
Discovery of quinolinone derivatives as potent FLT3 inhibitors
Keywords: Fms-like tyrosine kinase 3 (FLT3); Acute myeloid leukemia; QuinolinoneFLT3, fms-like tyrosine kinase 3; AML, acute myeloid leukemia; ITD, internal tandem duplication; HTRF, homogeneous time-resolved fluorescence; TR-FRET, time resolved-fluorescence resona