
Trivalent, Gal/GalNAc-containing ligands designed for the asialoglycoprotein receptor
Keywords: NIS, N-iodosuccinimide; TfOH, trifluoromethanesulfonic acid; NHS, N-hydroxysuccinimide; PyBOP, benzotriazol-1-yl-oxytripyrrolidino-phosphonium hexafluorophosphate; Tris, 2-amino-2-(hydroxymethyl)-1,3-propanediol; EEDQ, ethyl 1,2-dihydro-2-ethoxy-1-quinoli