
Synthesis and in vitro biological evaluation of 2,6,9-trisubstituted purines targeting multiple cyclin-dependent kinases
Keywords: Cyclin-dependent kinase; Inhibitor; Roscovitine; Cancer; Apoptosis; Cell cycleCDK, cyclin-dependent kinase; DIAD, diisopropyldiazadicarboxylate; NMP, N-methylpyrrolidone; PARP, poly(ADP-ribose)polymerase; TLC, thin layer chromatography