
A mass balance approach for calculation of recovery and binding enables the use of ultrafiltration as a rapid method for measurement of plasma protein binding for even highly lipophilic compounds
Keywords: ADME, absorption, distribution, metabolism, excretion; ED, equilibrium dialysis; EP, eppendorf; NSB, non-specific binding; PD, pharmacodynamics; PK, pharmacokinetics; PPB, plasma protein binding; RED, rapid equilibrium dialysis; UF, ultrafiltrationPlasma