Keywords: حمل و نقل مواد مخدر; 11βHSD; 11β-Hydroxysteroid dehydrogenase; ABC; ATP-binding cassette; AhR; aryl hydrocarbon receptor; ARNT; aryl hydrocarbon receptor nuclear translocator; BCRP; breast cancer resistance protein; CAR; constitutive androstane receptor; CYP; cytochrome P45
مقالات ISI حمل و نقل مواد مخدر (ترجمه نشده)
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Keywords: حمل و نقل مواد مخدر; Membrane transporter; Drug transporter; Posttranslational modification; Regulation;
Keywords: حمل و نقل مواد مخدر; Mebendazole; Inhibition; Drug transporter; Gastric cancer cells;
Keywords: حمل و نقل مواد مخدر; Intracellular drug concentration; Pharmacodynamics; OCT; MATE; PMAT; Drug transporter; ABC; ATP-binding cassette; ACC; acetyl-CoA carboxylase; AMP; adenosine monophosphate; AMPK; AMP-activated protein kinase; AUC; area under the concentration time curve;
Keywords: حمل و نقل مواد مخدر; Tyrosine kinase inhibitors; Drug transporter; Drug interaction; Therapeutic drug monitoring; Skin disorders; ADR; Adverse drug reaction; AUC; Area under the curve; BBB; Blood-brain barrier; BCRP/ABCG2; Breast cancer resistance protein; CNS; Central nerv
Keywords: حمل و نقل مواد مخدر; chronic kidney disease; drug excretion; drug metabolism; drug transporter; uremia;
Keywords: حمل و نقل مواد مخدر; Rilpivirine; Drug interaction; CYP; Drug transporter; PXR;
Inhibition of organic cation transporter (OCT) activities by carcinogenic heterocyclic aromatic amines
Keywords: حمل و نقل مواد مخدر; Drug transporter; Toxicokinetics; Organic cation transporter; Heterocyclic amines; Toxicity;
Inhibition of organic anion transporter (OAT) activity by cigarette smoke condensate
Keywords: حمل و نقل مواد مخدر; Drug transporter; Cigarette smoke; Pharmacokinetics; Organic anion transporter; Heterocyclic amines;
Effects of frequently used pharmaceutical excipients on the organic cation transporters 1-3 and peptide transporters 1/2 stably expressed in MDCKII cells
Keywords: حمل و نقل مواد مخدر; Pharmaceutical excipients; Solubilizing agents; Drug transporter; Uptake transport; Organic cation transporter (OCT); Peptide transporter (PEPT); Polyethylene glycol (PEG); Hydroxypropyl-β-cyclodextrin; Solutol HS 15 (macrogol 15 hydroxystearate, polyoxy
Physical and biological characteristics of multi drug resistance (MDR): An integral approach considering pH and drug resistance in cancer
Keywords: حمل و نقل مواد مخدر; Pharmacokinetic; Drug transporter; Membrane biophysics; Warburg effect;
Effects of natural nuclear factor-kappa B inhibitors on anticancer drug efflux transporter human P-glycoprotein
Keywords: حمل و نقل مواد مخدر; P-glycoprotein; Drug transporter; Anticancer drug; NF-κB; Phytochemical
Association of polymorphisms in drug transporter genes (SLCO1B1 and SLC10A1) and anti-tuberculosis drug-induced hepatotoxicity in a Chinese cohort
Keywords: حمل و نقل مواد مخدر; Drug transporter; Anti-tuberculosis drug; Hepatotoxicity;
Desmethyl bosentan displays a similar in vitro interaction profile as bosentan
Keywords: حمل و نقل مواد مخدر; Desmethyl bosentan; Hydroxy bosentan; Hydroxy desmethyl bosentan; 4-Hydroxymethyl ambrisentan; Drug transporter; Drug metabolising enzymes;
Modeling approach for multiple transporters-mediated drug–drug interactions in sandwich-cultured human hepatocytes: Effect of cyclosporin A on hepatic disposition of mycophenolic acid phenyl-glucuronide
Keywords: حمل و نقل مواد مخدر; Mathematical modeling; Sandwich-cultured human hepatocytes; Hepatic disposition; Drug transporter; Drug–drug interaction
Polarized location of SLC and ABC drug transporters in monolayer-cultured human hepatocytes
Keywords: حمل و نقل مواد مخدر; Canalicular secretion; Drug transporter; Hepatocytes; Polarization; Primary culture;
Age-related testicular toxicity of mGluR5 negative allosteric modulators appears to be unrelated to testis drug transporter maturity
Keywords: حمل و نقل مواد مخدر; Testis; mGluR5; Immaturity; Drug transporter; Rat;
Protein kinase C-dependent regulation of human hepatic drug transporter expression
Keywords: حمل و نقل مواد مخدر; Drug transporter; Hepatocyte; Protein kinase C; Phorbol ester; Regulation;
A Single Nucleotide Polymorphism in SLC7A5 Is Associated with Gastrointestinal Toxicity after High-Dose Melphalan and Autologous Stem Cell Transplantation for Multiple Myeloma
Keywords: حمل و نقل مواد مخدر; Pharmacogenetics; Multiple myeloma; High-dose melphalan; Autologous hematopoietic stem cell transplantation; Gastrointestinal toxicity; Drug transporter
Interaction profile of macitentan, a new non-selective endothelin-1 receptor antagonist, in vitro
Keywords: حمل و نقل مواد مخدر; Macitentan; Pulmonary arterial hypertension; Drug transporter; Drug metabolising enzymes; Induction;
The SLC22 family with transporters of organic cations, anions and zwitterions
Keywords: حمل و نقل مواد مخدر; Drug transporter; Cation transporter; Anion transporter; Urate transporter; SLC22; Drug excretion;
Role of organic cation transporter OCT2 and multidrug and toxin extrusion proteins MATE1 and MATE2-K for transport and drug interactions of the antiviral lamivudine
Keywords: حمل و نقل مواد مخدر; Lamivudine; MATE; OCT2; Trimethoprim; Drug transporter
Estrogen receptor-α mediates human multidrug resistance associated protein 3 induction by 17α-ethynylestradiol. Role of activator protein-1
Keywords: حمل و نقل مواد مخدر; Drug transporter; AP-1; Estrogen; Multidrug resistance; Nuclear receptor; c-JUN.
Polymorphisms in drug transporter genes (ABCB1, SLCO1B1 and ABCC2) and hepatitis induced by antituberculosis drugs
Keywords: حمل و نقل مواد مخدر; Drug transporter; Antituberculosis drug; Hepatitis
Interaction of the antiviral drug telaprevir with renal and hepatic drug transporters
Keywords: حمل و نقل مواد مخدر; OCT; MATE1; Telaprevir; OATP; Drug-drug interaction; Drug transporter;
Organic cation transporter OCT/SLC22A and H+/organic cation antiporter MATE/SLC47A are key molecules for nephrotoxicity of platinum agents
Keywords: حمل و نقل مواد مخدر; OCT, organic cation transporter; MATE, multidrug and toxin extrusion; Ctr1, copper transporter 1; DACH, diaminocyclohexaneCisplatin; Renal handling; Pharmacokinetics; Drug transporter; Copper transporter Ctr1
Nanoparticles attenuate P-glycoprotein/MDR1 function in A549 human alveolar epithelial cells
Keywords: حمل و نقل مواد مخدر; A549 cells; Rhodamine 123; Drug transporter; Release study;
Molecular and Cellular PharmacologyDifferential modulation of the expression of important drug metabolising enzymes and transporters by endothelin-1 receptor antagonists ambrisentan and bosentan in vitro
Keywords: حمل و نقل مواد مخدر; Bosentan; Ambrisentan; Pulmonary arterial hypertension; Drug transporter; Drug metabolising enzyme; Induction;
Efficient sequential synthesis of PET Probes of the COX-2 inhibitor [11C]celecoxib and its major metabolite [11C]SC-62807 and in vivo PET evaluation
Keywords: حمل و نقل مواد مخدر; Drug transporter; Biliary excretion; PET (positron emission tomography); Radiochemistry; Celecoxib; SC-62807
Strategies for bypassing the membrane barrier in multidrug resistant Gram-negative bacteria
Keywords: حمل و نقل مواد مخدر; Antibiotic; Bacterial efflux pump; Chemosensitizer; Drug transporter; Efflux pump inhibitor; Gram-negative bacteria; Lipopolysaccharide; MDR bacteria; Membrane permeability; Natural compound; Porin; Selectivity
Systematic Screening of Human ABCC3 Polymorphisms and Their Effects on MRP3 Expression and Function
Keywords: حمل و نقل مواد مخدر; ABCC3; drug transporter; human; MRP3; pharmacogenomics; pharmacokinetics; polymorphism;
Inhibition of anticancer drug efflux transporter P-glycoprotein by rosemary phytochemicals
Keywords: حمل و نقل مواد مخدر; P-glycoprotein; Drug transporter; Anticancer drug; Rosemary; Phytochemical
Cloning/characterization of the canine organic anion transporting polypeptide 1b4 (Oatp1b4) and classification of the canine OATP/SLCO members
Keywords: حمل و نقل مواد مخدر; BSP, bromosulfophthalein; CCK-8, cholecystokinin octapeptide; DPDPE, [D-penicillamine2,5]enkephalin; E17βG, estradiol-17β-glucuronide; HEK293, human embryonic kidney cells 293; OATP, organic anion transporting polypeptideOATP; Drug transporter; Kinetics;
Angiotensin II inhibits activity of human organic anion transporter 3 through activation of protein kinase Cα: Accelerating endocytosis of the transporter
Keywords: حمل و نقل مواد مخدر; Drug transporter; Regulation; Angiotensin II; Protein Kinase C; Endocytosis; COS-7 Cells
Major contribution of tubular secretion to creatinine clearance in mice
Keywords: حمل و نقل مواد مخدر; creatinine clearance; drug transporter; gender difference; glomerular filtration rate; ion transport
mTOR inhibitor everolimus ameliorates progressive tubular dysfunction in chronic renal failure rats
Keywords: حمل و نقل مواد مخدر; Mammalian target of rapamycin; Proximal tubule injury; Albuminuria; Drug transporter; Chronic kidney disease;
Cloning and pharmacological characterization of a novel gene encoding human nucleoside transporter 1 (hNT1) from a human breast cancer cDNA library
Keywords: حمل و نقل مواد مخدر; Breast cancer; Drug transporter; 5-Fluorouracil; Nucleoside transporter
Knockdown of PgP resensitizes leukemic cells to proteasome inhibitors
Keywords: حمل و نقل مواد مخدر; Cancer; Drug resistance; Proteasome inhibitors; Drug transporter; PgP; MDR-1;
Genotyping of eight polymorphic genes encoding drug-metabolizing enzymes and transporters using a customized oligonucleotide array
Keywords: حمل و نقل مواد مخدر; Genetic polymorphism; Drug-metabolizing enzyme; Drug transporter; Genotyping; Allele-specific primer extension
P-glycoprotein-deficient mice have proximal tubule dysfunction but are protected against ischemic renal injury
Keywords: حمل و نقل مواد مخدر; kidney dysfunction; drug transporter; ABC transporter; ischemia-reperfusion
Species Differences of Inhibitory Effects on PâglycoproteinâmediateD Drug Transport
Keywords: حمل و نقل مواد مخدر; multidrug resistance transporters; Pâglycoprotein; inhibition; species differences; drug interaction; drug transporter;
Identification of six putative human transporters with structural similarity to the drug transporter SLC22 family
Keywords: حمل و نقل مواد مخدر; Drug transporter; SLC22; Solute carrier; Anion; Cation
Orange juice increased the bioavailability of pravastatin, 3-hydroxy-3-methylglutaryl CoA reductase inhibitor, in rats and healthy human subjects
Keywords: حمل و نقل مواد مخدر; HMG-CoA reductase inhibitor; Orange juice; Bioavailability; Human; Drug interaction; Drug transporter; Intestine
Functional expression of sinusoidal and canalicular hepatic drug transporters in the differentiated human hepatoma HepaRG cell line
Keywords: حمل و نقل مواد مخدر; Drug transporter; Hepatocytes; HepaRG cells; Hepatoma; Detoxification
Pharmacogenetics: antidepressant drug response
Keywords: حمل و نقل مواد مخدر; basic sciences; pharmacogenetics; depression; antidepressant; metabolism; drug transporter; serotonin; noradrenaline; cytochrome P450;
Localization of organic anion transporting polypeptides in the rat and human ciliary body epithelium
Keywords: حمل و نقل مواد مخدر; organic anion transporter; ciliary body epithelium; drug transporter; unoprostone;