;