Pyrazolo[1,5-a]pyrimidine TRPC6 antagonists for the treatment of gastric cancer
Keywords: کانتین های غیر کیهانی; Nonselective cation channels; TRPC channels; Ca2+ signaling; Anticancer; Drug discovery; [Ca2+]i; Intracellular Ca2+ concentration; CCh; Carbachol; EC50; Half maximal stimulation; FMP; FLIPR membrane potential; PLC; phospholipase C; SAR; Structure-activit