Keywords: جذب بینی; Nasal absorption; Positron emission tomography; Pharmacokinetics; Nasopalatine; ViscosityPET, positron emission tomography; [18F]FDG, 2-deoxy-2-[18F]fluoro-d-glucose; HPC, hydroxypropylcellulose, H-grade; MRI, magnetic resonance image; VOIs, volumes of in
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Keywords: جذب بینی; Protein transduction domain (PTD); Translationally controlled tumor protein (TCTP); TCTP-PTD; Insulin; Nasal absorption;
The relationship between in vivo nasal drug clearance and in vitro nasal mucociliary clearance: Application to the prediction of nasal drug absorption
Keywords: جذب بینی; Nasal absorption; Mucociliary clearance; Prediction system; Nasal residence; Mucosal absorption; Nasal formulation;
Use of a non-covalent cell-penetrating peptide strategy to enhance the nasal delivery of interferon beta and its PEGylated form
Keywords: جذب بینی; Interferon β; PEGylation; Nasal absorption; Cell-penetrating peptides; Penetratin; Bioavailability
Zolpidem Mucoadhesive Formulations for Intranasal Delivery: Characterization, In Vitro Permeability, Pharmacokinetics, and Nasal Ciliotoxicity in Rats
Keywords: جذب بینی; bioavailability; excipients; formulation; nasal absorption; nasal drug delivery; permeability; pharmacokinetics; physicochemical properties; solubility;
The role of L-type amino acid transporters in the uptake of glyphosate across mammalian epithelial tissues
Keywords: جذب بینی; Glyphosate; Nasal absorption; Amino acid transporters; Caco-2Â cells; Olfactory epithelium; Nose to brain transport;
Improved Transnasal Transport and Brain Uptake of Tizanidine HCl-Loaded Thiolated Chitosan Nanoparticles for Alleviation of Pain
Keywords: جذب بینی; Chitosan; Nasal Drug Delivery; Nanoparticles; Nasal absorption; Paracellular transport;
Permeation and Systemic Absorption of R- and S-Baclofen Across the Nasal Mucosa
Keywords: جذب بینی; nasal absorption; nasal drug delivery; permeability; transporters; bioavailability; pharmacokinetics;
Formulation Optimization and Bioavailability After Oral and Nasal Administration in Rabbits of Puerarin-Loaded Microemulsion
Keywords: جذب بینی; microemulsion; formulation; bioavailability; oral absorption; nasal absorption; puerarin;
The role of intermolecular interactions with penetratin and its analogue on the enhancement of absorption of nasal therapeutic peptides
Keywords: جذب بینی; Cell-penetrating peptide (CPP); Penetratin analogues; Peptides; Nasal absorption; Intermolecular binding; Surface plasmon resonance (SPR)
Nasal absorption of mixtures of fast-acting and long-acting insulins
Keywords: جذب بینی; Absorption enhancer; Nasal absorption; Surfactants; Insulin; Diabetes; Drug delivery
Structural requirements of penetratin absorption enhancement efficiency for insulin delivery
Keywords: جذب بینی; Cell-penetrating peptide (CPP); Penetratin; Penetratin analogues; Insulin; Nasal absorption; Cytotoxicity
Effects of polyamidoamine (PAMAM) dendrimers on the nasal absorption of poorly absorbable drugs in rats
Keywords: جذب بینی; PAMAM dendrimer; Nasal absorption; Absorption enhancer; Insulin; Calcitonin; Toxicity
Thiolated Polycarbophil as an Adjuvant for Permeation Enhancement in Nasal Delivery of Antisense Oligonucleotides
Keywords: جذب بینی; phosphorothioate antisense oligonucleotides; polycarbophilâcysteine; thiomer; permeation enhancement; drug delivery system; tight junction; nasal absorption; cell culture; HPLC; polymer biodegradation;
Effect of cell-penetrating peptides on the nasal absorption of insulin
Keywords: جذب بینی; Cell-penetrating peptide (CPP); Penetratin; Octaarginine; Insulin; Nasal absorption
Preparation of ergoloid mesylate submicron emulsions for enhancing nasal absorption and reducing nasal ciliotoxicity
Keywords: جذب بینی; Ergoloid mesylate; Submicron emulsions; Nasal absorption; Microdialysis; Brain-targeting; Ciliotoxicity
The transnasal delivery of 5-fluorouracil to the rat brain is enhanced by acetazolamide (the inhibitor of the secretion of cerebrospinal fluid)
Keywords: جذب بینی; Nasal absorption; Cerebrospinal fluid; Brain delivery; Brain uptake clearance; Acetazolamide; 5-Fluorouracil
Identification of Tight Junction Modulating Lipids
Keywords: جذب بینی; tight junction; epithelial delivery/permeability; lipids/lipoproteins; mucosal delivery; nasal absorption; ether lipids; glycosylated sphingosine; oxidized lipid; alkylglycosides; ceramides;
Brain uptake of an anti-ischemic agent by nasal administration of microparticles
Keywords: جذب بینی; cerebrospinal fluid; chitosan; CNS; controlled release; drug targeting; microparticles; nasal absorption; polymeric drug carrier; spray drying;
Influence of fillers in powder formulations containing N-acetyl-l-cysteine on nasal peptide absorption
Keywords: جذب بینی; Nasal absorption; Powder formulation; Filler; Mucolytic agent; Peptide
Enhancement of nasal absorption of large molecular weight compounds by combination of mucolytic agent and nonionic surfactant
Keywords: جذب بینی; Nasal absorption; Absorption enhancement; Mucolytic agent; Nonionic surfactant; Calcitonin
Improved nasal absorption of salmon calcitonin by powdery formulation with N-acetyl-l-cysteine as a mucolytic agent
Keywords: جذب بینی; Nasal absorption; Absorption enhancement; Powdery formulation; Mucolytic agent; Salmon calcitonin
Rapid-onset intranasal delivery of metoclopramide hydrochloride: Part I. Influence of formulation variables on drug absorption in anesthetized rats
Keywords: جذب بینی; Nasal absorption; Metoclopramide; Rapid-onset; Absorption enhancers
Role of dopamine transporter (DAT) in dopamine transport across the nasal mucosa
Keywords: جذب بینی; Dopamine transporter; Nasal absorption; Olfactory transport
Metabolism of Dopamine by the Nasal Mucosa
Keywords: جذب بینی; nasal absorption; nasal metabolism; monoamine oxidase; permeability; olfactory; nasal mucosa; membrane transport; dopamine; DOPAC; MAO, monoamine oxidase; ALDH, aldehyde dehydrogenase; COMT,catechol-O-methyl transferase; CNS, central nervous system; HVA,
Positively charged polyethylenimines enhance nasal absorption of the negatively charged drug, low molecular weight heparin
Keywords: جذب بینی; Low molecular weight heparin; Polyethylenimine; Nasal absorption; Enoxaparin; Conductivity
Carrier mediated transport of chlorpheniramine and chlorcyclizine across bovine olfactory mucosa: Implications on noseâtoâbrain transport
Keywords: جذب بینی; olfactory mucosa; Pâglycoprotein; membrane transport proteins; CNS; diffusion; nasal absorption; activation energy; chlorpheniramine; chlorcyclizine;
Transport of hydroxyzine and triprolidine across bovine olfactory mucosa: Role of passive diffusion in the direct nose-to-brain uptake of small molecules
Keywords: جذب بینی; Olfactory mucosa; P-glycoprotein; Efflux; Membrane transport proteins; CNS; Diffusion; Nasal absorption; Etoposide; Hydroxyzine; Triprolidine;
Nasal mucoadhesive drug delivery: Background, applications, trends and future perspectives
Keywords: جذب بینی; Absorption enhancer; Microparticles; Microspheres; Mucoadhesion; Mucociliary clearance; Nasal absorption; Nasal drug delivery; Polymer;