
Discovery of spiro[indole-3,2â²-pyrrolidin]-2(1H)-one based inhibitors targeting Brr2, a core component of the U5 snRNP
Keywords: CDCl3; deuterated chloroform; DHX29; DEAH-Box helicase 29 (an ATP-dependent RNA helicase); DIPEA; N,Nâ²-diisopropylethylamine; DMSO-d6; dimethyl sulfoxide-d6; EDC·HCl; 1-(3-(dimethylamino)propyl)-3-ethylcarbodiimide hydrochloride; eIF4A1; eukaryotic ini