Keywords: نسبت خروجی; AUC; area under the concentration-time curve; AST; aspartate transaminase; ALT; alanine transaminase; BCRP; breast cancer resistance protein; BEI; biliary excretion index; CL/F; oral clearance; Clbiliary; in vitro biliary clearance; ER; Efflux Ratio; LCâ
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: نسبت خروجی; AP; apical; BL; basolateral; CB; (1E,4E)-1,5-bis (3-methoxy-4-hydroxy phenyl)-1,4-diene-3-pentanone; Cur; curcumin; DMEM; dulbecco's modified eagle's medium; DMSO; dimethyl sulfoxide; EDTA; ethylenediaminetetraacetic acid; ER; efflux ratio; FBS; fetal
The influence of compatibility of Si-Ni decoction with metabolism in intestinal bacteria on transports of toxic diterpenoid alkaloids from processed aconite root across Caco-2 monolayers
Keywords: نسبت خروجی; AD; Decoction of processed aconite root; ALD; Decoction of processed aconite root and honey-processed liquorice; AP; Apical; BCRP; Breast cancer resistance protein; BL; Basolateral; DDAs; Diester-diterpenoid alkaloids; EIC; Extracted ion chromatogram; ER;
Characterization of the IPEC-J2 MDR1 (iP-gp) cell line as a tool for identification of P-gp substrates
Keywords: نسبت خروجی; P-glycoprotein; Efflux ratio; ABCB1; MDR1-P-gp inhibitor; Digoxin; Rhodamine 123; Zosuquidar; Monolayer;
Assessment of HBEC-5i endothelial cell line cultivated in astrocyte conditioned medium as a human blood-brain barrier model for ABC drug transport studies
Keywords: نسبت خروجی; Blood-Brain Barrier; ABC transporters; Efflux ratio; Human in vitro models; Astrocyte conditioned medium;
The expected characteristics of an in vitro human Blood Brain Barrier model derived from cell lines, for studying how ABC transporters influence drug permeability
Keywords: نسبت خروجی; Blood-brain-barrier; ABC transporters; in vitro model; Pharmacological model; Drug permeability; Efflux ratio;
A systematic review of pharmacokinetic studies on herbal drug Fuzi: Implications for Fuzi as personalized medicine
Keywords: نسبت خروجی; Aconitum carmichaeli Debx.; Aconitum alkaloids; Pharmacokinetics; Herb-drug interactions; Toxicology; Personalized medicine; DMEs; drug-metabolizing enzymes; ETs; efflux transporters; BB; bioavailability barrier; DDAs; diester-diterpene alkaloids; MDAs; m
Abcb1a (P-glycoprotein) limits brain exposure of the anticancer drug candidate seliciclib in vivo in adult mice
Keywords: نسبت خروجی; Seliciclib; Blood-brain barrier; P-glycoproptein; Mice; Microdialysis; BBB; blood brain barrier; ER; efflux ratio; CDK; cyclin-dependent kinase; ABCB1/P-gp/MDR1; ATP-binding Cassette B1/P-glycoprotein/Multidrug Resistance Protein 1; CSF; arteficial cerebr
P-Glycoprotein in skin contributes to transdermal absorption of topical corticosteroids
Keywords: نسبت خروجی; P-gp; P-glycoprotein; BCRP; breast cancer resistance protein; SC; stratum corneum; ABC; ATP-binding cassette; MDR1; multidrug resistance 1; MDCK II; Madin-Darby canine kidney II; BL; basal; AP; apical; ER; efflux ratio; Papp; apparent permeability coeffic
Validation of UHPLC-MS/MS methods for the determination of kaempferol and its metabolite 4-hydroxyphenyl acetic acid, and application to in vitro blood-brain barrier and intestinal drug permeability studies
Keywords: نسبت خروجی; 4-HPAA; 4-hydroxyphenyl acetic acid; ACN; acetonitrile; BSA; bovine serum albumin; Cal; calibrator; CCl; cell layer capacitance; CNS; central nervous system; CV%; coefficient of variation; CPT-cAMP; 8-(4-chlorophenylthio)-adenosine-3â²,5â²-cyclic monoph
Research paperEffects of herbal drugs in Mahuang decoction and their main components on intestinal transport characteristics of Ephedra alkaloids evaluated by a Caco-2 cell monolayer model
Keywords: نسبت خروجی; TCM; traditional Chinese medicine; MHP; multi-herb prescription; LEP; l-ephedrine; DPEP; d-pseudoephedrine; LMEP; l-methylephedrine; P-gp; P-glycoprotein; ER; efflux ratio; AP; apical; BL; basolateral; Papp; apparent permeability; PAB; permeability from A
Establishment of Optimized MDCK Cell Lines for Reliable Efflux Transport Studies
Keywords: نسبت خروجی; ABC transporter; Pâglycoprotein; MDCK; Cell lines; homogenous population; PCR; bidirectional transport assays; Pgp; Pâglycoprotein; MDCK; MadinâDarby canine kidney cell line; ABC transporters; ATPâbinding cassette transporters; ER; efflux ratio; N
Transport of ginkgolides with different lipophilicities based on an hCMEC/D3 cell monolayer as a blood–brain barrier cell model
Keywords: نسبت خروجی; Transport; BBB; Ginkgolide; hCMEC/D3 cell; Apparent permeability coefficients; Efflux ratio; Lipophilicity
Kinase domain inhibition of leucine rich repeat kinase 2 (LRRK2) using a [1,2,4]triazolo[4,3-b]pyridazine scaffold
Keywords: نسبت خروجی; AD; Alzheimer's disease; ANK; ankyrin repeat domain; ARM; armadillo repeat domain; AUC; area under the curve; BA; brain availability; BBB; blood brain barrier; BCRP; breast cancer related protein; BI; brain impairment; CSD; Cambridge Structural Database
Accelerated Caco-2 cell permeability model for drug discovery
Keywords: نسبت خروجی; Drug permeability; Caco-2 cells; P-glycoprotein; Puromycin; Accelerated model; Efflux ratio; Drug discovery
Evaluation of various PAMPA models to identify the most discriminating method for the prediction of BBB permeability
Keywords: نسبت خروجی; Permeability; Solubility; PAMPA; Caco-2; Efflux ratio; Log BB; Blood–brain barrier
P-glycoprotein and cytochrome P450 3A4 involvement in risperidone transport using an in vitro Caco-2/TC7 model and an in vivo model
Keywords: نسبت خروجی; ab; apical to basolateral; AQ; absorptive quotient; AUCT; area under the curve; ba; basolateral to apical; ClR; renal clearance; Cmax; maximum plasma concentration; CYP; cytochrome P450; ER; efflux ratio; F; fraction not metabolised; FA; fraction absorbed
Modulation of drug transport by selected flavonoids: Involvement of P-gp and OCT?
Keywords: نسبت خروجی; OCT; organic cation transporter; P-gp; P-glycoprotein; MDR; multidrug resistance; TEA; tetraethylammoniumbromide; MES; 2-(N-morpholino)-ethanesulfonic acid; TEER; transepithelial electrical resistance; DMEM; Dulbecco's modified eagle medium; FBS; fetal