Keywords: 1-AA; 1-aminoanthracene; 2-EP; 2-ethylpyridine; 2-PIC; 2-picolylamine; AMP; amphetamine; AMY1; amylose tris-(3,5-dimethyl-phenylcarbamate); BEH; bridged ethylene hybrid silica; CCH; cannabicyclohexanol; CEL1; cellulose tris-(3,5-dimethyl-phenylcarbamate);
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An SAR study of hydroxy-trifluoromethylpyrazolines as inhibitors of Orai1-mediated store operated Ca2+ entry in MDA-MB-231 breast cancer cells using a convenient Fluorescence Imaging Plate Reader assay
Keywords: FLIPR; Fluorescence Imaging Plate Reader; STIM1; stromal interaction molecule 1; ER; endoplasmic reticulum; TNBC; triple negative breast cancer; SAR; structure activity relationship; LHS; left hand side; RHS; right hand side; THF; tetrahydrofuran; i-PrOH;
Discovery of spiro[indole-3,2â²-pyrrolidin]-2(1H)-one based inhibitors targeting Brr2, a core component of the U5 snRNP
Keywords: CDCl3; deuterated chloroform; DHX29; DEAH-Box helicase 29 (an ATP-dependent RNA helicase); DIPEA; N,Nâ²-diisopropylethylamine; DMSO-d6; dimethyl sulfoxide-d6; EDC·HCl; 1-(3-(dimethylamino)propyl)-3-ethylcarbodiimide hydrochloride; eIF4A1; eukaryotic ini
Traditional uses, phytochemistry, pharmacology and toxicology of the genus Cimicifuga: A review
Keywords: TCM; traditional Chinese medicine; TLC; thin-layer chromatography; PCA; principal component analysis; XMT; brand name of the alcoholic extract of C. foetida; FST; forced swimming test; TST; tail suspension test; MeOH; methanol; i-PrOH; isopropanolic; CH;
Structure-based design of a new series of N-(piperidin-3-yl)pyrimidine-5-carboxamides as renin inhibitors
Keywords: AcOH; acetic acid; Ang I; angiotensin I; Ang II; angiotensin II; AUC; area under the blood concentration-time curve; C5min; concentration in plasma 5Â min after administration; CLtotal; total clearance; Cmax; maximum concentration in plasma; DIEA; N,N-d
Polymeric pH-sensitive membranes-A review
Keywords: AA; acrylic acid; AAm; acryl amide; AFM; atomic force microscopy; AIBN; 2,2â²-azo-bisisobutyronitrile; AMPS; 2-acrylamido-2-methylpropanesulfonic acid; AOHOBA; 4-(6-(acryloyloxy)hexyloxy) benzoic acid; ATRP; atom transfer radical polymerisation; BP; benz
Evaluation of new leptin fragments on food intake and body weight of normal rats
Keywords: 2-Cl-Z; 2-chloro-benzyloxycarbonyl; AAA; amino acid analysis; BOP; benzotriazol-1-yl-oxy-tris(dimethylamino) phosphonium hexafluorophosphate; Bzl; benzyl; CD; circular dichroism; CH3CN; acetonitrile; CHO; Formyl; CSF; Cerebrospinal fluid; DCM; dichloromet
Disproportionation reaction of diarylmethylisopropyl ethers: a versatile access to diarylmethanes from diarylcarbinols speeded up by the use of microwave irradiation
Keywords: Disproportionation; Diarylcarbinols; Diarylmethanes; i-PrOH; CBr4; TfOH; Microwave heating;
Solvatochromism of 3-[2-(aryl)benzoxazol-5-yl]alanine derivatives
Keywords: BoxAnt; N-Boc-3-[2-(9-anthryl)benzoxazol-5-yl]-l-alanine methyl ester; BoxPhAnt; N-Boc-3-[2-[4-(9â²-(10â²-butyl)anthryl)phenyl]benzoxazol-5-yl]-l-alanine methyl ester; MeOH; methanol; EtOH; ethanol; 1-BuOH; 1-butanol; i-PrOH; 2-propanol; 1-PeOH; 1-penta