دانلود مقالات ISI درباره arylpiperazines طولانی زنجیره ای + ترجمه فارسی

New N- and O-arylpiperazinylalkyl pyrimidines and 2-methylquinazolines derivatives as 5-HT7 and 5-HT1A receptor ligands: Synthesis, structure-activity relationships, and molecular modeling studies

Keywords: arylpiperazines طولانی زنجیره ای; 5-HT7 receptor ligands; 5-HT1A receptor ligands; Long-chain arylpiperazines; Molecular modeling;

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2017 سفارش ترجمه

α-Adrenoceptor antagonistic and hypotensive properties of novel arylpiperazine derivatives of pyrrolidin-2-one

Keywords: arylpiperazines طولانی زنجیره ای; α-Adrenoceptors antagonists; Hypotensive activity; Pyrrolidin-2-one derivatives; Long-chain arylpiperazines

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2015 سفارش ترجمه

Antidepressant- and anxiolytic-like activity of 7-phenylpiperazinylalkyl-1,3-dimethyl-purine-2,6-dione derivatives with diversified 5-HT1A receptor functional profile

Keywords: arylpiperazines طولانی زنجیره ای; Purine-2,6-diones; Long-chain arylpiperazines; Depression; Anxiety; 5-HT1A receptor agonist/antagonist; 5-HT2A receptor antagonist; 5-HT7 receptor antagonist;

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2015 سفارش ترجمه

Structure-activity relationships and molecular studies of novel arylpiperazinylalkyl purine-2,4-diones and purine-2,4,8-triones with antidepressant and anxiolytic-like activity

Keywords: arylpiperazines طولانی زنجیره ای; Imidazo[2,1-f]purine-2,4-diones; Tricyclic theophylline derivatives; Serotonin; Long-chain arylpiperazines; Schizophrenia; Depression;

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2015 سفارش ترجمه

Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT1A activity. Part 5

Keywords: arylpiperazines طولانی زنجیره ای; Pyrido[1,2-c]pyrimidines; Antidepressants; Dual SSRI/5-HT1A activity; Quinoline derivatives; SERT; serotonin transporter; SAR; structure-activity relationship; 5-HT1AR; serotonin 5-HT1A receptors; 8-OH-DPAT; 8-hydroxy-2-(di-n-propylamino)tetralin; Ki; inh

دانلود رایگان متن کامل مقاله ISI 65 صفحه سال انتشار : 2015 سفارش ترجمه

New 7-arylpiperazinylalkyl-8-morpholin-4-yl-purine-2,6-dione derivatives with anxiolytic activity – Synthesis, crystal structure and structure–activity study

Keywords: arylpiperazines طولانی زنجیره ای; Long-chain arylpiperazines; Purine-2,6-dione derivatives; 5-HT receptor ligands; X-ray structure analysis

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2014 سفارش ترجمه

Solid-supported synthesis, molecular modeling, and biological activity of long-chain arylpiperazine derivatives with cyclic amino acid amide fragments as 5-HT7 and 5-HT1A receptor ligands

Keywords: arylpiperazines طولانی زنجیره ای; Long-chain arylpiperazines; Solid-phase synthesis; Prolinamides; Pipecolic acid; 1,2,3,4-Tetrahydroisoquinoline-3-carboxamides; Hydrogen bonding; 5-HT7 receptor ligands; 5-HT1A receptor ligands;

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2014 سفارش ترجمه

Antidepressant and antipsychotic activity of new quinoline- and isoquinoline-sulfonamide analogs of aripiprazole targeting serotonin 5-HT1A/5-HT2A/5-HT7 and dopamine D2/D3 receptors

Keywords: arylpiperazines طولانی زنجیره ای; Quinoline-sulfonamides; Isoquinoline-sulfonamides; Long-chain arylpiperazines; 2,3-Dichlorophenylpiperazine; Serotonin; Dopamine; 5-HT2A antagonist; D2 partial agonist; 5-HT7 antagonist; Aripiprazole; Depression; Schizophrenia

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2013 سفارش ترجمه

Quinoline- and isoquinoline-sulfonamide derivatives of LCAP as potent CNS multi-receptor-5-HT1A/5-HT2A/5-HT7 and D2/D3/D4-agents: The synthesis and pharmacological evaluation

Keywords: arylpiperazines طولانی زنجیره ای; Quinolinesulfonamides/isoquinolinesulfonamides; Long-chain arylpiperazines; 5-HT2A receptor antagonist; 5-HT7 receptor antagonist; D2 antagonist; Depression; Anxiety; Schizophrenia;

دانلود رایگان متن کامل مقاله ISI 12 صفحه سال انتشار : 2012 سفارش ترجمه

The multiobjective based design, synthesis and evaluation of the arylsulfonamide/amide derivatives of aryloxyethyl- and arylthioethyl- piperidines and pyrrolidines as a novel class of potent 5-HT7 receptor antagonists

Keywords: arylpiperazines طولانی زنجیره ای; Solid-phase synthesis; BAL linker; Virtual combinatorial library; Virtual screening; Long-chain arylpiperazines; Alicyclic amines; Arylsulfonamides; Aryloxyalkyl-piperidines; Aryloxyalkyl-pyrrolidines; 5-HT7 antagonists

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2012 سفارش ترجمه

Synthesis and structural investigation of some pyrimido[5,4-c]quinolin-4(3H)-one derivatives with a long-chain arylpiperazine moiety as potent 5-HT1A/2A and 5-HT7 receptor ligands

Keywords: arylpiperazines طولانی زنجیره ای; Pyrimidoquinolones; Long-chain arylpiperazines; 5-HT receptor ligands; Molecular modeling;

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2011 سفارش ترجمه

The influence of an ethylene spacer on the 5-HT1A and 5-HT2A receptor affinity of arylpiperazine derivatives of amides with N-acylated amino acids and 3-differently substituted pyrrolidine-2,5-diones

Keywords: arylpiperazines طولانی زنجیره ای; Long-chain arylpiperazines; Succinimides; Spirosuccinimides; Pyrrolidine-2,5-dione; 2-Azaspiro[4.5]decane-1,3-dione; Pyrrolidine-5-one-carboxamide; Prolinamides; Solid-phase synthesis; 5-HT1A/5-HT2A receptor ligands;

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2009 سفارش ترجمه

7-Arylpiperazinylalkyl and 7-tetrahydroisoquinolinylalkyl derivatives of 8-alkoxy-purine-2,6-dione and some of their purine-2,6,8-trione analogs as 5-HT1A, 5-HT2A, and 5-HT7 serotonin receptor ligands

Keywords: arylpiperazines طولانی زنجیره ای; Purine-2,6-diones; Purine-2,6,8-triones; Long-chain arylpiperazines; 5-HT1A; 5-HT2A; 5-HT7 receptor ligands

دانلود رایگان متن کامل مقاله ISI 12 صفحه سال انتشار : 2007 سفارش ترجمه

Novel class of arylpiperazines containing N-acylated amino acids: Their synthesis, 5-HT1A, 5-HT2A receptor affinity, and in vivo pharmacological evaluation

Keywords: arylpiperazines طولانی زنجیره ای; Long-chain arylpiperazines; Succinimides; Pyrrolidine-2,5-dione; Prolinamides; Solid-phase synthesis; 5-HT1A/5-HT2A receptor ligands; 5-HT1A receptor agonists; Four-plate test; Forced swimming test; Tail suspension test

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2007 سفارش ترجمه

Arylpiperazines with N-acylated amino acids as 5-HT1A receptor ligands

Keywords: arylpiperazines طولانی زنجیره ای; Long-chain arylpiperazines; Succinimides; Pyroglutamates; Solid-phase synthesis; BAL linker; 5-HT1A receptor ligands; Fujita–Ban analysis

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2006 سفارش ترجمه