Keywords: مشابه دارو; Algal drugs; Enzyme inhibitors; Dementia; Diabetes; Drug likeness; Inflammation; Structure activity relationship
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Molecular docking study and anticonvulsant activity of synthesized 4-((4,6-dimethyl-6H-1,3-thiazin-2-yl)phenylsulfonyl)urea/thiourea derivatives
Keywords: مشابه دارو; Anticonvulsant; Sulfonylurea; Molecular docking; Neurotoxicity; Rotarod; Drug likeness;
A systems pharmacology perspective to decipher the mechanism of action of Parangichakkai chooranam, a Siddha formulation for the treatment of psoriasis
Keywords: مشابه دارو; Psoriasis; Parangichakkai chooranam; Siddha; Systems pharmacology; Drug likeness; Pathways;
Quinoline-azetidinone hybrids: Synthesis and in vitro antiproliferation activity against Hep G2 and Hep 3B human cell lines
Keywords: مشابه دارو; Quinoline; Azetidinone; Antiproliferation; Drug likeness;
The molecular shape and the field similarities as criteria to interpret SAR studies for fragment-based design of platinum(IV) anticancer agents. Correlation of physicochemical properties with cytotoxicity
Keywords: مشابه دارو; Platinum-based drugs; Anticancer agents; Cytotoxicity; Structure-activity relationship; Shape and field similarity; XED field; Drug likeness; Structure-related molecular properties; Stereo-electronic effects;
Synthesis of novel pyrazole–thiadiazole hybrid as potential potent and selective cyclooxygenase-2 (COX-2) inhibitors
Keywords: مشابه دارو; Pyrazoles; Thiadiazole; COX-1 and COX-2; Cytotoxicity; Docking; Drug likeness
Softening the Rule of Five-where to draw the line?
Keywords: مشابه دارو; NGVDGCNFYWLIFO-UHFFFAOYSA-N; Lipinski Rules; Soft Rule of Five; Utility functions; Analytic hierarchy process; Drug likeness; Decision theory; Molecular properties;
A comparison of the chemical properties of drugs and FEMA/FDA notified GRAS chemical compounds used in the food industry
Keywords: مشابه دارو; GRAS; Drug likeness; QSAR; Molecular properties