دانلود مقالات ISI درباره Ki ثابت نگهدارنده + ترجمه فارسی

مهار کننده قوی تریروزیناز، نوروفلاوان از کمپیلتروپیس هیرتللا و مکانیسم مهارکننده با سوسپانسیون مولکولی

Highly potent tyrosinase inhibitor, neorauflavane from Campylotropis hirtella and inhibitory mechanism with molecular docking

Keywords: Ki ثابت نگهدارنده; IC50, the inhibitor concentration leading 50% activity loss; Ki, inhibition constant; Kiapp, apparent Ki; K, rate constant; Vmax, maximum velocity; Km, Michaelis−Menten constant; Kobs, apparent first-order rate constant for the transition from νi to νs; ν

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2016 سفارش ترجمه

بررسی اثر ضدرنگدانه کالکون sulfonylamino مصنوعی

Evaluation of anti-pigmentary effect of synthetic sulfonylamino chalcone

Keywords: Ki ثابت نگهدارنده; Chalcone; Depigmentation; Sulfonylamino chalcone; TyrosinaseIC50, the inhibitor concentration leading to 50 % activity loss; Ki, inhibition constant; TRP-1, tyrosinase related protein-1; TRP-2, tyrosinase related protein-2; α-MSH, α-melanocyte stimulating

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2017 سفارش ترجمه

Comparison of the susceptibility of porcine and human dipeptidyl-peptidase IV to inhibition by protein-derived peptides

Keywords: Ki ثابت نگهدارنده; α-la, alpha-lactalbumin; GIP, glucose-dependent insulinotropic polypeptide; β-lg, beta-lactoglobulin; GLP-1, glucagon-like peptide-1; Gly-Pro-p-NA, Gly-Pro-para-nitroanilide; Ki, inhibition constant; Lf, lactoferrin; NPY, neuropeptide Y; pDPP-IV, porcine

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2015 سفارش ترجمه

Comparative analysis of human CYP3A4 and rat CYP3A1 induction and relevant gene expression by bisphenol A and diethylstilbestrol: Implications for toxicity testing paradigms

Keywords: Ki ثابت نگهدارنده; BPA, bisphenol A; DES, diethylstilbestrol; DMSO, dimethyl sulfoxide; EC50, half maximal effective concentration; EDC, endocrine-disrupting chemical; EPA, Environmental Protection Agency; Ki, inhibition constant; LOAEL, lowest observed adverse effect level

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2013 سفارش ترجمه

Stereo-selective binding of monoclonal antibodies to the poly-gamma-d-glutamic acid capsular antigen of Bacillus anthracis

Keywords: Ki ثابت نگهدارنده; γDPGA, γ-linked d-polyglutamic acid; γLPGA, γ-linked l-polyglutamic acid; mAb, monoclonal antibody; pAb, polyclonal antibody; SPR, surface plasmon resonance; KI, inhibition constant; KD, dissociation constantAntibody; Anthrax; Polyglutamic acid capsule; S

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2013 سفارش ترجمه

In vitro inhibitory effects of asiaticoside and madecassoside on human cytochrome P450

Keywords: Ki ثابت نگهدارنده; BOMCC, 7-benzyloxymethyloxy-3-cyanocoumarin; CYP, cytochrome P450; DBOMF, dibenzyloxymethylfluorescein; EOMCC, ethoxymethyloxy-3-cyanocoumarin; IC50, median inhibitory concentration; Ki, inhibition constant; Km, the Michaelis constant; MW, molecular weigh

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2011 سفارش ترجمه

Tyrosinase inhibitory activity of a 6-isoprenoid-substituted flavanone isolated from Dalea elegans

Keywords: Ki ثابت نگهدارنده; IC50, the inhibitor concentration leading to 50% activity loss; KI, inhibition constant; Vmax, maximum velocity; Km, Michaelis–Menten constant; A, absorbance; PPO, polyphenol oxidase; l-DOPA, 3,4-dihydroxy-l-phenylalanine; TLC, thin layer chromatography;

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2011 سفارش ترجمه

SARS-CoV 3CLpro inhibitory effects of quinone-methide triterpenes from Tripterygium regelii

Keywords: Ki ثابت نگهدارنده; IC50, the inhibitor concentration leading to 50% activity loss; Ki, inhibition constant; Km, Michaelis–Menten constant; Vmax, maximum velocity; NMR, nuclear magnetic resonanceSARS-CoV; 3CLpro; Tripterygium regelii; Quinone-methide; Celastrol; Iguesterin

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2010 سفارش ترجمه

Caloxin 1b3: A novel plasma membrane Ca2+-pump isoform 1 selective inhibitor that increases cytosolic Ca2+ in endothelial cells

Keywords: Ki ثابت نگهدارنده; [Ca2+]i, cytosolic [Ca2+]; EDTA, ethylenediamine tetra-acetic acid; EGTA, ethylene glycol-bis(-aminoethyl ether)-N,N,N′,N′-tetraacetic acid; exdom, extracellular domain; HEPES, N-2-hydroxyethylpiperazine-N′-2-ethanesulfonic acid; Ki, inhibition constant;

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2010 سفارش ترجمه

Experimental and theoretical affinity studies of substituted phenols to chlorocatechol 1,2-dioxygenases: A step toward the comprehension of inhibitor/substrate binding to intradiol dioxygenases

Keywords: Ki ثابت نگهدارنده; CCD, chlorocatechol 1,2-dioxygenase; Ki, inhibition constant; pKa, acid–base dissociation constant; AM1, Austin model 1; DPE, deprotonation enthalpies; Hf, heat of formation; EHOMO, energy of the highest occupied molecular orbital; HOMO, highest occupied

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2010 سفارش ترجمه

Xanthones with neuraminidase inhibitory activity from the seedcases of Garcinia mangostana

Keywords: Ki ثابت نگهدارنده; Garcinia mangostana; Xanthone; Neuraminidase; Time-dependentI, intensity at ex: 365 nm, em: 450 nm; IC50, the inhibitor concentration leading to 50% activity loss; Ki, inhibition constant; Kiapp, apparent Ki; kobs, apparent first-order rate constant for t

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2010 سفارش ترجمه

Biflavonoids from Torreya nucifera displaying SARS-CoV 3CLpro inhibition

Keywords: Ki ثابت نگهدارنده; SARS, severe acute respiratory syndrome; CoV, coronavirus; IC50, concentration producing a 50% reducing in activity; Ki, inhibition constant; Vmax, maximum velocity; Km, Michaelis-Menten constant; RFUs, relative fluorescence unitsSARS-CoV 3CLpro; Torreya

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2010 سفارش ترجمه

Tricyclic antidepressants and mecamylamine bind to different sites in the human α4β2 nicotinic receptor ion channel

Keywords: Ki ثابت نگهدارنده; AChR, nicotinic acetylcholine receptor; NCA, noncompetitive antagonist; TCAs, tricyclic antidepressants; κ-BTx, κ-bungarotoxin; RT, room temperature; BS buffer, binding saline buffer; Ki, inhibition constant; Kd, dissociation constant; Ka, association con

دانلود رایگان متن کامل مقاله ISI 12 صفحه سال انتشار : 2010 سفارش ترجمه

Tyrosinase inhibitory effects of 1,3-diphenylpropanes from Broussonetia kazinoki

Keywords: Ki ثابت نگهدارنده; IC50, The inhibitor concentration leading to 50% activity loss; Ki, inhibition constant; Kiapp, apparent Ki; k, rate constant; Vmax, maximum velocity; Km, Michaelis–Menten constant; kobs, apparent first-order rate constant for the transition from vi to vs

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2009 سفارش ترجمه

Characteristic of neuraminidase inhibitory xanthones from Cudrania tricuspidata

Keywords: Ki ثابت نگهدارنده; I, intensity at ex: 365 nm, em: 450 nm; IC50, the inhibitor concentration leading to 50% activity loss; Ki, inhibition constant; Kiapp, apparent Ki; kobs, apparent first-order rate constant for the transition from vi to vs; vi, initial velocity; vs, stead

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2009 سفارش ترجمه

Designing Out Disulfide Bonds of Leech Carboxypeptidase Inhibitor: Implications for Its Folding, Stability and Function

Keywords: Ki ثابت نگهدارنده; bis-ANS, 4,4'-bis(1-anilinonaphthalene-8-sulfonate); BPTI, bovine pancreatic trypsin inhibitor; CPA, carboxypeptidase A; GdnHCl, guanidine hydrochloride; GSH, reduced glutathione; GSSG, oxidized glutathione; Ki, inhibition constant; LCI, leech carboxypept

دانلود رایگان متن کامل مقاله ISI 18 صفحه سال انتشار : 2009 سفارش ترجمه

Synergistic Ca2+ and Cu2+ requirements of the FGF1–S100A13 interaction measured by quartz crystal microbalance: An initial step in amlexanox-reversible non-classical release of FGF1

Keywords: Ki ثابت نگهدارنده; FGF1, fibroblast growth factor-1; EC50, median effective concentration; ka, association rate constant; KD, dissociation constant; Ki, inhibition constant; Cys, cysteine; QCM, quartz crystal microbalance; GST, glutathione S-transferase; MW, molecular weigh

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2008 سفارش ترجمه

Identification of dynorphin a from zebrafish: A comparative study with mammalian dynorphin A

Keywords: Ki ثابت نگهدارنده; dynorphin A; opioid receptors; radioligand binding; [35S]GTPγS stimulation; zebrafishEC50, mean effective dose; GDP, guanosine 5′-diphosphate; GTPγS, guanosine 5′-[γ-thio]triphosphate; IE, Ile-enkephalin; Ki, inhibition constant; mDYN A, mammalian dynorph

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2007 سفارش ترجمه

Effects of chronic opioid exposure on guinea pig mu opioid receptor in Chinese hamster ovary cells: Comparison with human and rat receptor

Keywords: Ki ثابت نگهدارنده; Bmax, maximum receptor binding; CHO, Chinese hamster ovary; DAMGO, [d-AIa2,N-Me-Phe4,Gly5-ol]-enkephalin; DPDPE, [d-Pen2,5]-enkephalin; Emax, maximum effect; gp, guinea pig; hu, human; Ki, inhibition constant; M3G, morphine-3-β-d-glucuronide; M6G, morphin

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2007 سفارش ترجمه