Keywords: موجودی شیمیایی جدید; Immobilized artificial membrane; Time-of-flight mass spectrometry; Blood-brain barrier; Quantitative structure-activity relationship; Liquid chromatography; High-throughput; AA; ammonium acetate; APC; Amemiya predictive criterion; BBB; blood-brain barrier
مقالات ISI موجودی شیمیایی جدید (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: موجودی شیمیایی جدید; Salts; Gemfibrozil; Intrinsic dissolution rate; Surface dissolution imaging; Focus variation; GEM; gemfibrozil; DSC; differential scanning calorimetry; XRPD; X-ray powder diffraction; API; active pharmaceutical ingredient; BCS; biopharmaceutical classific
Keywords: موجودی شیمیایی جدید; Spray drying; Solid dispersion; Amorphous; Poorly soluble drugs; Formulation; AFM; Atomic force microscopy; ANN; Artificial neural networks; ANOVA; Analysis of variance; API; Active pharmaceutical ingredient; ASD; Amorphous solid dispersion; ATC; Atorvast
Keywords: موجودی شیمیایی جدید; Propylene glycol (PG); Polyethylene glycol (PEG) 400; Pharmasolve (NMP); Combination vehicle; Tolerability; Safety; Rat; ALP; Alkaline Phosphatase; EDTA; Ethylene diamino tetra acetic acid; i.v; Intravenous; IVC; Individually ventilated cages; Kg; Kilogra
Capillary electrophoresis in the context of drug discovery
Keywords: موجودی شیمیایی جدید; ACE; affinity capillary electrophoresis; AGP; α-acid glycoprotein; AH; adrenaline hydrochloride; AIμEA; automatic micro-enzyme assay; AL; amlodipine; AT; antithrombin III; Bag3; Bcl2-associated anthanogene 3; BGE; background electrolyte; CM; chylomicron
Keywords: موجودی شیمیایی جدید; NCE; new chemical entity; SNI; spared nerve injury; SNL; spinal nerve ligation; PR; progressive ratio; 5-CSRTT; 5-choice serial reaction time task; SD; stimulus duration; ITI; inter trial interval; LH; limited hold; ICSS; intracranial self-stimulation; Nb
Keywords: موجودی شیمیایی جدید; CPR; Cytochrome P450 reductase;; CYP; Cytochrome P450;; DME; Drug metabolizing enzyme;; EC; Electrochemical cell;; EDES; Electrochemically-driven enzymatic system;; EMMA; Electrophoretically-mediated microanalysis;; FMO; Flavin-containing monooxygenase;;
In vitro secondary pharmacological profiling: An IQ-DruSafe industry survey on current practices
Keywords: موجودی شیمیایی جدید; AUC; Area Under the Curve; CRO; Contract Research Organization; CTA; Clinical Trial Authorization; GLP; Good Laboratory Practice; hERG; human ether-a-go-go-related gene; ICH; International Conference on Harmonization; IND; Investigational New Drug; IQ; In
Scratching the surface: Exploratory analysis of key opinion leaders on rate limiting factors in novel adjuvanted-vaccine development
Keywords: موجودی شیمیایی جدید; CARG; compound annual growth rate; EPhMRA; European Pharmaceutical Marketing Research Association for the Anatomical Classification of Pharmaceutical Products; FDA; Food and Drug Administration; GSK; Glaxo Smith Kline; HBV; Hepatitis B Virus; HPV; Human P
In vitro and in vivo evaluation of novel cinnamyl sulfonamide hydroxamate derivative against colon adenocarcinoma
Keywords: موجودی شیمیایی جدید; ACFs; aberrant crypt foci; AO/EB; acridine orange/ethidium bromide; CPCSEA; Committee for the Purpose of Control and Supervision of Experiments on Animals; CMC; carboxymethylcellulose; DMEM; Dulbecco's minimum essential media; DMSO; dimethyl sulfoxide;
Coupling ultra-high-pressure liquid chromatography with mass spectrometry for in-vitro drug-metabolism studies
Keywords: موجودی شیمیایی جدید; ADC; Analog-to-digital converter; ADMET; Absorption, distribution, metabolism, excretion and toxicity; APCI; Atmospheric pressure chemical ionization; CYP; Cytochrome P450; DDI; Drug-drug interaction; DMPK; Drug metabolism and pharmacokinetics; DT; Dwell
The development and registration of topical pharmaceuticals
Keywords: موجودی شیمیایی جدید; Formulation; Topical; Regulatory routes; New Chemical Entity; Active Pharmaceutical Ingredient
Discovery of novel A3 adenosine receptor ligands based on chromone scaffold
Keywords: موجودی شیمیایی جدید; [3H]CCPA; [3H](2R,3R,4S,5R)-2-[2-chloro-6-(cyclopentylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol; [3H]HEMADO; [3H] 2-(1-Hexynyl)-N6-methyladenosine; [3H]NECA; [3H]adenosine-5â²-(N-ethylcarboxamide); AR; Adenosine receptor; Arg; arginine; Asn; as
A perspective on PSE in pharmaceutical process development and innovation
Keywords: موجودی شیمیایی جدید; ANN; artificial neural network; API; active pharmaceutical ingredient; CAMD; computer-aided molecular design; CFD; computational fluid dynamics; CP; continuous processing; CPM; continuous pharmaceutical manufacturing; CPP; critical process parameter; CQA;
Validation of the 96 well Caco-2 cell culture model for high throughput permeability assessment of discovery compounds
Keywords: موجودی شیمیایی جدید; ADME; absorption, distribution, metabolism, elimination; BCS; biopharmaceutics classification system; BMS; Bristol-Myers Squibb Company; HBSS; Hank's balanced salt solution; HEPES; N-2-hydroxyethylpiperazine-Nâ²-2-ethanesulfonic acid; IAM; immobilized ar
New model for intravenous drug administration and blood sampling in the awake rat, designed to increase quality and throughput for in vivo pharmacokinetic analysis
Keywords: موجودی شیمیایی جدید; ADME; absorption distribution metabolism excretion; AUC; area under the curve; Cl; total plasma clearance; Cmax; maximum plasma concentration; Hct; haematocrit; LC-MS/MS; liquid chromatography coupled to tandem mass spectrometry; NCE; new chemical entity;
A novel high-throughput automated chip-based nanoelectrospray tandem mass spectrometric method for PAMPA sample analysis
Keywords: موجودی شیمیایی جدید; ADME; absorption, distribution, metabolism, elimination; DMSO; di-methyl sulphoxide; IAM; immobilized artificial membrane; LC/MS; liquid chromatography/mass spectrometry; HPLC; high pressure liquid chromatography; MDCK; mardin darby canine kidney cells; N
A combined cell based approach to identify P-glycoprotein substrates and inhibitors in a single assay
Keywords: موجودی شیمیایی جدید; A to B; apical to basolateral; ADME; absorption, distribution, metabolism, elimination; B to A; basolateral to apical; BCRP; breast cancer resistance protein; HBSS; Hank's balanced salt solution; HEPES; N-2-hydroxyethylpiperazine-Nâ²-2-ethanesulfonic aci
Lignans, bacteriocides and organochlorine compounds activate the human pregnane X receptor (PXR)
Keywords: موجودی شیمیایی جدید; AR; androgen receptor; β-Gal; β-galactosidase; CYP3A; cytochrome P4503A; DMEM; Dulbecco's modified Eagle medium; DMSO; dimethyl sulfoxide; DR3; direct repeat with 3 nucleotide spacer; EC50; effective concentration for half-maximal response; ER; estrogen