Kinetics of human cannabinoid 1 (CB1) receptor antagonists: Structure-kinetics relationships (SKR) and implications for insurmountable antagonism
Keywords: Residence time; Structure-kinetics relationships; Cannabinoid 1 receptor; Insurmountable antagonism; Radioligand binding; Preincubation; Rimonabant (PubChem CID: 104850); CP55940 (PubChem CID: 104895); Antagonist 1 (CAS Registry Number: 1207203-10-8); Ant